ZA200804083B - Bi-aryl meta-pyrimidine inhibitors of kinases - Google Patents

Bi-aryl meta-pyrimidine inhibitors of kinases

Info

Publication number
ZA200804083B
ZA200804083B ZA200804083A ZA200804083A ZA200804083B ZA 200804083 B ZA200804083 B ZA 200804083B ZA 200804083 A ZA200804083 A ZA 200804083A ZA 200804083 A ZA200804083 A ZA 200804083A ZA 200804083 B ZA200804083 B ZA 200804083B
Authority
ZA
South Africa
Prior art keywords
kinases
pyrimidine inhibitors
aryl meta
meta
aryl
Prior art date
Application number
ZA200804083A
Other languages
English (en)
Inventor
Cao Jon Jianguo
Hood John
Lohse Dan
Mak Chi Ching
Mcpherson Andrew Noronha Glenn
Pathak Ved
Renick Joel
Richard M Soll
Zeng Binqi
Original Assignee
Targegen Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Targegen Inc filed Critical Targegen Inc
Publication of ZA200804083B publication Critical patent/ZA200804083B/xx

Links

ZA200804083A 2005-11-01 2006-10-26 Bi-aryl meta-pyrimidine inhibitors of kinases ZA200804083B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US73262905P 2005-11-01 2005-11-01

Publications (1)

Publication Number Publication Date
ZA200804083B true ZA200804083B (en) 2009-09-30

Family

ID=40413957

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200804083A ZA200804083B (en) 2005-11-01 2006-10-26 Bi-aryl meta-pyrimidine inhibitors of kinases

Country Status (3)

Country Link
CN (1) CN101370792B (xx)
UA (3) UA109411C2 (xx)
ZA (1) ZA200804083B (xx)

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20120114355A (ko) * 2010-01-13 2012-10-16 글락소스미스클라인 엘엘씨 화합물 및 방법
WO2012060847A1 (en) * 2010-11-07 2012-05-10 Targegen, Inc. Compositions and methods for treating myelofibrosis
CN103242240B (zh) * 2012-02-10 2016-01-06 上海温康化学研发有限公司 一种磺酰胺类化合物的中间体、其盐及其制备方法
CN105796562A (zh) * 2012-09-10 2016-07-27 杨子娇 化合物在制备防治青光眼病的药物中的用途
CN103664798A (zh) * 2012-09-20 2014-03-26 杨育新 一类治疗创伤性脑损伤疾病的化合物及其用途
CN103664799A (zh) * 2012-09-25 2014-03-26 杨子娇 一类治疗房角狭窄的化合物及其用途
CN103664907A (zh) * 2012-09-25 2014-03-26 杨子娇 一类治疗房角狭窄的化合物及其用途
CN103724331A (zh) * 2012-10-11 2014-04-16 韩冰 一类治疗脑性瘫痪的化合物及其用途
EP2970205B1 (en) * 2013-03-14 2019-05-08 Tolero Pharmaceuticals, Inc. Jak2 and alk2 inhibitors and methods for their use
RS57662B1 (sr) * 2013-12-11 2018-11-30 Biogen Ma Inc Biaril jedinjenja korisna za lečenje humanih bolesti u onkologiji, neurologiji i imunologiji
CN103992262B (zh) * 2014-06-12 2015-11-11 苏州明锐医药科技有限公司 塞瑞替尼及其中间体的制备方法
CN106188063A (zh) * 2015-05-08 2016-12-07 中国科学院上海药物研究所 用作Lp-PLA2抑制剂的双环类化合物、其制备方法及医药用途
CN108689949A (zh) * 2018-07-02 2018-10-23 湖南华腾制药有限公司 一种嘧啶类衍生物及其制备方法
CN110305140B (zh) 2019-07-30 2020-08-04 上海勋和医药科技有限公司 二氢吡咯并嘧啶类选择性jak2抑制剂
US20220402948A1 (en) * 2019-09-26 2022-12-22 Betta Pharmaceuticals Co., Ltd. Egfr inhibitor, composition and preparation method therefor
US20240108633A1 (en) * 2020-12-29 2024-04-04 Onquality Pharmaceuticals China Ltd. Method for preventing or treating disease or condition associated with antitumor agent
AU2021416682B2 (en) * 2021-01-11 2024-01-11 Guangzhou Salustier Biosciences Co., Ltd. 2-aminopyrimidine compound and pharmaceutical composition thereof and application thereof
CN112920124B (zh) * 2021-01-29 2024-03-01 安徽医科大学 一种嘧啶-2,4-二胺类化合物及其制备方法与应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0004887D0 (en) * 2000-03-01 2000-04-19 Astrazeneca Uk Ltd Chemical compounds

Also Published As

Publication number Publication date
CN101370792B (zh) 2013-03-20
UA109412C2 (uk) 2015-08-25
CN101370792A (zh) 2009-02-18
UA99899C2 (ru) 2012-10-25
UA109411C2 (uk) 2015-08-25

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