AR109356A2 - Sales y polimorfos de 8-fluoro-2-{4-[(metilamino)metil]fenil}-1,3,4,5-tetrahidro-6h-acepino[5,4,3-cd]indol-6-ona - Google Patents

Sales y polimorfos de 8-fluoro-2-{4-[(metilamino)metil]fenil}-1,3,4,5-tetrahidro-6h-acepino[5,4,3-cd]indol-6-ona

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Publication number
AR109356A2
AR109356A2 ARP170102290A ARP170102290A AR109356A2 AR 109356 A2 AR109356 A2 AR 109356A2 AR P170102290 A ARP170102290 A AR P170102290A AR P170102290 A ARP170102290 A AR P170102290A AR 109356 A2 AR109356 A2 AR 109356A2
Authority
AR
Argentina
Prior art keywords
tetrahydro
fluoro
phenyl
methyl
acepino
Prior art date
Application number
ARP170102290A
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English (en)
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43859823&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR109356(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of AR109356A2 publication Critical patent/AR109356A2/es

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06—Peri-condensed systems
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    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
    • C07C309/01—Sulfonic acids
    • C07C309/02—Sulfonic acids having sulfo groups bound to acyclic carbon atoms
    • C07C309/19—Sulfonic acids having sulfo groups bound to acyclic carbon atoms of a saturated carbon skeleton containing rings
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    • C07C57/02—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms with only carbon-to-carbon double bonds as unsaturation
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    • C07C57/145—Maleic acid
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    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Abstract

Reivindicación 1: Una sal camsilato de 8-fluoro-2-{4-[(metilamino)metil]fenil}-1,3,4,5-tetrahidro-6H-azepino[5,4,3-cd]indol-6-ona. Reivindicación 2: La sal de la reivindicación 1, caracterizada porque es la sal es cristalina. Reivindicación 3: La sal de la reivindicación 1, caracterizada porque la sal es una sal cristalina anhidra.
ARP170102290A 2010-02-12 2017-08-16 Sales y polimorfos de 8-fluoro-2-{4-[(metilamino)metil]fenil}-1,3,4,5-tetrahidro-6h-acepino[5,4,3-cd]indol-6-ona AR109356A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US30427710P 2010-02-12 2010-02-12

Publications (1)

Publication Number Publication Date
AR109356A2 true AR109356A2 (es) 2018-11-21

Family

ID=43859823

Family Applications (2)

Application Number Title Priority Date Filing Date
ARP110100427A AR080164A1 (es) 2010-02-12 2011-02-11 Sales y polimorfos de 8-fluoro-2-{4-[(metilamino)metil]fenil}-1,3,4,5-tetrahidro-6h-acepino[5,4,3-cd]indol-6-ona
ARP170102290A AR109356A2 (es) 2010-02-12 2017-08-16 Sales y polimorfos de 8-fluoro-2-{4-[(metilamino)metil]fenil}-1,3,4,5-tetrahidro-6h-acepino[5,4,3-cd]indol-6-ona

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ARP110100427A AR080164A1 (es) 2010-02-12 2011-02-11 Sales y polimorfos de 8-fluoro-2-{4-[(metilamino)metil]fenil}-1,3,4,5-tetrahidro-6h-acepino[5,4,3-cd]indol-6-ona

Country Status (30)

Country Link
US (5) US8754072B2 (es)
EP (4) EP2534153B1 (es)
JP (6) JP5745283B2 (es)
KR (2) KR102108226B1 (es)
CN (2) CN102884066B (es)
AR (2) AR080164A1 (es)
AU (1) AU2011213944B2 (es)
CA (2) CA3024216C (es)
CY (3) CY1118319T1 (es)
DK (2) DK2534153T3 (es)
ES (2) ES2607806T3 (es)
HK (1) HK1176617A1 (es)
HR (2) HRP20161742T1 (es)
HU (3) HUE030969T2 (es)
IL (1) IL220921B (es)
LT (3) LT2534153T (es)
LU (1) LUC00093I2 (es)
MX (1) MX343383B (es)
NL (1) NL300958I2 (es)
NO (1) NO2018039I1 (es)
NZ (1) NZ601445A (es)
PL (2) PL2534153T3 (es)
PT (2) PT3150610T (es)
RS (2) RS59494B1 (es)
RU (1) RU2570198C2 (es)
SG (2) SG182533A1 (es)
SI (2) SI3150610T1 (es)
SM (1) SMT201600462B (es)
TW (1) TWI545123B (es)
WO (1) WO2011098971A1 (es)

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