SG11201502802PA - Hepatitis c virus inhibitors - Google Patents

Hepatitis c virus inhibitors

Info

Publication number
SG11201502802PA
SG11201502802PA SG11201502802PA SG11201502802PA SG11201502802PA SG 11201502802P A SG11201502802P A SG 11201502802PA SG 11201502802P A SG11201502802P A SG 11201502802PA SG 11201502802P A SG11201502802P A SG 11201502802PA SG 11201502802P A SG11201502802P A SG 11201502802PA
Authority
SG
Singapore
Prior art keywords
hepatitis
virus inhibitors
virus
inhibitors
Prior art date
Application number
SG11201502802PA
Other languages
English (en)
Inventor
Li-Qiang Sun
Eric Mull
Eric P Gillis
Michael S Bowsher
Qian Zhao
Kishore V Renduchintala
Kandhasamy Sarkunam
Pulicharla Nagalakshmi
Suresh P V K Babu
Paul Michael Scola
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of SG11201502802PA publication Critical patent/SG11201502802PA/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B59/00Introduction of isotopes of elements into organic compounds ; Labelled organic compounds per se
    • C07B59/002Heterocyclic compounds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08Tripeptides
    • C07K5/0802Tripeptides with the first amino acid being neutral
    • C07K5/0804Tripeptides with the first amino acid being neutral and aliphatic
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08Tripeptides
    • C07K5/0827Tripeptides containing heteroatoms different from O, S, or N
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/05Isotopically modified compounds, e.g. labelled
SG11201502802PA 2012-10-19 2012-10-19 Hepatitis c virus inhibitors SG11201502802PA (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US2012/061094 WO2014062196A1 (fr) 2012-10-19 2012-10-19 Inhibiteurs du virus de l'hépatite c

Publications (1)

Publication Number Publication Date
SG11201502802PA true SG11201502802PA (en) 2015-05-28

Family

ID=47144142

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11201502802PA SG11201502802PA (en) 2012-10-19 2012-10-19 Hepatitis c virus inhibitors

Country Status (30)

Country Link
US (1) US9499550B2 (fr)
EP (1) EP2909205B1 (fr)
JP (1) JP6154474B2 (fr)
KR (1) KR20150074051A (fr)
CN (1) CN104918941A (fr)
AR (1) AR088768A1 (fr)
AU (1) AU2012392557B2 (fr)
BR (1) BR112015007879A2 (fr)
CA (1) CA2888755A1 (fr)
CY (1) CY1118729T1 (fr)
DK (1) DK2909205T3 (fr)
EA (1) EA025560B1 (fr)
ES (1) ES2613766T3 (fr)
HK (1) HK1212332A1 (fr)
HR (1) HRP20161694T1 (fr)
HU (1) HUE031625T2 (fr)
IL (1) IL238286B (fr)
LT (1) LT2909205T (fr)
MA (1) MA37992B1 (fr)
MX (1) MX360452B (fr)
PH (1) PH12015500814A1 (fr)
PL (1) PL2909205T3 (fr)
PT (1) PT2909205T (fr)
RS (1) RS55592B1 (fr)
SG (1) SG11201502802PA (fr)
SI (1) SI2909205T1 (fr)
SM (1) SMT201700117B (fr)
TW (1) TWI570125B (fr)
WO (1) WO2014062196A1 (fr)
ZA (1) ZA201503458B (fr)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2014071007A1 (fr) 2012-11-02 2014-05-08 Bristol-Myers Squibb Company Inhibiteurs du virus de l'hépatite c
US9643999B2 (en) 2012-11-02 2017-05-09 Bristol-Myers Squibb Company Hepatitis C virus inhibitors
US9598433B2 (en) 2012-11-02 2017-03-21 Bristol-Myers Squibb Company Hepatitis C virus inhibitors
WO2014070974A1 (fr) 2012-11-05 2014-05-08 Bristol-Myers Squibb Company Inhibiteurs du virus de l'hépatite c
WO2014137869A1 (fr) 2013-03-07 2014-09-12 Bristol-Myers Squibb Company Inhibiteurs du virus de l'hépatite c
JP2020193181A (ja) * 2019-05-30 2020-12-03 東ソー株式会社 芳香族ニトリル化合物の製造方法
WO2020247736A1 (fr) * 2019-06-07 2020-12-10 University Of Massachusetts Inhibiteurs de protéase ns3/4a du virus de l'hépatite c
CN112094229B (zh) * 2020-10-12 2022-11-22 苏州康润医药有限公司 6-(三氟甲基)异喹啉-5-醇的合成方法
CN114805204B (zh) * 2022-04-01 2023-09-15 云南师范大学 一种制备4-碘异喹啉-1(2h)-酮类化合物的方法

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