HK1102422A1 - Combinations comprising dipeptidylpeptidase-iv inhibitors and antidiabetic agents - Google Patents

Combinations comprising dipeptidylpeptidase-iv inhibitors and antidiabetic agents

Info

Publication number
HK1102422A1
HK1102422A1 HK07106890.1A HK07106890A HK1102422A1 HK 1102422 A1 HK1102422 A1 HK 1102422A1 HK 07106890 A HK07106890 A HK 07106890A HK 1102422 A1 HK1102422 A1 HK 1102422A1
Authority
HK
Hong Kong
Prior art keywords
inhibitors
insulin
glucose
fructose
nvp
Prior art date
Application number
HK07106890.1A
Other languages
English (en)
Inventor
Boerk Balkan
Thomas Edward Hughes
David Grenville Holmes
Edwin Bernard Villhauer
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27049636&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1102422(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of HK1102422A1 publication Critical patent/HK1102422A1/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4025—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
HK07106890.1A 2000-01-21 2007-06-27 Combinations comprising dipeptidylpeptidase-iv inhibitors and antidiabetic agents HK1102422A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US48923400A 2000-01-21 2000-01-21
US61926200A 2000-07-19 2000-07-19

Publications (1)

Publication Number Publication Date
HK1102422A1 true HK1102422A1 (en) 2007-11-23

Family

ID=27049636

Family Applications (4)

Application Number Title Priority Date Filing Date
HK07106890.1A HK1102422A1 (en) 2000-01-21 2007-06-27 Combinations comprising dipeptidylpeptidase-iv inhibitors and antidiabetic agents
HK07106895A HK1102405A1 (en) 2000-01-21 2007-06-27 Combinations comprising dipeptidypeptidase-iv inhibitors and antidiabetic agents
HK07106894.7A HK1102424A1 (en) 2000-01-21 2007-06-27 Combinations comprising dipeptidylpeptidase-iv inhibitors and antidiabetic agents
HK07107617.1A HK1108359A1 (en) 2000-01-21 2007-07-16 Combinations comprising dipeptidylpeptidase-iv inhibitors and antidiabetic agents -iv

Family Applications After (3)

Application Number Title Priority Date Filing Date
HK07106895A HK1102405A1 (en) 2000-01-21 2007-06-27 Combinations comprising dipeptidypeptidase-iv inhibitors and antidiabetic agents
HK07106894.7A HK1102424A1 (en) 2000-01-21 2007-06-27 Combinations comprising dipeptidylpeptidase-iv inhibitors and antidiabetic agents
HK07107617.1A HK1108359A1 (en) 2000-01-21 2007-07-16 Combinations comprising dipeptidylpeptidase-iv inhibitors and antidiabetic agents -iv

Country Status (18)

Country Link
US (1) US20030139434A1 (xx)
EP (5) EP1741445B1 (xx)
JP (7) JP2003520226A (xx)
CN (3) CN1400908A (xx)
AT (2) ATE346613T1 (xx)
AU (1) AU2001237321A1 (xx)
BR (1) BRPI0107715B8 (xx)
CA (2) CA2673615C (xx)
CY (6) CY1106303T1 (xx)
DE (3) DE60132723T2 (xx)
DK (5) DK1741446T3 (xx)
ES (5) ES2275654T5 (xx)
FR (1) FR08C0017I2 (xx)
HK (4) HK1102422A1 (xx)
LU (1) LU91436I2 (xx)
NL (1) NL300346I1 (xx)
PT (5) PT1248604E (xx)
WO (1) WO2001052825A2 (xx)

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ATE385421T1 (de) 2008-02-15
US20030139434A1 (en) 2003-07-24
CY1114466T1 (el) 2016-10-05
PT1741445E (pt) 2013-11-11
PT1743655E (pt) 2014-09-09
ES2275654T3 (es) 2007-06-16
CA2673615A1 (en) 2001-07-26
EP1741446B1 (en) 2008-02-06
WO2001052825A3 (en) 2002-03-28
CY1107423T1 (el) 2010-07-28
HK1102424A1 (en) 2007-11-23
EP1741445B1 (en) 2013-08-14
BRPI0107715B1 (pt) 2016-07-05
EP1741446A3 (en) 2007-01-17
JP2011116772A (ja) 2011-06-16
CY2008010I1 (el) 2009-11-04
JP5835910B2 (ja) 2015-12-24
WO2001052825A2 (en) 2001-07-26
ES2301142T3 (es) 2008-06-16
DE60132723D1 (de) 2008-03-20
HK1108359A1 (en) 2008-05-09
EP1248604B1 (en) 2006-11-29
DK1741445T3 (da) 2013-11-04
JP2011162550A (ja) 2011-08-25
FR08C0017I2 (fr) 2010-12-31
NL300346I1 (xx) 2008-07-01
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DE122008000018I1 (de) 2008-08-14
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CN1977842A (zh) 2007-06-13
CY2008010I2 (el) 2009-11-04
CA2397554A1 (en) 2001-07-26
JP6104331B2 (ja) 2017-03-29
DE60124861D1 (de) 2007-01-11
ATE346613T1 (de) 2006-12-15
EP1741446A2 (en) 2007-01-10
BR0107715A (pt) 2002-11-19
EP1248604B2 (en) 2012-02-29
DK1248604T4 (da) 2012-05-21
EP1741447A3 (en) 2007-01-17
DK1743655T3 (da) 2014-08-18
PT1248604E (pt) 2007-01-31
JP2015214572A (ja) 2015-12-03
DK1248604T3 (da) 2007-02-19
EP1741445A2 (en) 2007-01-10
EP1741445A3 (en) 2007-01-24
PT1741447E (pt) 2013-12-11
JP6374995B2 (ja) 2018-08-15
HK1102405A1 (en) 2007-11-23
BRPI0107715B8 (pt) 2021-05-25
CN1400908A (zh) 2003-03-05
CY1106303T1 (el) 2011-10-12
DE60132723T2 (de) 2009-01-29
AU2001237321A1 (en) 2001-07-31
ES2275654T5 (es) 2012-06-07
CA2673615C (en) 2013-07-16
JP2003520226A (ja) 2003-07-02
CA2397554C (en) 2009-09-22
ES2487897T3 (es) 2014-08-25
ES2433476T3 (es) 2013-12-11
JP5824224B2 (ja) 2015-11-25
CY1114593T1 (el) 2016-10-05
JP6095589B2 (ja) 2017-03-15

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