NO952872D0 - 2,6-diaminopurin-derivater - Google Patents
2,6-diaminopurin-derivaterInfo
- Publication number
- NO952872D0 NO952872D0 NO952872A NO952872A NO952872D0 NO 952872 D0 NO952872 D0 NO 952872D0 NO 952872 A NO952872 A NO 952872A NO 952872 A NO952872 A NO 952872A NO 952872 D0 NO952872 D0 NO 952872D0
- Authority
- NO
- Norway
- Prior art keywords
- diaminopurine derivatives
- diaminopurine
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/16—Purine radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/16—Purine radicals
- C07H19/167—Purine radicals with ribosyl as the saccharide radical
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biotechnology (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Immunology (AREA)
- Pulmonology (AREA)
- Oncology (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Cardiology (AREA)
- Transplantation (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Hydrogenated Pyridines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB939301000A GB9301000D0 (en) | 1993-01-20 | 1993-01-20 | Chemical compounds |
PCT/EP1994/000145 WO1994017090A1 (en) | 1993-01-20 | 1994-01-18 | 2,6-diaminopurine derivatives |
Publications (3)
Publication Number | Publication Date |
---|---|
NO952872D0 true NO952872D0 (no) | 1995-07-19 |
NO952872L NO952872L (no) | 1995-09-13 |
NO305603B1 NO305603B1 (no) | 1999-06-28 |
Family
ID=10728948
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO952872A NO305603B1 (no) | 1993-01-20 | 1995-07-19 | 2,6-diaminopurin-derivater, anvendelse derav samt farmas°ytisk blanding |
Country Status (29)
Country | Link |
---|---|
US (2) | US5925624A (no) |
EP (1) | EP0680488B1 (no) |
JP (1) | JP3768232B2 (no) |
KR (1) | KR960700261A (no) |
CN (1) | CN1043997C (no) |
AP (1) | AP457A (no) |
AT (1) | ATE164849T1 (no) |
AU (1) | AU679714B2 (no) |
CA (1) | CA2153688A1 (no) |
CZ (1) | CZ187995A3 (no) |
DE (1) | DE69409503T2 (no) |
DK (1) | DK0680488T3 (no) |
EC (1) | ECSP941104A (no) |
ES (1) | ES2117249T3 (no) |
FI (1) | FI953489A (no) |
GB (1) | GB9301000D0 (no) |
HU (1) | HU211914A9 (no) |
IL (1) | IL108372A (no) |
IS (1) | IS4121A (no) |
NO (1) | NO305603B1 (no) |
NZ (1) | NZ259880A (no) |
PE (1) | PE54194A1 (no) |
PL (1) | PL309975A1 (no) |
RU (1) | RU2129561C1 (no) |
SI (1) | SI9400021A (no) |
SK (1) | SK281229B6 (no) |
TW (1) | TW267168B (no) |
WO (1) | WO1994017090A1 (no) |
ZA (1) | ZA94335B (no) |
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TW528755B (en) * | 1996-12-24 | 2003-04-21 | Glaxo Group Ltd | 2-(purin-9-yl)-tetrahydrofuran-3,4-diol derivatives |
JP3861413B2 (ja) * | 1997-11-05 | 2006-12-20 | ソニー株式会社 | 情報配信システム、情報処理端末装置、携帯端末装置 |
YU44900A (sh) | 1998-01-31 | 2003-01-31 | Glaxo Group Limited | Derivati 2-(purin-9-il)tetrahidrofuran-3,4-diola |
US6479487B1 (en) | 1998-02-26 | 2002-11-12 | Aventis Pharmaceuticals Inc. | 6, 9-disubstituted 2-[trans-(4-aminocyclohexyl)amino] purines |
US6413974B1 (en) | 1998-02-26 | 2002-07-02 | Aventis Pharmaceuticals Inc. | 6,9,-disubstituted 2-[trans-(4-aminocyclohexyl) amino] purines |
CA2320448C (en) * | 1998-02-26 | 2005-02-01 | Aventis Pharmaceuticals Inc. | 6,9-disubstituted 2-[trans-(4-aminocyclohexyl)amino]purines |
YU76100A (sh) | 1998-06-02 | 2003-12-31 | Osi Pharmaceuticals Inc. | Pirolo(2,3-d) pirimidin preparati i njihova primena |
US6686366B1 (en) | 1998-06-02 | 2004-02-03 | Osi Pharmaceuticals, Inc. | Compounds specific to adenosine A3 receptor and uses thereof |
US6878716B1 (en) | 1998-06-02 | 2005-04-12 | Osi Pharmaceuticals, Inc. | Compounds specific to adenosine A1 receptor and uses thereof |
GB9813535D0 (en) | 1998-06-23 | 1998-08-19 | Glaxo Group Ltd | Chemical compounds |
ATE246701T1 (de) * | 1998-06-23 | 2003-08-15 | Glaxo Group Ltd | 2-(purin-9-yl)-tetrahydrofuran-3,4-diol derivate |
GB9813554D0 (en) * | 1998-06-23 | 1998-08-19 | Glaxo Group Ltd | Chemical compounds |
GB9813540D0 (en) * | 1998-06-23 | 1998-08-19 | Glaxo Group Ltd | Chemical compounds |
GB9813565D0 (en) * | 1998-06-23 | 1998-08-19 | Glaxo Group Ltd | Chemical compounds |
US6664252B2 (en) | 1999-12-02 | 2003-12-16 | Osi Pharmaceuticals, Inc. | 4-aminopyrrolo[2,3-d]pyrimidine compounds specific to adenosine A2a receptor and uses thereof |
US7160890B2 (en) | 1999-12-02 | 2007-01-09 | Osi Pharmaceuticals, Inc. | Compounds specific to adenosine A3 receptor and uses thereof |
US6680322B2 (en) | 1999-12-02 | 2004-01-20 | Osi Pharmaceuticals, Inc. | Compounds specific to adenosine A1 receptors and uses thereof |
JP2003531111A (ja) | 1999-12-17 | 2003-10-21 | アライアッド・ファーマシューティカルズ・インコーポレーテッド | プロトンポンプインヒビター |
EP1939203B1 (en) * | 2000-04-25 | 2014-11-19 | ICOS Corporation | Inhibitors of human phosphatidyl-inositol 3-kinase delta isoform |
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US6680324B2 (en) | 2000-12-01 | 2004-01-20 | Osi Pharmaceuticals, Inc. | Compounds specific to adenosine A1 receptors and uses thereof |
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US5106837A (en) * | 1988-03-16 | 1992-04-21 | The Scripps Research Institute | Adenosine derivatives with therapeutic activity |
US4757747A (en) * | 1986-04-08 | 1988-07-19 | Vickers, Incorporated | Power transmission |
AU8274187A (en) * | 1986-10-31 | 1988-05-25 | Warner-Lambert Company | Heteroaromatic derivatives of adenosine |
US4968697A (en) * | 1987-02-04 | 1990-11-06 | Ciba-Geigy Corporation | 2-substituted adenosine 5'-carboxamides as antihypertensive agents |
FI880405A (fi) | 1987-02-04 | 1988-08-05 | Ciba Geigy Ag | Adenosin-5'-karboxamidderivat. |
US5219840A (en) * | 1987-04-06 | 1993-06-15 | Sandoz Ltd. | Antihypertensive 9-(2,N6 -disubstituted adenyl) ribofuranuronic acid derivatives |
LU87181A1 (fr) * | 1987-04-06 | 1988-11-17 | Sandoz Sa | Nouveaux derives de l'acide furannuronique,leur preparation et leur utilisation comme medicaments |
CA1339964C (en) * | 1988-03-16 | 1998-07-21 | Dennis A. Carson | Substituted adenine derivatives useful as therapeutic agents |
JPH0725785B2 (ja) * | 1989-01-11 | 1995-03-22 | 日本臓器製薬株式会社 | アデノシン誘導体及び該化合物を有効成分として含有する医薬組成物 |
DE3924424A1 (de) * | 1989-07-24 | 1991-01-31 | Boehringer Mannheim Gmbh | Nucleosid-derivate, verfahren zu deren herstellung, deren verwendung als arzneimittel sowie deren verwendung bei der nucleinsaeure-sequenzierung |
IE903747A1 (en) * | 1989-10-19 | 1991-04-24 | Searle & Co | Method of treating gastrointestinal motility disorders |
US5459255A (en) * | 1990-01-11 | 1995-10-17 | Isis Pharmaceuticals, Inc. | N-2 substituted purines |
DE4025879A1 (de) * | 1990-08-16 | 1992-02-20 | Sandoz Ag | Neue adenosin derivate, deren herstellung und verwendung |
FR2687678B1 (fr) * | 1992-01-31 | 1995-03-31 | Union Pharma Scient Appl | Nouveaux derives de l'adenosine, leurs procedes de preparation, compositions pharmaceutiques les contenant. |
US5773423A (en) * | 1993-07-13 | 1998-06-30 | The United States Of America As Represented By The Department Of Health And Human Services | A3 adenosine receptor agonists |
-
1993
- 1993-01-20 GB GB939301000A patent/GB9301000D0/en active Pending
-
1994
- 1994-01-14 IS IS4121A patent/IS4121A/is unknown
- 1994-01-18 CN CN94191527A patent/CN1043997C/zh not_active Expired - Fee Related
- 1994-01-18 NZ NZ259880A patent/NZ259880A/en unknown
- 1994-01-18 RU RU95122754A patent/RU2129561C1/ru active
- 1994-01-18 DK DK94905100T patent/DK0680488T3/da active
- 1994-01-18 AU AU58851/94A patent/AU679714B2/en not_active Ceased
- 1994-01-18 DE DE69409503T patent/DE69409503T2/de not_active Expired - Lifetime
- 1994-01-18 AT AT94905100T patent/ATE164849T1/de not_active IP Right Cessation
- 1994-01-18 ES ES94905100T patent/ES2117249T3/es not_active Expired - Lifetime
- 1994-01-18 US US08/446,727 patent/US5925624A/en not_active Expired - Fee Related
- 1994-01-18 ZA ZA94335A patent/ZA94335B/xx unknown
- 1994-01-18 AP APAP/P/1994/000613A patent/AP457A/en active
- 1994-01-18 KR KR1019950702963A patent/KR960700261A/ko active IP Right Grant
- 1994-01-18 CZ CZ951879A patent/CZ187995A3/cs unknown
- 1994-01-18 JP JP51665294A patent/JP3768232B2/ja not_active Expired - Fee Related
- 1994-01-18 PL PL94309975A patent/PL309975A1/xx unknown
- 1994-01-18 EP EP94905100A patent/EP0680488B1/en not_active Expired - Lifetime
- 1994-01-18 WO PCT/EP1994/000145 patent/WO1994017090A1/en not_active Application Discontinuation
- 1994-01-18 CA CA002153688A patent/CA2153688A1/en not_active Abandoned
- 1994-01-18 SK SK918-95A patent/SK281229B6/sk unknown
- 1994-01-19 SI SI9400021A patent/SI9400021A/sl unknown
- 1994-01-19 IL IL108372A patent/IL108372A/en not_active IP Right Cessation
- 1994-05-30 TW TW083104895A patent/TW267168B/zh active
- 1994-06-14 EC EC1994001104A patent/ECSP941104A/es unknown
- 1994-06-15 PE PE1994244634A patent/PE54194A1/es not_active Application Discontinuation
-
1995
- 1995-06-28 HU HU95P/P00514P patent/HU211914A9/hu unknown
- 1995-07-19 NO NO952872A patent/NO305603B1/no not_active IP Right Cessation
- 1995-07-19 FI FI953489A patent/FI953489A/fi unknown
-
1997
- 1997-09-22 US US08/934,540 patent/US5889178A/en not_active Expired - Lifetime
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