DK1307457T3 - Azabicycliske forbindelser, deres fremstilling og deres anvendelse som medikamenter, især som antibakterielle midler - Google Patents
Azabicycliske forbindelser, deres fremstilling og deres anvendelse som medikamenter, især som antibakterielle midlerInfo
- Publication number
- DK1307457T3 DK1307457T3 DK01958173T DK01958173T DK1307457T3 DK 1307457 T3 DK1307457 T3 DK 1307457T3 DK 01958173 T DK01958173 T DK 01958173T DK 01958173 T DK01958173 T DK 01958173T DK 1307457 T3 DK1307457 T3 DK 1307457T3
- Authority
- DK
- Denmark
- Prior art keywords
- drugs
- preparation
- antibacterial agents
- azabicyclic compounds
- azabicyclic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/08—Bridged systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/08—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pulmonology (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0010121A FR2812635B1 (fr) | 2000-08-01 | 2000-08-01 | Nouveaux composes heterocycliques, preparation et utilisation comme medicaments notamment comme anti- bacteriens |
PCT/FR2001/002418 WO2002010172A1 (fr) | 2000-08-01 | 2001-07-24 | Composes azabicycliques, leur preparation et leur utilisation comme medicaments, notamment comme anti-bacteriens |
Publications (1)
Publication Number | Publication Date |
---|---|
DK1307457T3 true DK1307457T3 (da) | 2004-08-09 |
Family
ID=8853181
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK01958173T DK1307457T3 (da) | 2000-08-01 | 2001-07-24 | Azabicycliske forbindelser, deres fremstilling og deres anvendelse som medikamenter, især som antibakterielle midler |
Country Status (42)
Country | Link |
---|---|
US (5) | US7112592B2 (da) |
EP (1) | EP1307457B1 (da) |
JP (2) | JP4515704B2 (da) |
KR (1) | KR100632906B1 (da) |
CN (1) | CN1289500C (da) |
AP (1) | AP1614A (da) |
AR (1) | AR031716A1 (da) |
AT (1) | ATE263768T1 (da) |
AU (2) | AU7990501A (da) |
BG (1) | BG66094B1 (da) |
BR (1) | BRPI0112986B8 (da) |
CA (1) | CA2417475C (da) |
CR (1) | CR6895A (da) |
CZ (1) | CZ294956B6 (da) |
DE (1) | DE60102702T2 (da) |
DK (1) | DK1307457T3 (da) |
DZ (1) | DZ3397A1 (da) |
EA (1) | EA004920B1 (da) |
EC (1) | ECSP034460A (da) |
EE (1) | EE05183B1 (da) |
ES (1) | ES2220793T3 (da) |
FR (1) | FR2812635B1 (da) |
HK (1) | HK1060356A1 (da) |
HR (1) | HRP20030034B1 (da) |
HU (1) | HU226889B1 (da) |
IL (2) | IL154187A0 (da) |
MA (1) | MA26938A1 (da) |
ME (2) | ME00060B (da) |
MX (1) | MXPA03000881A (da) |
NO (1) | NO324940B1 (da) |
NZ (1) | NZ523707A (da) |
OA (1) | OA12347A (da) |
PL (2) | PL216028B1 (da) |
PT (1) | PT1307457E (da) |
RS (1) | RS50214B (da) |
SI (1) | SI1307457T1 (da) |
SK (1) | SK287597B6 (da) |
TR (1) | TR200400859T4 (da) |
TW (1) | TWI292401B (da) |
UA (1) | UA73791C2 (da) |
WO (1) | WO2002010172A1 (da) |
ZA (1) | ZA200300676B (da) |
Families Citing this family (95)
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FR2812635B1 (fr) * | 2000-08-01 | 2002-10-11 | Aventis Pharma Sa | Nouveaux composes heterocycliques, preparation et utilisation comme medicaments notamment comme anti- bacteriens |
FR2835186B1 (fr) | 2002-01-28 | 2006-10-20 | Aventis Pharma Sa | Nouveaux composes heterocycliques, actifs comme inhibiteurs de beta-lactamases |
FR2844273B1 (fr) * | 2002-09-05 | 2008-04-04 | Aventis Pharma Sa | Nouveaux composes heterocycliques, procede et intermediaires de preparation et utilisation comme medicament, notamment comme inhibiteurs de beta-lactamases et anti-bacteriens. |
US7439253B2 (en) * | 2002-12-06 | 2008-10-21 | Novexel | Heterocyclic compounds, their preparation and their use as medicaments, in particular as antibacterials and beta-lactamase inhibitors |
FR2848210B1 (fr) * | 2002-12-06 | 2007-10-19 | Aventis Pharma Sa | Nouveaux composes heterocycliques, leur preparation et leur utilisation comme medicaments, notamment comme anti-bacteriens et inhibiteurs de beta-lactamases |
CN103724330B (zh) | 2005-12-07 | 2015-08-19 | 巴斯利尔药物股份公司 | 单环-内酰胺类抗生素与β-内酰胺酶抑制剂的有效的联合应用 |
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MX2009004290A (es) * | 2006-10-23 | 2009-07-27 | Irm Llc | Inhibidores de proteasas de catepsina. |
JPWO2008093737A1 (ja) | 2007-01-31 | 2010-05-20 | 大日本住友製薬株式会社 | アミド誘導体 |
FR2914923B1 (fr) * | 2007-04-12 | 2013-06-14 | Novexel | Nouveaux composes heterocycliques azotes,leur preparation et leur utilisation comme medicaments antibacteriens. |
WO2008150470A1 (en) | 2007-05-31 | 2008-12-11 | Shionogi & Co., Ltd. | Oxyimino compounds and the use thereof |
FR2921060B1 (fr) * | 2007-09-14 | 2012-06-15 | Novexel | Nouveau procede de preparation d'une piperidine disubsituee et nouveaux intermediaires |
PL2666774T3 (pl) * | 2008-01-18 | 2015-06-30 | Merck Sharp & Dohme | Inhibitory beta-laktamazy |
US8518934B2 (en) | 2008-06-11 | 2013-08-27 | Shonogi & Co., Ltd. | Oxycarbamoyl compounds and the use thereof |
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FR2936798B1 (fr) | 2008-10-03 | 2012-09-28 | Novexel | Nouveaux composes heterocycliques azotes, leur preparation et leur utilisation comme medicaments antibacteriens. |
FR2937034B1 (fr) | 2008-10-10 | 2012-11-23 | Novexel | Nouveaux composes heterocycliques azotes, leur preparation et leur utilisation comme medicaments antibacteriens |
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CN110078728B (zh) * | 2019-05-23 | 2020-10-23 | 江西富祥药业股份有限公司 | 一种阿维巴坦中间体、制备方法及其应用 |
WO2021106864A1 (en) * | 2019-11-25 | 2021-06-03 | Eisai R&D Management Co., Ltd. | Process for the preparation of producing pyrazolo[1,5-a] pyrimidine derivatives |
US11814385B2 (en) | 2021-06-25 | 2023-11-14 | University Of South Florida | Small molecule inhibitors targeting Clostridioides difficile sporulation |
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JPS4939678B1 (da) * | 1968-05-06 | 1974-10-28 | ||
US4024147A (en) * | 1972-06-30 | 1977-05-17 | John Wyeth & Brother Limited | Heterocyclic compounds |
US4049821A (en) * | 1976-05-12 | 1977-09-20 | A. H. Robins Company, Inc. | Method of treating allergy |
EP0260057A3 (en) * | 1986-09-02 | 1989-02-01 | The University Of Melbourne | 2-oxo-4-carboxy-pyrimidines |
JPS63119471A (ja) * | 1986-09-02 | 1988-05-24 | ザ・ユニバーシテイ・オブ・メルボルン | 2−オキソ−4−カルボキシ−ピリミジン |
JP2895630B2 (ja) * | 1993-12-29 | 1999-05-24 | フアイザー・インコーポレイテツド | ジアザビシクロニューロキニンアンタゴニスト |
TW358097B (en) * | 1996-05-24 | 1999-05-11 | Hoffmann La Roche | Beta-lactams and their process and pharmaceutical compositions |
HUP0001741A3 (en) * | 1996-08-02 | 2000-11-28 | Smithkline Beecham Plc | Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use, process for preparing them, pharmaceuticals contg. them and their use |
ATE271544T1 (de) * | 1997-02-10 | 2004-08-15 | Pfizer Prod Inc | 2-amino-6-(2-substituierte-4-phenoxy)- substituierte-pyridine |
US6060585A (en) * | 1997-03-04 | 2000-05-09 | Wisconsin Alumni Research Foundation | β-polypeptide foldamers of well-defined secondary structure |
KR100207096B1 (ko) * | 1997-07-08 | 1999-07-15 | 이명환 | 시사프라이드의 제조 방법 |
KR20010042851A (ko) * | 1998-04-20 | 2001-05-25 | 후지야마 아키라 | cGMP 포스포디에스터라제 억제자로서의 안트라닐산유도체 |
GB9817029D0 (en) * | 1998-08-05 | 1998-09-30 | Smithkline Beecham Plc | Novel compounds |
FR2784682B1 (fr) * | 1998-10-15 | 2002-12-06 | Hoechst Marion Roussel Inc | Nouveaux derives 2-halogene de 5-0-desosaminylerythronolide a, leur procede de preparation et leur application comme medicaments |
US6635657B1 (en) * | 1998-12-23 | 2003-10-21 | Eli Lilly And Company | Aromatic amides |
IL144096A0 (en) * | 1999-01-02 | 2002-05-23 | Aventis Pharma Gmbh | Novel malonic acid derivatives, processes for their preparation, their use and pharmaceutical compositions containing them (inhibition of factor xa activity) |
FR2812635B1 (fr) * | 2000-08-01 | 2002-10-11 | Aventis Pharma Sa | Nouveaux composes heterocycliques, preparation et utilisation comme medicaments notamment comme anti- bacteriens |
FR2835186B1 (fr) * | 2002-01-28 | 2006-10-20 | Aventis Pharma Sa | Nouveaux composes heterocycliques, actifs comme inhibiteurs de beta-lactamases |
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