UY31545A1 - Nuevos derivados de 2-carboxamida cianoaminourea, sus sales y profarmacos farmacéuticamente aceptables, procesos de preparacion y aplicaciones - Google Patents

Nuevos derivados de 2-carboxamida cianoaminourea, sus sales y profarmacos farmacéuticamente aceptables, procesos de preparacion y aplicaciones

Info

Publication number
UY31545A1
UY31545A1 UY31545A UY31545A UY31545A1 UY 31545 A1 UY31545 A1 UY 31545A1 UY 31545 A UY31545 A UY 31545A UY 31545 A UY31545 A UY 31545A UY 31545 A1 UY31545 A1 UY 31545A1
Authority
UY
Uruguay
Prior art keywords
salts
profarms
cianoaminourea
carboxamide
applications
Prior art date
Application number
UY31545A
Other languages
English (en)
Inventor
Vito Guagnano
Pascal Furet
Robin Alec Fairhurst
Giorgio Caravatti
Patricia Imbach
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of UY31545A1 publication Critical patent/UY31545A1/es

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Abstract

La presente invencion relata los compuestos de formula I y sus sales, en donde los sustituyente son como los definidos en la descripcion; a composiciones y uso de los compuestos en el tratamiento de enfermedades mejoradas por la inhibicion de la fosfadiltilinositol 3-cinasa
UY31545A 2007-12-20 2008-12-18 Nuevos derivados de 2-carboxamida cianoaminourea, sus sales y profarmacos farmacéuticamente aceptables, procesos de preparacion y aplicaciones UY31545A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP07150228 2007-12-20

Publications (1)

Publication Number Publication Date
UY31545A1 true UY31545A1 (es) 2009-08-03

Family

ID=39273277

Family Applications (1)

Application Number Title Priority Date Filing Date
UY31545A UY31545A1 (es) 2007-12-20 2008-12-18 Nuevos derivados de 2-carboxamida cianoaminourea, sus sales y profarmacos farmacéuticamente aceptables, procesos de preparacion y aplicaciones

Country Status (28)

Country Link
US (1) US8940771B2 (es)
EP (1) EP2240475B1 (es)
JP (1) JP2011506560A (es)
KR (1) KR20100093129A (es)
CN (1) CN101952282A (es)
AR (1) AR069798A1 (es)
AU (1) AU2008340053A1 (es)
BR (1) BRPI0820722A2 (es)
CA (1) CA2710122A1 (es)
CL (1) CL2008003822A1 (es)
CO (1) CO6321276A2 (es)
CR (1) CR11491A (es)
DO (1) DOP2010000183A (es)
EA (1) EA201000947A1 (es)
EC (1) ECSP10010271A (es)
ES (1) ES2437595T3 (es)
IL (1) IL206286A0 (es)
MA (1) MA31903B1 (es)
NI (1) NI201000107A (es)
PA (1) PA8809001A1 (es)
PE (1) PE20091523A1 (es)
SM (1) SMP201000096B (es)
SV (1) SV2010003598A (es)
TN (1) TN2010000293A1 (es)
TW (1) TW200930364A (es)
UY (1) UY31545A1 (es)
WO (1) WO2009080694A1 (es)
ZA (1) ZA201003928B (es)

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MA31903B1 (fr) 2010-12-01
SMAP201000096A (it) 2010-09-10
AU2008340053A1 (en) 2009-07-02
KR20100093129A (ko) 2010-08-24
EP2240475B1 (en) 2013-09-25
TN2010000293A1 (en) 2011-11-11
CO6321276A2 (es) 2011-09-20
SMP201000096B (it) 2011-09-09
WO2009080694A1 (en) 2009-07-02
EA201000947A1 (ru) 2011-02-28
PE20091523A1 (es) 2009-10-29
AR069798A1 (es) 2010-02-17
ZA201003928B (en) 2011-04-28
US8940771B2 (en) 2015-01-27
EP2240475A1 (en) 2010-10-20
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BRPI0820722A2 (pt) 2015-06-16
CR11491A (es) 2010-08-05
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US20090163469A1 (en) 2009-06-25
CA2710122A1 (en) 2009-07-02
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ECSP10010271A (es) 2010-07-30
CL2008003822A1 (es) 2009-06-26
ES2437595T3 (es) 2014-01-13
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SV2010003598A (es) 2011-03-23
JP2011506560A (ja) 2011-03-03

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