US3832460A
(en)
|
1971-03-19 |
1974-08-27 |
C Kosti |
Anesthetic-vasoconstrictor-antihistamine composition for the treatment of hypertrophied oral tissue
|
US4140755A
(en)
|
1976-02-13 |
1979-02-20 |
Hoffmann-La Roche Inc. |
Sustained release tablet formulations
|
US5077290A
(en)
|
1990-10-11 |
1991-12-31 |
Merck & Co., Inc. |
Morpholine derivatives compositions and use
|
US6638905B2
(en)
|
1993-06-18 |
2003-10-28 |
The Salk Institute For Biological Studies |
Cloning and recombinant production of CFR receptor(s)
|
US5795909A
(en)
|
1996-05-22 |
1998-08-18 |
Neuromedica, Inc. |
DHA-pharmaceutical agent conjugates of taxanes
|
US6624138B1
(en)
|
2001-09-27 |
2003-09-23 |
Gp Medical |
Drug-loaded biological material chemically treated with genipin
|
TW530054B
(en)
|
1997-09-24 |
2003-05-01 |
Duphar Int Res |
New piperazine and piperidine compounds
|
PA8474101A1
(es)
|
1998-06-19 |
2000-09-29 |
Pfizer Prod Inc |
Compuestos de pirrolo [2,3-d] pirimidina
|
CA2343148C
(en)
|
1998-09-10 |
2005-11-15 |
Nycomed Danmark A/S |
Quick release pharmaceutical compositions of drug substances
|
PT1235830E
(pt)
|
1999-12-10 |
2004-04-30 |
Pfizer Prod Inc |
Compostos de pirrolo¬2,3-d|pirimidina como inibidores das proteina cinases
|
EE05180B1
(et)
|
1999-12-24 |
2009-06-15 |
Aventis Pharma Limited |
Asaindooli sisaldav farmatseutiline kompositsioon raviotstarbeliseks kasutamiseks, asaindoolid ning nende kasutamine ravimite valmistamiseks, mis on ette nhtud proteiinikinaasi kataltilise toime prssimiseks
|
TR200302105T4
(tr)
|
2000-04-07 |
2004-02-23 |
Laboratoire Medidom S. A. |
Siklosporin, hiyalüronik asit ve polisorbat içeren göz formülasyonları.
|
CA2412560C
(en)
|
2000-06-26 |
2008-12-30 |
Pfizer Products Inc. |
Pyrrolo[2,3-d]pyrimidine compounds as immunosuppressive agents
|
SE0102439D0
(sv)
|
2001-07-05 |
2001-07-05 |
Astrazeneca Ab |
New compounds
|
CA2455181C
(en)
|
2001-08-01 |
2010-04-06 |
Merck & Co., Inc. |
Benzimidazo[4,5-f]isoquinolinone derivatives
|
US6995144B2
(en)
|
2002-03-14 |
2006-02-07 |
Eisai Co., Ltd. |
Nitrogen containing heterocyclic compounds and medicines containing the same
|
TW200403058A
(en)
|
2002-04-19 |
2004-03-01 |
Bristol Myers Squibb Co |
Heterocyclo inhibitors of potassium channel function
|
EP1501514B1
(en)
|
2002-05-03 |
2012-12-19 |
Exelixis, Inc. |
Protein kinase modulators and methods of use
|
WO2004000318A2
(en)
|
2002-06-21 |
2003-12-31 |
Cellular Genomics, Inc. |
Certain amino-substituted monocycles as kinase modulators
|
US20040067985A1
(en)
|
2002-10-04 |
2004-04-08 |
Fortuna Haviv |
Method of inhibiting angiogenesis
|
SE0203753D0
(sv)
|
2002-12-17 |
2002-12-17 |
Astrazeneca Ab |
New compounds
|
US7444183B2
(en)
|
2003-02-03 |
2008-10-28 |
Enteromedics, Inc. |
Intraluminal electrode apparatus and method
|
AU2004212421B2
(en)
|
2003-02-07 |
2009-08-20 |
Vertex Pharmaceuticals Incorporated |
Heteroaryl substituted pyrolls useful as inhibitors of protein kinases
|
US20040265909A1
(en)
|
2003-04-11 |
2004-12-30 |
Jeff Blaney |
Compound libraries and methods for drug discovery
|
SE0301373D0
(sv)
|
2003-05-09 |
2003-05-09 |
Astrazeneca Ab |
Novel compounds
|
SE0301372D0
(sv)
|
2003-05-09 |
2003-05-09 |
Astrazeneca Ab |
Novel compounds
|
US20050043346A1
(en)
|
2003-08-08 |
2005-02-24 |
Pharmacia Italia S.P.A. |
Pyridylpyrrole derivatives active as kinase inhibitors
|
US20050153989A1
(en)
|
2004-01-13 |
2005-07-14 |
Ambit Biosciences Corporation |
Pyrrolopyrimidine derivatives and analogs and their use in the treatment and prevention of diseases
|
WO2005115985A1
(en)
|
2004-05-27 |
2005-12-08 |
Pfizer Limited |
Aminopyridine derivatives as selective dopamine d3 agonists
|
US7138423B2
(en)
|
2004-07-20 |
2006-11-21 |
Bristol-Myers Squibb Company |
Arylpyrrolidine derivatives as NK-1 /SSRI antagonists
|
SA05260265A
(ar)
|
2004-08-30 |
2005-12-03 |
استرازينيكا ايه بي |
مركبات جديدة
|
MY179032A
(en)
|
2004-10-25 |
2020-10-26 |
Cancer Research Tech Ltd |
Ortho-condensed pyridine and pyrimidine derivatives (e.g.purines) as protein kinase inhibitors
|
US7517870B2
(en)
|
2004-12-03 |
2009-04-14 |
Fondazione Telethon |
Use of compounds that interfere with the hedgehog signaling pathway for the manufacture of a medicament for preventing, inhibiting, and/or reversing ocular diseases related with ocular neovascularization
|
AR054416A1
(es)
|
2004-12-22 |
2007-06-27 |
Incyte Corp |
Pirrolo [2,3-b]piridin-4-il-aminas y pirrolo [2,3-b]pirimidin-4-il-aminas como inhibidores de las quinasas janus. composiciones farmaceuticas.
|
RU2434871C2
(ru)
|
2005-02-03 |
2011-11-27 |
Вертекс Фармасьютикалз Инкорпорейтед |
Пирролопиримидины, применимые в качестве ингибиторов протеинкиназы
|
CA2603959A1
(en)
|
2005-04-08 |
2006-10-19 |
Eisai R & D Management Co., Ltd. |
Therapeutic agent for dyskinesia
|
CN101228161B
(zh)
|
2005-05-20 |
2012-10-10 |
沃泰克斯药物股份有限公司 |
适用作蛋白激酶抑制剂的吡咯并吡啶类
|
WO2007011760A2
(en)
|
2005-07-15 |
2007-01-25 |
Kalypsys, Inc. |
Inhibitors of mitotic kinesin
|
EP2270014A1
(en)
|
2005-09-22 |
2011-01-05 |
Incyte Corporation |
Azepine inhibitors of janus kinases
|
US20130137681A1
(en)
|
2005-12-13 |
2013-05-30 |
Incyte Corporation |
HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINES AND PYRROLO[2,3-b]PYRIMIDINES AS JANUS KINASE INHIBITORS
|
KR101391900B1
(ko)
|
2005-12-13 |
2014-05-02 |
인사이트 코포레이션 |
야누스 키나아제 억제제로서의 헤테로아릴 치환된 피롤로[2,3-b]피리딘 및 피롤로[2,3-b]피리미딘
|
PE20071241A1
(es)
|
2006-01-17 |
2008-01-14 |
Schering Corp |
Compuestos derivados de hidantoina para el tratamiento de trastornos inflamatorios
|
AU2007265368A1
(en)
|
2006-06-29 |
2008-01-03 |
Alantos Pharmaceuticals Holding, Inc. |
Metalloprotease inhibitors
|
BRPI0718029A2
(pt)
|
2006-11-06 |
2013-11-26 |
Supergen Inc |
Derivados de imidazo(1,2-b)piridazina e pirazolo(1,5-a)pirimidina e seu uso como inibidores da proteína cinase
|
JP5492565B2
(ja)
|
2006-12-22 |
2014-05-14 |
インサイト・コーポレイション |
Janusキナーゼ阻害剤としての置換複素環
|
KR101549876B1
(ko)
|
2007-06-13 |
2015-09-03 |
인사이트 코포레이션 |
야누스 키나제 억제제(R)―3―(4―(7H―피롤로[2,3-d]피리미딘―4―일)―1H―피라졸―1―일)―3―사이클로펜틸프로판니트릴의 염
|
CL2008001709A1
(es)
|
2007-06-13 |
2008-11-03 |
Incyte Corp |
Compuestos derivados de pirrolo [2,3-b]pirimidina, moduladores de quinasas jak; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como cancer, psoriasis, artritis reumatoide, entre otras.
|
BRPI0820544A2
(pt)
|
2007-11-16 |
2015-06-16 |
Incyte Corp |
4-pirazolil-n-arilpirimidin-2-aminas e pirazolil-n-heteroarilpirimidin-2-aminas como inibidores de janus cinase
|
EP2288610B8
(en)
|
2008-03-11 |
2016-10-12 |
Incyte Holdings Corporation |
Azetidine and cyclobutane derivatives as jak inhibitors
|
US20110294836A1
(en)
|
2008-06-20 |
2011-12-01 |
Metabolex, Inc. |
Aryl gpr119 agonists and uses thereof
|
CL2009001884A1
(es)
|
2008-10-02 |
2010-05-14 |
Incyte Holdings Corp |
Uso de 3-ciclopentil-3-[4-(7h-pirrolo[2,3-d]pirimidin-4-il)-1h-pirazol-1-il)propanonitrilo, inhibidor de janus quinasa, y uso de una composición que lo comprende para el tratamiento del ojo seco.
|
JOP20190231A1
(ar)
|
2009-01-15 |
2017-06-16 |
Incyte Corp |
طرق لاصلاح مثبطات انزيم jak و المركبات الوسيطة المتعلقة به
|
NZ596374A
(en)
|
2009-05-22 |
2014-01-31 |
Incyte Corp |
3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]octane- or heptane-nitrile as jak inhibitors
|
ES2487542T3
(es)
|
2009-05-22 |
2014-08-21 |
Incyte Corporation |
Derivados de N-(hetero)aril-pirrolidina de pirazol-4-il-pirrolo[2,3-d]pirimidinas y pirrol-3-il-pirrolo[2,3-d]pirimidinas como inhibidores de cinasas Janus
|
US9249145B2
(en)
|
2009-09-01 |
2016-02-02 |
Incyte Holdings Corporation |
Heterocyclic derivatives of pyrazol-4-yl-pyrrolo[2,3-d]pyrimidines as janus kinase inhibitors
|
CN102596960B
(zh)
|
2009-10-09 |
2016-01-20 |
因西特控股公司 |
3-(4-(7H-吡咯并[2,3-d]嘧啶-4-基)-1H-吡唑-1-基)-3-环戊基丙腈的羟基衍生物、酮基衍生物和葡糖苷酸衍生物
|
CA2790070C
(en)
|
2010-02-18 |
2018-03-06 |
Incyte Corporation |
Cyclobutane and methylcyclobutane derivatives as janus kinase inhibitors
|
SI3050882T1
(en)
|
2010-03-10 |
2018-06-29 |
Incyte Holdings Corporation |
Piperidin-4-yl azetidine derivatives, as inhibitors of JAK1
|
TWI499421B
(zh)
|
2010-05-21 |
2015-09-11 |
Incyte Corp |
Jak抑制劑的局部製劑
|
JP5917544B2
(ja)
|
2010-11-19 |
2016-05-18 |
インサイト・ホールディングス・コーポレイションIncyte Holdings Corporation |
Jak阻害剤としての複素環置換ピロロピリジンおよびピロロピリミジン
|
PE20140146A1
(es)
|
2010-11-19 |
2014-02-06 |
Incyte Corp |
Derivados de pirrolopiridina y pirrolopirimidina sustituidos con ciclobutilo como inhibidores de jak
|
WO2012073143A1
(en)
|
2010-12-01 |
2012-06-07 |
Pfizer Inc. |
Kat ii inhibitors
|
US8987271B2
(en)
|
2010-12-22 |
2015-03-24 |
Eutropics Pharmaceuticals, Inc. |
2,2′-biphenazine compounds and methods useful for treating disease
|
CN103732226B
(zh)
|
2011-02-18 |
2016-01-06 |
诺瓦提斯药物公司 |
mTOR/JAK抑制剂组合疗法
|
EA023364B1
(ru)
|
2011-05-23 |
2016-05-31 |
Мерк Патент Гмбх |
Производные пиридина и пиразина
|
ES2560611T3
(es)
|
2011-06-20 |
2016-02-22 |
Incyte Holdings Corporation |
Derivados de fenil de azetidinilo, carboxamida de piridilo o pirazinilo como inhibidores de JAK
|
EP2741747A1
(en)
|
2011-08-10 |
2014-06-18 |
Novartis Pharma AG |
JAK P13K/mTOR COMBINATION THERAPY
|
TW201313721A
(zh)
|
2011-08-18 |
2013-04-01 |
Incyte Corp |
作為jak抑制劑之環己基氮雜環丁烷衍生物
|
UA111854C2
(uk)
|
2011-09-07 |
2016-06-24 |
Інсайт Холдінгс Корпорейшн |
Способи і проміжні сполуки для отримання інгібіторів jak
|
CA3123737A1
(en)
|
2011-09-09 |
2013-03-14 |
Lantheus Medical Imaging, Inc. |
Compositions, methods, and systems for the synthesis and use of imaging agents
|
TW201406761A
(zh)
|
2012-05-18 |
2014-02-16 |
Incyte Corp |
做爲jak抑制劑之哌啶基環丁基取代之吡咯并吡啶及吡咯并嘧啶衍生物
|
US20150197525A1
(en)
|
2012-06-15 |
2015-07-16 |
Concert Pharmaceuticals, Inc. |
Deuterated derivatives of ruxolitinib
|
CN104768548B
(zh)
|
2012-09-28 |
2018-08-10 |
范德比尔特大学 |
作为选择性bmp抑制剂的稠合杂环化合物
|
UA120834C2
(uk)
|
2012-11-15 |
2020-02-25 |
Інсайт Холдінгс Корпорейшн |
Лікарські форми руксолітинібу зі сповільненим вивільненням
|
US20160115167A1
(en)
|
2013-03-04 |
2016-04-28 |
The Brigham And Women's Hospital, Inc. |
Bmp inhibitors and methods of use thereof
|
EP2970205B1
(en)
|
2013-03-14 |
2019-05-08 |
Tolero Pharmaceuticals, Inc. |
Jak2 and alk2 inhibitors and methods for their use
|
CN105555313A
(zh)
|
2013-08-20 |
2016-05-04 |
因赛特公司 |
在c-反应蛋白水平较高的实体肿瘤患者中的存活益处
|
RU2703301C2
(ru)
|
2013-10-21 |
2019-10-16 |
Мерк Патент Гмбх |
Соединения гетероарила в качестве ингибиторов btk и их применение
|
WO2016118638A1
(en)
|
2015-01-20 |
2016-07-28 |
Merial Inc. |
Anthelmintic compounds, compositions and method of using thereof
|
BR112019000941A2
(pt)
*
|
2016-07-20 |
2019-04-30 |
Novartis Ag |
derivados de aminopiridina e seu uso como inibidores seletivos de alk-2
|
WO2018106820A1
(en)
|
2016-12-07 |
2018-06-14 |
Kura Oncology, Inc. |
Methods of promoting beta cell proliferation
|
CN113015527A
(zh)
*
|
2018-08-21 |
2021-06-22 |
西拉肿瘤学公司 |
治疗骨髓纤维化的血小板计数诊断方法
|
WO2021062163A1
(en)
|
2019-09-27 |
2021-04-01 |
Disc Medicine, Inc. |
Methods for treating myelofibrosis and related conditions
|
EP4041243A4
(en)
|
2019-09-27 |
2023-10-18 |
Disc Medicine, Inc. |
METHOD FOR TREATING ANEMIA IN CHRONIC DISEASES
|
TW202214239A
(zh)
|
2020-06-16 |
2022-04-16 |
美商英塞特公司 |
用於治療貧血之alk2抑制劑
|