ZA200002263B - Process for the synthesis of nucleoside analogs. - Google Patents

Process for the synthesis of nucleoside analogs.

Info

Publication number
ZA200002263B
ZA200002263B ZA200002263A ZA200002263A ZA200002263B ZA 200002263 B ZA200002263 B ZA 200002263B ZA 200002263 A ZA200002263 A ZA 200002263A ZA 200002263 A ZA200002263 A ZA 200002263A ZA 200002263 B ZA200002263 B ZA 200002263B
Authority
ZA
South Africa
Prior art keywords
synthesis
nucleoside analogs
nucleoside
analogs
Prior art date
Application number
ZA200002263A
Other languages
English (en)
Inventor
Robert William Scott
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of ZA200002263B publication Critical patent/ZA200002263B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H21/00—Compounds containing two or more mononucleotide units having separate phosphate or polyphosphate groups linked by saccharide radicals of nucleoside groups, e.g. nucleic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/14—Pyrrolo-pyrimidine radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Genetics & Genomics (AREA)
  • General Health & Medical Sciences (AREA)
  • Biotechnology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
ZA200002263A 1999-05-11 2000-05-09 Process for the synthesis of nucleoside analogs. ZA200002263B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US13365199P 1999-05-11 1999-05-11

Publications (1)

Publication Number Publication Date
ZA200002263B true ZA200002263B (en) 2001-12-24

Family

ID=22459680

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200002263A ZA200002263B (en) 1999-05-11 2000-05-09 Process for the synthesis of nucleoside analogs.

Country Status (22)

Country Link
US (1) US6271370B1 (de)
EP (1) EP1052264B1 (de)
JP (1) JP2001011092A (de)
KR (1) KR100403900B1 (de)
CN (1) CN1275575A (de)
AR (1) AR028991A1 (de)
AT (1) ATE291582T1 (de)
AU (1) AU3401100A (de)
BR (1) BR0002089A (de)
CA (1) CA2307951A1 (de)
CZ (1) CZ20001710A3 (de)
DE (1) DE60018833D1 (de)
HU (1) HUP0001843A3 (de)
ID (1) ID25992A (de)
IL (1) IL136027A0 (de)
IN (1) IN186850B (de)
MX (1) MXPA00004532A (de)
PL (1) PL340109A1 (de)
RU (1) RU2200738C2 (de)
TR (1) TR200001340A2 (de)
YU (1) YU25500A (de)
ZA (1) ZA200002263B (de)

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RU2019109570A (ru) 2016-09-06 2020-10-08 Ф. Хоффманн-Ля Рош Аг 8-(азетидин-1-ил)-[1,2,4]триазоло[1,5-а]пиридинилы, композиции и способы их применения
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JP2020510061A (ja) 2017-03-14 2020-04-02 エフ．ホフマン−ラ ロシュ アーゲーＦ． Ｈｏｆｆｍａｎｎ−Ｌａ Ｒｏｃｈｅ Ａｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ ピラゾロクロロフェニル化合物、組成物及びその使用方法
TW201900648A (zh) 2017-05-22 2019-01-01 瑞士商赫孚孟拉羅股份公司 治療性化合物及組成物以及其使用方法
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JP7339263B2 (ja) 2018-01-15 2023-09-05 エフ． ホフマン－ラ ロシュ アーゲー Ｊａｋ阻害剤としてのピラゾロピリミジン化合物
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Also Published As

Publication number Publication date
HUP0001843A2 (hu) 2001-06-28
CZ20001710A3 (cs) 2001-09-12
YU25500A (sh) 2003-08-29
MXPA00004532A (es) 2002-03-08
HUP0001843A3 (en) 2001-09-28
EP1052264A3 (de) 2001-06-13
RU2200738C2 (ru) 2003-03-20
HU0001843D0 (en) 2000-07-28
JP2001011092A (ja) 2001-01-16
ID25992A (id) 2000-11-16
DE60018833D1 (de) 2005-04-28
KR20010069193A (ko) 2001-07-23
TR200001340A2 (tr) 2000-12-21
IL136027A0 (en) 2001-05-20
US6271370B1 (en) 2001-08-07
CA2307951A1 (en) 2000-11-11
AU3401100A (en) 2000-11-16
EP1052264B1 (de) 2005-03-23
EP1052264A2 (de) 2000-11-15
CN1275575A (zh) 2000-12-06
AR028991A1 (es) 2003-06-04
BR0002089A (pt) 2001-01-02
PL340109A1 (en) 2000-11-20
KR100403900B1 (ko) 2003-11-01
ATE291582T1 (de) 2005-04-15
IN186850B (de) 2001-11-24

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