DK1660458T3 - 2, 4-pyrimidindiaminer egnede i behandling af neoplastiske sygdomme, in-flammatoriske lidelser og lidelser i immunsystemet. - Google Patents

2, 4-pyrimidindiaminer egnede i behandling af neoplastiske sygdomme, in-flammatoriske lidelser og lidelser i immunsystemet.

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Publication number
DK1660458T3
DK1660458T3 DK04764093.3T DK04764093T DK1660458T3 DK 1660458 T3 DK1660458 T3 DK 1660458T3 DK 04764093 T DK04764093 T DK 04764093T DK 1660458 T3 DK1660458 T3 DK 1660458T3
Authority
DK
Denmark
Prior art keywords
disorders
treatment
immune system
neoplastic diseases
diamines useful
Prior art date
Application number
DK04764093.3T
Other languages
English (en)
Inventor
Carlos Garcia-Echeverria
Takanori Kanazawa
Eiji Kawahara
Keiichi Masuya
Naoko Matsuura
Takahiro Miyake
Osamu Ohmori
Ichiro Umemura
Ruo Steensma
Greg Chopiuk
Jiqing Jiang
Yongqin Wan
Qiang Ding
Qiong Zhang
Nathanael Schiander Gray
Donald Karanewsky
Original Assignee
Irm Llc
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34196260&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK1660458(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GB0319227A external-priority patent/GB0319227D0/en
Priority claimed from GB0322370A external-priority patent/GB0322370D0/en
Application filed by Irm Llc, Novartis Ag filed Critical Irm Llc
Application granted granted Critical
Publication of DK1660458T3 publication Critical patent/DK1660458T3/da

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
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    • C04B35/63—Preparing or treating the powders individually or as batches ; preparing or treating macroscopic reinforcing agents for ceramic products, e.g. fibres; mechanical aspects section B using additives specially adapted for forming the products, e.g.. binder binders
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
DK04764093.3T 2003-08-15 2004-08-13 2, 4-pyrimidindiaminer egnede i behandling af neoplastiske sygdomme, in-flammatoriske lidelser og lidelser i immunsystemet. DK1660458T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0319227A GB0319227D0 (en) 2003-08-15 2003-08-15 Organic compounds
GB0322370A GB0322370D0 (en) 2003-09-24 2003-09-24 Organic compounds
PCT/EP2004/009099 WO2005016894A1 (en) 2003-08-15 2004-08-13 2, 4-pyrimidinediamines useful in the treatment of neoplastic diseases, inflammatory and immune system disorders

Publications (1)

Publication Number Publication Date
DK1660458T3 true DK1660458T3 (da) 2012-05-07

Family

ID=34196260

Family Applications (2)

Application Number Title Priority Date Filing Date
DK10010291.2T DK2287156T3 (da) 2003-08-15 2004-08-13 2,4-Di(phenylamino)-pyrimidiner egnede i behandling af neoplastiske sygdomme, inflammatoriske lidelser og lidelser i immunsystemet
DK04764093.3T DK1660458T3 (da) 2003-08-15 2004-08-13 2, 4-pyrimidindiaminer egnede i behandling af neoplastiske sygdomme, in-flammatoriske lidelser og lidelser i immunsystemet.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DK10010291.2T DK2287156T3 (da) 2003-08-15 2004-08-13 2,4-Di(phenylamino)-pyrimidiner egnede i behandling af neoplastiske sygdomme, inflammatoriske lidelser og lidelser i immunsystemet

Country Status (32)

Country Link
US (2) US7893074B2 (da)
EP (2) EP1660458B1 (da)
JP (2) JP4607879B2 (da)
KR (1) KR100904570B1 (da)
AR (1) AR045458A1 (da)
AT (1) ATE542801T1 (da)
AU (2) AU2004264382A1 (da)
BR (2) BR122019017579B8 (da)
CA (1) CA2533320A1 (da)
CO (1) CO5680434A2 (da)
CY (2) CY1112571T1 (da)
DK (2) DK2287156T3 (da)
EC (1) ECSP066371A (da)
ES (2) ES2380206T3 (da)
HK (1) HK1091813A1 (da)
HR (2) HRP20120335T1 (da)
IL (1) IL173129A0 (da)
IS (1) IS2873B (da)
MA (1) MA27994A1 (da)
MX (1) MXPA06001759A (da)
MY (1) MY147449A (da)
NO (1) NO333306B1 (da)
NZ (1) NZ585188A (da)
PL (2) PL2287156T3 (da)
PT (2) PT1660458E (da)
RU (1) RU2395500C2 (da)
SG (1) SG145749A1 (da)
SI (2) SI2287156T1 (da)
TN (1) TNSN06052A1 (da)
TW (1) TWI378923B (da)
WO (1) WO2005016894A1 (da)
ZA (1) ZA200600464B (da)

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