PA8791601A1 - Compuestos de biciclolactama sustituida - Google Patents

Compuestos de biciclolactama sustituida

Info

Publication number
PA8791601A1
PA8791601A1 PA20088791601A PA8791601A PA8791601A1 PA 8791601 A1 PA8791601 A1 PA 8791601A1 PA 20088791601 A PA20088791601 A PA 20088791601A PA 8791601 A PA8791601 A PA 8791601A PA 8791601 A1 PA8791601 A1 PA 8791601A1
Authority
PA
Panama
Prior art keywords
compounds
bicycolactama
substituted
same
compositions
Prior art date
Application number
PA20088791601A
Other languages
English (en)
Inventor
Lee Dow Robert
John Munchhof Michael
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of PA8791601A1 publication Critical patent/PA8791601A1/es

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/12—Ophthalmic agents for cataracts
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Abstract

LA INVENCIÓN PROPORCIONA COMPUESTOS DE FÓRMULA(1).Y LA SAL FARMACÉUTICAMENTE ACEPTABLE DE LOS MISMOS,EN EL QUE R1,R2,R3,R4,R5a,R5b,R5c,R5d,Q,A,Z,Y R7 SON COMO SE HA DESCRITO EN ESTE DOCUMENTO;COMPOSICIONES DE LOS MISMOS;Y USOS DE LOS MISMOS.
PA20088791601A 2007-08-02 2008-07-30 Compuestos de biciclolactama sustituida PA8791601A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US95350707P 2007-08-02 2007-08-02

Publications (1)

Publication Number Publication Date
PA8791601A1 true PA8791601A1 (es) 2009-12-16

Family

ID=39926534

Family Applications (1)

Application Number Title Priority Date Filing Date
PA20088791601A PA8791601A1 (es) 2007-08-02 2008-07-30 Compuestos de biciclolactama sustituida

Country Status (34)

Country Link
US (2) US20090036425A1 (es)
EP (1) EP2185567B1 (es)
JP (1) JP4629808B2 (es)
KR (1) KR20100032443A (es)
CN (1) CN101772504A (es)
AP (1) AP2010005163A0 (es)
AR (1) AR067780A1 (es)
AT (1) ATE502948T1 (es)
AU (1) AU2008281545B2 (es)
BR (1) BRPI0815067A2 (es)
CA (1) CA2695291C (es)
CL (1) CL2008002227A1 (es)
CO (1) CO6251365A2 (es)
CR (1) CR11223A (es)
CY (1) CY1111628T1 (es)
DE (1) DE602008005757D1 (es)
DK (1) DK2185567T3 (es)
DO (1) DOP2010000046A (es)
EA (1) EA201000050A1 (es)
EC (1) ECSP109932A (es)
ES (1) ES2361716T3 (es)
HN (1) HN2008001191A (es)
HR (1) HRP20110335T1 (es)
MA (1) MA31580B1 (es)
PA (1) PA8791601A1 (es)
PE (1) PE20090897A1 (es)
PL (1) PL2185567T3 (es)
PT (1) PT2185567E (es)
SI (1) SI2185567T1 (es)
TN (1) TN2010000053A1 (es)
TW (1) TWI356059B (es)
UA (1) UA94833C2 (es)
WO (1) WO2009016462A2 (es)
ZA (1) ZA201000255B (es)

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Also Published As

Publication number Publication date
JP4629808B2 (ja) 2011-02-09
CA2695291C (en) 2012-04-17
DE602008005757D1 (de) 2011-05-05
HN2008001191A (es) 2012-01-17
ATE502948T1 (de) 2011-04-15
EA201000050A1 (ru) 2010-08-30
EP2185567B1 (en) 2011-03-23
CO6251365A2 (es) 2011-02-21
SI2185567T1 (sl) 2011-06-30
JP2010535190A (ja) 2010-11-18
CN101772504A (zh) 2010-07-07
WO2009016462A3 (en) 2009-03-26
US7718645B2 (en) 2010-05-18
BRPI0815067A2 (pt) 2015-02-10
DK2185567T3 (da) 2011-05-16
CA2695291A1 (en) 2009-02-05
TWI356059B (en) 2012-01-11
HRP20110335T1 (hr) 2011-06-30
KR20100032443A (ko) 2010-03-25
WO2009016462A2 (en) 2009-02-05
AU2008281545A1 (en) 2009-02-05
MA31580B1 (fr) 2010-08-02
AU2008281545B2 (en) 2011-12-08
TW200916471A (en) 2009-04-16
AP2010005163A0 (en) 2010-02-28
ZA201000255B (en) 2011-03-30
CL2008002227A1 (es) 2009-04-17
PL2185567T3 (pl) 2011-07-29
CY1111628T1 (el) 2015-10-07
CR11223A (es) 2010-02-04
DOP2010000046A (es) 2010-03-31
US20090137551A1 (en) 2009-05-28
ECSP109932A (es) 2010-03-31
UA94833C2 (en) 2011-06-10
US20090036425A1 (en) 2009-02-05
PT2185567E (pt) 2011-05-27
EP2185567A2 (en) 2010-05-19
ES2361716T3 (es) 2011-06-21
PE20090897A1 (es) 2009-08-06
AR067780A1 (es) 2009-10-21
TN2010000053A1 (fr) 2011-09-26

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