SG11201707122QA - Pharmaceutical formulations of bruton's tyrosine kinase inhibtor - Google Patents

Pharmaceutical formulations of bruton's tyrosine kinase inhibtor

Info

Publication number
SG11201707122QA
SG11201707122QA SG11201707122QA SG11201707122QA SG11201707122QA SG 11201707122Q A SG11201707122Q A SG 11201707122QA SG 11201707122Q A SG11201707122Q A SG 11201707122QA SG 11201707122Q A SG11201707122Q A SG 11201707122QA SG 11201707122Q A SG11201707122Q A SG 11201707122QA
Authority
SG
Singapore
Prior art keywords
bruton
tyrosine kinase
pharmaceutical formulations
inhibtor
kinase inhibtor
Prior art date
Application number
SG11201707122QA
Inventor
Harisha Atluri
Ching Wah Chong
Robert Kuehl
Heow Tan
Original Assignee
Pharmacyclics Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=56848552&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG11201707122Q(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacyclics Llc filed Critical Pharmacyclics Llc
Publication of SG11201707122QA publication Critical patent/SG11201707122QA/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
SG11201707122QA 2015-03-03 2016-03-02 Pharmaceutical formulations of bruton's tyrosine kinase inhibtor SG11201707122QA (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562127717P 2015-03-03 2015-03-03
US201562193518P 2015-07-16 2015-07-16
PCT/US2016/020467 WO2016141068A1 (en) 2015-03-03 2016-03-02 Pharmaceutical formulations of bruton's tyrosine kinase inhibtor

Publications (1)

Publication Number Publication Date
SG11201707122QA true SG11201707122QA (en) 2017-09-28

Family

ID=56848552

Family Applications (2)

Application Number Title Priority Date Filing Date
SG10202102078VA SG10202102078VA (en) 2015-03-03 2016-03-02 Pharmaceutical formulations of a bruton’s tyrosine kinase inhibitor
SG11201707122QA SG11201707122QA (en) 2015-03-03 2016-03-02 Pharmaceutical formulations of bruton's tyrosine kinase inhibtor

Family Applications Before (1)

Application Number Title Priority Date Filing Date
SG10202102078VA SG10202102078VA (en) 2015-03-03 2016-03-02 Pharmaceutical formulations of a bruton’s tyrosine kinase inhibitor

Country Status (22)

Country Link
US (8) US9655857B2 (en)
EP (2) EP3265084B1 (en)
JP (2) JP7149076B2 (en)
KR (1) KR20170122220A (en)
CN (1) CN107427498A (en)
AU (3) AU2016226279B2 (en)
BR (2) BR122023020985A2 (en)
CA (3) CA3177990A1 (en)
DK (1) DK3265084T3 (en)
FI (1) FI3265084T3 (en)
HK (1) HK1249015A1 (en)
IL (2) IL293284A (en)
LT (1) LT3265084T (en)
MX (5) MX2017011270A (en)
NZ (1) NZ734446A (en)
PT (1) PT3265084T (en)
RS (1) RS65234B1 (en)
RU (1) RU2017133990A (en)
SG (2) SG10202102078VA (en)
TW (4) TWI733027B (en)
WO (1) WO2016141068A1 (en)
ZA (1) ZA201907661B (en)

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NZ702548A (en) 2012-06-04 2015-11-27 Pharmacyclics Llc Crystalline forms of a bruton’s tyrosine kinase inhibitor
JP6575950B2 (en) 2012-07-24 2019-09-18 ファーマサイクリックス エルエルシー Mutations with resistance to Bruton tyrosine kinase (Btk) inhibitors
US9795604B2 (en) 2013-10-25 2017-10-24 Pharmacyclics Llc Methods of treating and preventing graft versus host disease
CA3210338A1 (en) * 2013-12-02 2015-06-11 Pharmacyclics Llc Methods of treating and preventing alloantibody driven chronic graft versus host disease
JP2017523206A (en) * 2014-08-07 2017-08-17 ファーマサイクリックス エルエルシー New formulation of breton-type tyrosine kinase inhibitor
BR122023020985A2 (en) 2015-03-03 2023-12-26 Pharmacyclics Llc SOLID TABLET FORMULATION OF A BRUTON'S TYROSINE KINASE INHIBITOR
EP3270976A4 (en) 2015-03-20 2019-02-27 The Trustees of the University of Pennsylvania Vaccines with cd40 ligand as an adjuvant
MA41901A (en) * 2015-04-06 2021-04-14 Janssen Pharmaceutica Nv COMPOSITIONS CONTAINING IBRUTINIB
AU2017208472B2 (en) * 2016-01-19 2022-09-01 Janssen Pharmaceutica Nv Formulations/compositions comprising a BTK inhibitor
CN108653231A (en) * 2017-04-01 2018-10-16 北京赛林泰医药技术有限公司 Composition and preparation method thereof containing bruton's tyrosine kinase inhibitor
US11730725B2 (en) 2017-09-26 2023-08-22 Tesaro, Inc. Niraparib formulations
CZ2017787A3 (en) * 2017-12-08 2019-06-19 Zentiva, K.S. Pharmaceutical compositions containing ibrutinib
CA3089537A1 (en) 2018-01-20 2019-07-25 Natco Pharma Limited Pharmaceutical compositions comprising ibrutinib
CA3098497A1 (en) 2018-05-03 2019-11-07 Juno Therapeutics, Inc. Combination therapy of a chimeric antigen receptor (car) t cell therapy and a kinase inhibitor
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US10688050B1 (en) 2018-12-21 2020-06-23 Synthon B.V. Pharmaceutical composition comprising ibrutinib
US20210228479A1 (en) * 2020-01-29 2021-07-29 Farmakeio Nutraceuticals Llc Steroidal compositions and method of making and use
US11433072B1 (en) 2021-06-10 2022-09-06 Hikma Pharmaceuticals USA, Inc. Oral dosage forms of ibrutinib
WO2022260667A1 (en) * 2021-06-10 2022-12-15 Hikma Pharmaceuticals Usa Inc. Oral dosage forms of ibrutinib
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