MX2016004509A - Compuestos que contienen nitrogeno y su uso. - Google Patents

Compuestos que contienen nitrogeno y su uso.

Info

Publication number
MX2016004509A
MX2016004509A MX2016004509A MX2016004509A MX2016004509A MX 2016004509 A MX2016004509 A MX 2016004509A MX 2016004509 A MX2016004509 A MX 2016004509A MX 2016004509 A MX2016004509 A MX 2016004509A MX 2016004509 A MX2016004509 A MX 2016004509A
Authority
MX
Mexico
Prior art keywords
containing compounds
nitrogen containing
formula
preventing
compound
Prior art date
Application number
MX2016004509A
Other languages
English (en)
Inventor
Bhagwat Sachin
Keshav Deshpande Prasad
Sampatrao Pawar Shivaji
Bhawsar Satish
Vithalbhai Patel Mahesh
Dattatraya Yeole Ravindra
Original Assignee
Wockhardt Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wockhardt Ltd filed Critical Wockhardt Ltd
Publication of MX2016004509A publication Critical patent/MX2016004509A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/439Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • A61K31/546Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine containing further heterocyclic rings, e.g. cephalothin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Abstract

Se describen compuestos de la Fórmula (I), su preparación y uso en evitar o tratar una infección bacteriana. (ver Fórmula).
MX2016004509A 2013-10-11 2014-10-10 Compuestos que contienen nitrogeno y su uso. MX2016004509A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN3216MU2013 IN2013MU03216A (es) 2013-10-11 2014-10-10
PCT/IB2014/065195 WO2015052682A1 (en) 2013-10-11 2014-10-10 Nitrogen containing compounds and their use

Publications (1)

Publication Number Publication Date
MX2016004509A true MX2016004509A (es) 2016-10-28

Family

ID=51945946

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2016004509A MX2016004509A (es) 2013-10-11 2014-10-10 Compuestos que contienen nitrogeno y su uso.

Country Status (10)

Country Link
US (1) US9434728B1 (es)
EP (1) EP3055311B1 (es)
JP (1) JP6411482B2 (es)
CN (1) CN106414444B (es)
AU (1) AU2014333436A1 (es)
CA (1) CA2926773A1 (es)
IN (1) IN2013MU03216A (es)
MX (1) MX2016004509A (es)
RU (1) RU2016113755A (es)
WO (1) WO2015052682A1 (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20160132414A (ko) 2014-03-14 2016-11-18 욱크하르트 리미티드 소듐 (2s, 5r)-6-(벤질옥시)-7-옥소-1,6-다이아자바이사이클로[3.2.1]옥테인-2-카복실레이트의 제조 공정
WO2018053057A2 (en) * 2016-09-19 2018-03-22 Merck Sharp & Dohme Corp. Process for preparing beta-lactamase inhibitor hydroxylurea intermediates
JOP20190061A1 (ar) * 2016-09-28 2019-03-26 Novartis Ag مثبطات بيتا-لاكتاماز
CN111138456A (zh) * 2019-12-27 2020-05-12 山东安弘制药有限公司 一种头霉素中间体化合物的制备方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2812635B1 (fr) 2000-08-01 2002-10-11 Aventis Pharma Sa Nouveaux composes heterocycliques, preparation et utilisation comme medicaments notamment comme anti- bacteriens
EP3260551A1 (en) * 2008-06-19 2017-12-27 Astra Zeneca Holding France Use of (1r,2s,5r) 1,6-diazabicyclo [3.2.1] octane-2-carboxamide, 7-oxo-6-(sulfooxy)-, monosodium salt as a diagnostic reagent for detecting serine beta-lactamases
FR2936798B1 (fr) * 2008-10-03 2012-09-28 Novexel Nouveaux composes heterocycliques azotes, leur preparation et leur utilisation comme medicaments antibacteriens.
FR2936951B1 (fr) 2008-10-10 2010-12-03 Novexel Nouvelles combinaisons de composes heterocycliques azotes antibacteriens avec d'autres composes antibacteriens et leur utilisation comme medicaments
FR2937034B1 (fr) * 2008-10-10 2012-11-23 Novexel Nouveaux composes heterocycliques azotes, leur preparation et leur utilisation comme medicaments antibacteriens
ES2640520T3 (es) * 2011-09-13 2017-11-03 Wockhardt Limited Compuestos que contienen nitrógeno y su uso

Also Published As

Publication number Publication date
CA2926773A1 (en) 2015-04-16
CN106414444B (zh) 2018-02-02
CN106414444A (zh) 2017-02-15
AU2014333436A1 (en) 2016-05-05
JP6411482B2 (ja) 2018-10-24
JP2016532661A (ja) 2016-10-20
IN2013MU03216A (es) 2015-07-03
US9434728B1 (en) 2016-09-06
WO2015052682A1 (en) 2015-04-16
US20160257684A1 (en) 2016-09-08
RU2016113755A3 (es) 2018-06-26
EP3055311B1 (en) 2017-08-09
RU2016113755A (ru) 2017-11-16
EP3055311A1 (en) 2016-08-17

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