PT3759083T - Derivados de 2,4-diaminoquinazolina e seus usos no tratamento de infeções por vírus, cancro ou alergias - Google Patents

Derivados de 2,4-diaminoquinazolina e seus usos no tratamento de infeções por vírus, cancro ou alergias

Info

Publication number
PT3759083T
PT3759083T PT197088172T PT19708817T PT3759083T PT 3759083 T PT3759083 T PT 3759083T PT 197088172 T PT197088172 T PT 197088172T PT 19708817 T PT19708817 T PT 19708817T PT 3759083 T PT3759083 T PT 3759083T
Authority
PT
Portugal
Prior art keywords
medical uses
diaminoquinazoline derivatives
diaminoquinazoline
derivatives
medical
Prior art date
Application number
PT197088172T
Other languages
English (en)
Original Assignee
Janssen Sciences Ireland Unlimited Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Sciences Ireland Unlimited Co filed Critical Janssen Sciences Ireland Unlimited Co
Publication of PT3759083T publication Critical patent/PT3759083T/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Transplantation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
PT197088172T 2018-03-01 2019-02-28 Derivados de 2,4-diaminoquinazolina e seus usos no tratamento de infeções por vírus, cancro ou alergias PT3759083T (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP18159583 2018-03-01

Publications (1)

Publication Number Publication Date
PT3759083T true PT3759083T (pt) 2022-07-05

Family

ID=61557126

Family Applications (1)

Application Number Title Priority Date Filing Date
PT197088172T PT3759083T (pt) 2018-03-01 2019-02-28 Derivados de 2,4-diaminoquinazolina e seus usos no tratamento de infeções por vírus, cancro ou alergias

Country Status (30)

Country Link
US (2) US11597704B2 (pt)
EP (2) EP4059924A1 (pt)
JP (1) JP2021514981A (pt)
KR (1) KR20200128394A (pt)
CN (1) CN111868040A (pt)
AR (1) AR114420A1 (pt)
AU (1) AU2019226342B2 (pt)
BR (1) BR112020017702A2 (pt)
CA (1) CA3091076A1 (pt)
CL (3) CL2020002253A1 (pt)
DK (1) DK3759083T3 (pt)
EA (1) EA202092052A1 (pt)
ES (1) ES2923579T3 (pt)
HR (1) HRP20220781T1 (pt)
HU (1) HUE059149T2 (pt)
IL (2) IL276952B2 (pt)
JO (1) JOP20200208A1 (pt)
LT (1) LT3759083T (pt)
MA (1) MA52411B1 (pt)
MD (1) MD3759083T2 (pt)
MX (2) MX2020009071A (pt)
PH (1) PH12020551345A1 (pt)
PL (1) PL3759083T3 (pt)
PT (1) PT3759083T (pt)
RS (1) RS63401B1 (pt)
SG (1) SG11202008293YA (pt)
SI (1) SI3759083T1 (pt)
TW (1) TW201945003A (pt)
UA (1) UA127590C2 (pt)
WO (1) WO2019166532A1 (pt)

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CN114555565B (zh) * 2019-12-13 2024-03-05 四川科伦博泰生物医药股份有限公司 含氮并环化合物、其制备方法及用途
AU2020416484A1 (en) * 2020-01-02 2022-08-25 Jiangsu Hengrui Medicine Co., Ltd. Crystal form of pyridopyrimidine derivative and preparation method thereof

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Also Published As

Publication number Publication date
JP2021514981A (ja) 2021-06-17
EP4059924A1 (en) 2022-09-21
JOP20200208A1 (ar) 2020-08-30
CL2020002253A1 (es) 2021-01-15
AU2019226342B2 (en) 2024-02-15
MX2020009071A (es) 2020-10-08
MX2023001803A (es) 2023-03-10
PH12020551345A1 (en) 2021-09-06
RS63401B1 (sr) 2022-08-31
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