GT199200028A - Derivados de quinuclidina - Google Patents

Derivados de quinuclidina

Info

Publication number
GT199200028A
GT199200028A GT199200028A GT199200028A GT199200028A GT 199200028 A GT199200028 A GT 199200028A GT 199200028 A GT199200028 A GT 199200028A GT 199200028 A GT199200028 A GT 199200028A GT 199200028 A GT199200028 A GT 199200028A
Authority
GT
Guatemala
Prior art keywords
compounds
quinuclidine derivatives
disorders
antagonists
mind
Prior art date
Application number
GT199200028A
Other languages
English (en)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=24845673&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=GT199200028(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of GT199200028A publication Critical patent/GT199200028A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Psychiatry (AREA)
  • Rheumatology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

SE REFIERE A NUEVOS DERIVADOS DE QUINUCLIDINA, A COMPOSICIONES FARMACEUTICAS QUE CONTIENEN ESTOS COMPUESTOS Y AL USO DEESTOS COMPUESTOS EN EL TRATAMIENTO DE LOS TRASTORNOS GASTROINTESTINALES, TRASTORNOS INFLAMATORIOS, TRASTORNOS DEL SISTEMA NERVIOSO CENTRAL Y DOLOR. ESTOS COMPUESTOS SON ANTAGONISTAS DE LA SUSTANCIA P Y TIENEN LA ESTRUCTURA QUIMICA CONTENIDA EN LA FICHA TECNICA RESPECTIVA Y LAS SALES FARMACEUTICA MENTE ACEPTABLES DE DICHOS COMPUESTOS.
GT199200028A 1991-05-31 1992-05-29 Derivados de quinuclidina GT199200028A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US70840491A 1991-05-31 1991-05-31

Publications (1)

Publication Number Publication Date
GT199200028A true GT199200028A (es) 1993-11-20

Family

ID=24845673

Family Applications (1)

Application Number Title Priority Date Filing Date
GT199200028A GT199200028A (es) 1991-05-31 1992-05-29 Derivados de quinuclidina

Country Status (41)

Country Link
US (3) US5807867A (es)
EP (1) EP0587723B1 (es)
JP (2) JPH0733386B2 (es)
KR (1) KR100214905B1 (es)
CN (1) CN1048492C (es)
AP (1) AP299A (es)
AT (1) ATE135006T1 (es)
AU (1) AU657552B2 (es)
BG (1) BG61694B1 (es)
BR (1) BR9206073A (es)
CA (1) CA2102179C (es)
CZ (1) CZ281403B6 (es)
DE (4) DE122006000066I1 (es)
DK (1) DK0587723T3 (es)
EG (1) EG19944A (es)
ES (1) ES2084361T3 (es)
FI (1) FI114475B (es)
GR (1) GR3019687T3 (es)
GT (1) GT199200028A (es)
HU (1) HU217548B (es)
IE (1) IE72473B1 (es)
IL (1) IL102008A (es)
IS (1) IS1611B (es)
LU (1) LU91293I2 (es)
MA (1) MA22539A1 (es)
MX (1) MX9202554A (es)
NL (1) NL300250I2 (es)
NO (2) NO302701B1 (es)
NZ (2) NZ270673A (es)
OA (1) OA09867A (es)
PL (1) PL171379B1 (es)
PT (1) PT100546B (es)
RO (1) RO110499B1 (es)
RU (1) RU2103269C1 (es)
SK (1) SK390692A3 (es)
TW (1) TW204349B (es)
UA (1) UA27776C2 (es)
UY (1) UY23422A1 (es)
WO (1) WO1992021677A1 (es)
YU (1) YU48995B (es)
ZA (1) ZA923942B (es)

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IL109646A0 (en) * 1993-05-19 1994-08-26 Pfizer Heteroatom substituted alkyl benzylamino-quinuclidines
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TW458774B (en) 1995-10-20 2001-10-11 Pfizer Antiemetic pharmaceutical compositions
IL123740A0 (en) * 1997-03-28 1998-10-30 Pfizer NK-1 receptor antagonists for the treatment of delayed emesis
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Also Published As

Publication number Publication date
JPH07285965A (ja) 1995-10-31
US6222038B1 (en) 2001-04-24
YU48995B (sh) 2003-04-30
FI114475B (fi) 2004-10-29
UY23422A1 (es) 1992-11-12
KR100214905B1 (ko) 1999-08-02
CN1048492C (zh) 2000-01-19
FI935297A (fi) 1993-11-29
PT100546B (pt) 1999-12-31
IS1611B (is) 1996-10-18
NL300250I2 (nl) 2007-03-01
NO934312L (no) 1993-11-29
NO302701B1 (no) 1998-04-14
JPH0733386B2 (ja) 1995-04-12
SK278788B6 (sk) 1998-02-04
TW204349B (es) 1993-04-21
PT100546A (pt) 1993-08-31
HU217548B (hu) 2000-02-28
US5939433A (en) 1999-08-17
ES2084361T3 (es) 1996-05-01
CA2102179A1 (en) 1992-12-01
DE122006000066I2 (de) 2007-12-06
IL102008A0 (en) 1992-12-30
MX9202554A (es) 1992-11-01
BG98248A (bg) 1994-07-29
DE69208877T2 (de) 1996-07-25
DE69208877D1 (de) 1996-04-11
IL102008A (en) 1995-12-08
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OA09867A (en) 1994-08-15
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IS3871A (is) 1992-12-02
AP299A (en) 1994-01-14
US5807867A (en) 1998-09-15
NO2007003I1 (no) 2007-03-26
UA27776C2 (uk) 2000-10-16
GR3019687T3 (en) 1996-07-31
EG19944A (en) 1997-02-27
HUT70151A (en) 1995-09-28
EP0587723B1 (en) 1996-03-06
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NO2007003I2 (no) 2011-04-18
RO110499B1 (ro) 1996-01-30
DE122006000066I1 (de) 2007-03-22
YU56492A (sh) 1995-03-27
CZ281403B6 (cs) 1996-09-11
AU1990192A (en) 1993-01-08
NZ270673A (en) 1997-07-27
NL300250I1 (nl) 2007-02-01
SK390692A3 (en) 1998-02-04
NO934312D0 (no) 1993-11-29
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IE72473B1 (en) 1997-04-23
IE921729A1 (en) 1992-12-02
BG61694B1 (bg) 1998-03-31
BR9206073A (pt) 1994-12-06
NZ242956A (en) 1995-06-27
RU2103269C1 (ru) 1998-01-27
CN1067428A (zh) 1992-12-30
MA22539A1 (fr) 1992-12-31
HU9303393D0 (en) 1994-03-28
AU657552B2 (en) 1995-03-16
ATE135006T1 (de) 1996-03-15
EP0587723A1 (en) 1994-03-23
WO1992021677A1 (en) 1992-12-10
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PL171379B1 (en) 1997-04-30

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