MA30890B1 - Compose indole - Google Patents
Compose indoleInfo
- Publication number
- MA30890B1 MA30890B1 MA31871A MA31871A MA30890B1 MA 30890 B1 MA30890 B1 MA 30890B1 MA 31871 A MA31871 A MA 31871A MA 31871 A MA31871 A MA 31871A MA 30890 B1 MA30890 B1 MA 30890B1
- Authority
- MA
- Morocco
- Prior art keywords
- indole compound
- agent
- prodruce
- gluckkinase
- prophylaxis
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/433—Thidiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Abstract
LA PRÉSENTE INVENTION CONCERNE UN ACTIVATEUR DE GLUCOKINASE UTILE EN TANT QU'AGENT PHARMACEUTIQUE TEL QU'UN AGENT POUR LA PROPHYLAXIE OU LE TRAITEMENT DU DIABÈTE, DE L'OBÉSITÉ ET AUTRES CONDITIONS SIMILAIRES. LA PRÉSENTE INVENTION PROPOSE UN ACTIVATEUR DE GLUCOKINASE CONTENANT UN COMPOSÉ REPRÉSENTÉ PAR LA FORMULE (I) : DANS LAQUELLE R1 EST UN ATOME D'HYDROGÈNE OU UN ATOME D'HALOGÈNE; R2 EST UN GROUPE REPRÉSENTÉ PAR DANS LAQUELLE CHAQUE SYMBOLE EST DÉFINI DANS LA DESCRIPTION, OU UN SEL DE CELUI-CI OU UN PROMÉDICAMENT DE CELUI-CI.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2006285551 | 2006-10-19 |
Publications (1)
Publication Number | Publication Date |
---|---|
MA30890B1 true MA30890B1 (fr) | 2009-11-02 |
Family
ID=39010108
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MA31871A MA30890B1 (fr) | 2006-10-19 | 2009-05-13 | Compose indole |
Country Status (26)
Country | Link |
---|---|
US (4) | US8410087B2 (fr) |
EP (2) | EP2074119A1 (fr) |
JP (1) | JP5260507B2 (fr) |
KR (1) | KR101444486B1 (fr) |
CN (1) | CN101573357B (fr) |
AU (1) | AU2007310064B2 (fr) |
BR (1) | BRPI0717722A2 (fr) |
CA (1) | CA2666973C (fr) |
CL (1) | CL2008001017A1 (fr) |
CR (1) | CR10748A (fr) |
EC (1) | ECSP099330A (fr) |
GE (1) | GEP20115241B (fr) |
IL (1) | IL198154A (fr) |
MA (1) | MA30890B1 (fr) |
ME (1) | ME00681B (fr) |
MX (1) | MX2009003972A (fr) |
MY (1) | MY158052A (fr) |
NO (1) | NO20091948L (fr) |
NZ (1) | NZ576570A (fr) |
PE (1) | PE20090884A1 (fr) |
RU (1) | RU2454415C9 (fr) |
TN (1) | TN2009000129A1 (fr) |
TW (1) | TWI460176B (fr) |
UA (1) | UA97257C2 (fr) |
WO (1) | WO2008050821A1 (fr) |
ZA (1) | ZA200902585B (fr) |
Families Citing this family (70)
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EP2134684B1 (fr) * | 2007-04-16 | 2017-08-02 | AbbVie Inc. | Indole 7-substitué en tant qu'inhibiteurs de mcl-1 |
US8318746B2 (en) | 2007-04-27 | 2012-11-27 | Takeda Pharmaceutical Company Limited | Nitrogen-containing five-membered heterocyclic compound |
EP2025674A1 (fr) | 2007-08-15 | 2009-02-18 | sanofi-aventis | Tetrahydronaphthaline substituée, son procédé de fabrication et son utilisation en tant que médicament |
JP5323834B2 (ja) | 2007-08-17 | 2013-10-23 | エルジー・ライフ・サイエンシーズ・リミテッド | 細胞壊死阻害剤としてのインドール化合物 |
CN101896483B (zh) | 2007-12-20 | 2013-11-20 | 株式会社Lg生命科学 | 葡糖激酶激活剂和包含其作为活性成分的药物组合物 |
JP5188583B2 (ja) * | 2008-01-04 | 2013-04-24 | エルジー・ライフ・サイエンシーズ・リミテッド | 細胞、組織及び臓器保存効果を有するインドール及びインダゾール誘導体 |
EP2242745A1 (fr) * | 2008-02-07 | 2010-10-27 | Sanofi-Aventis | Nouvelles imidazolidines substituées par un phényle, procédé de production, médicaments contenant ces composés et leur utilisation |
JP5528348B2 (ja) | 2008-04-10 | 2014-06-25 | 武田薬品工業株式会社 | 縮合環化合物およびその用途 |
EP2266983B1 (fr) * | 2008-04-16 | 2013-06-05 | Takeda Pharmaceutical Company Limited | Composé hétérocyclique azoté à cinq chaînons |
AR072297A1 (es) * | 2008-06-27 | 2010-08-18 | Novartis Ag | Derivados de indol-2-il-piridin-3-ilo, composicion farmaceutica que los comprende y su uso en medicamentos para el tratamiento de enfermedades mediadas por la sintasa aldosterona. |
WO2010021686A1 (fr) * | 2008-08-18 | 2010-02-25 | Promega Corporation | Composés luminogènes et procédés de détection des enzymes 3a du cytochrome p450 |
UY32126A (es) | 2008-09-25 | 2010-04-30 | Takeda Pharmaceutical | Composición farmacéutica sólida |
EP2351743A4 (fr) | 2008-10-27 | 2012-05-09 | Takeda Pharmaceutical | Composé bicyclique |
WO2010076884A1 (fr) | 2008-12-29 | 2010-07-08 | 武田薬品工業株式会社 | Nouveau composé cyclique condensé et utilisation de celui-ci |
US20120022078A1 (en) * | 2009-04-09 | 2012-01-26 | Msd K.K. | Aryl indole derivatives |
EP2440541A1 (fr) | 2009-06-09 | 2012-04-18 | Takeda Pharmaceutical Company Limited | Nouveau composé cyclique fondu et son utilisation |
CN102548556A (zh) | 2009-07-28 | 2012-07-04 | 武田药品工业株式会社 | 片剂 |
WO2011107494A1 (fr) | 2010-03-03 | 2011-09-09 | Sanofi | Nouveaux dérivés aromatiques de glycoside, médicaments contenants ces composés, et leur utilisation |
NZ603777A (en) | 2010-04-27 | 2013-08-30 | Takeda Pharmaceutical | Bicyclic compound derivatives and their use as acc inhibitors. |
PE20130283A1 (es) | 2010-06-16 | 2013-03-25 | Takeda Pharmaceutical | Cristal de compuesto de amida |
WO2011159781A2 (fr) * | 2010-06-17 | 2011-12-22 | Senomyx, Inc. | Modulateurs de goût amer |
EP2582709B1 (fr) | 2010-06-18 | 2018-01-24 | Sanofi | Dérivés d'azolopyridin-3-one en tant qu'inhibiteurs de lipases et de phospholipases |
US8530413B2 (en) | 2010-06-21 | 2013-09-10 | Sanofi | Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments |
TW201215387A (en) | 2010-07-05 | 2012-04-16 | Sanofi Aventis | Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament |
TW201215388A (en) | 2010-07-05 | 2012-04-16 | Sanofi Sa | (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments |
TW201221505A (en) | 2010-07-05 | 2012-06-01 | Sanofi Sa | Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament |
EP2617726A4 (fr) | 2010-09-17 | 2014-05-14 | Takeda Pharmaceutical | Agent thérapeutique du diabète |
JP5824517B2 (ja) | 2010-11-30 | 2015-11-25 | 武田薬品工業株式会社 | 二環性化合物 |
US8952185B2 (en) | 2011-02-17 | 2015-02-10 | Takeda Pharmaceutical Company Limited | Production method of optically active dihydrobenzofuran derivative |
WO2013037390A1 (fr) | 2011-09-12 | 2013-03-21 | Sanofi | Dérivés amides d'acide 6-(4-hydroxyphényl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylique en tant qu'inhibiteurs de kinase |
EP2760862B1 (fr) | 2011-09-27 | 2015-10-21 | Sanofi | Dérivés d'amide d'acide 6-(4-hydroxyphényl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylique utilisés comme inhibiteurs de kinase |
WO2013057944A1 (fr) * | 2011-10-19 | 2013-04-25 | 興和株式会社 | Nouveau composé de spiroindoline, et agent thérapeutique le contenant |
EP2772485A4 (fr) | 2011-10-24 | 2015-06-10 | Takeda Pharmaceutical | Composé bicyclique |
JP6129850B2 (ja) | 2012-01-12 | 2017-05-17 | 武田薬品工業株式会社 | Mch受容体拮抗剤としてのベンゾイミダゾール誘導体 |
EP2816032A4 (fr) | 2012-02-13 | 2015-09-30 | Takeda Pharmaceutical | Composé à noyaux aromatiques |
JP6095580B2 (ja) | 2012-02-13 | 2017-03-15 | 武田薬品工業株式会社 | 芳香環化合物 |
CN104254322B (zh) | 2012-02-15 | 2017-06-13 | 武田药品工业株式会社 | 片剂 |
US9238639B2 (en) | 2012-02-24 | 2016-01-19 | Takeda Pharmaceutical Company Limited | Aromatic ring compound |
CA2868713A1 (fr) | 2012-03-29 | 2013-10-03 | Takeda Pharmaceutical Company Limited | Compose de type cycle aromatique |
JP6399660B2 (ja) * | 2012-04-10 | 2018-10-03 | ザ・リージエンツ・オブ・ザ・ユニバーシテイー・オブ・カリフオルニア | 癌治療用組成物および方法 |
EP2848621A4 (fr) | 2012-05-10 | 2016-06-01 | Takeda Pharmaceutical | Composé cyclique aromatique |
EP2848622A4 (fr) | 2012-05-10 | 2015-11-04 | Takeda Pharmaceutical | Composé cyclique aromatique |
JP6122879B2 (ja) | 2012-06-05 | 2017-04-26 | 武田薬品工業株式会社 | 固形製剤 |
JP2015127299A (ja) | 2012-07-19 | 2015-07-09 | 武田薬品工業株式会社 | 固形製剤 |
WO2014085486A2 (fr) | 2012-11-30 | 2014-06-05 | Waters Technologies Corporation | Procédés et appareil pour l'analyse de métabolites de la vitamine d |
WO2014142363A1 (fr) | 2013-03-14 | 2014-09-18 | Takeda Pharmaceutical Company Limited | Dérivés de spiro azétidine isoxazole et leur utilisation en tant qu'antagonistes de sstr5 |
WO2014165816A1 (fr) | 2013-04-05 | 2014-10-09 | North Carolina Central University | Composés utiles dans le traitement de troubles métaboliques et leur synthèse |
AR096848A1 (es) | 2013-07-09 | 2016-02-03 | Takeda Pharmaceuticals Co | Derivados de indazol con actividad antagonista del receptor de la hormona concentradora de melanina (mch) |
JP6397410B2 (ja) | 2013-08-09 | 2018-09-26 | 武田薬品工業株式会社 | 芳香環化合物 |
CN105658625B (zh) * | 2013-08-22 | 2019-05-03 | 株式会社Lg化学 | 作为细胞坏死阻碍剂的吲哚酰胺化合物 |
JO3442B1 (ar) | 2013-10-07 | 2019-10-20 | Takeda Pharmaceuticals Co | مضادات ذات نوع فرعي من مستقبل سوماتوستاتين 5 (sstr5) |
US9428470B2 (en) | 2014-02-13 | 2016-08-30 | Takeda Pharmaceutical Company Limited | Heterocyclic compound |
US9346776B2 (en) | 2014-02-13 | 2016-05-24 | Takeda Pharmaceutical Company Limited | Fused heterocyclic compound |
CN104098498A (zh) * | 2014-07-30 | 2014-10-15 | 天津市斯芬克司药物研发有限公司 | 一种吲唑类化合物及其制备方法 |
JOP20180029A1 (ar) | 2017-03-30 | 2019-01-30 | Takeda Pharmaceuticals Co | مركب حلقي غير متجانس |
AR111199A1 (es) | 2017-03-31 | 2019-06-12 | Takeda Pharmaceuticals Co | Compuesto aromático agonista de gpr40 |
JOP20180028A1 (ar) | 2017-03-31 | 2019-01-30 | Takeda Pharmaceuticals Co | مركب ببتيد |
JPWO2018181847A1 (ja) | 2017-03-31 | 2020-03-05 | 武田薬品工業株式会社 | 芳香環化合物 |
IL277495B1 (en) | 2018-03-23 | 2024-04-01 | Carmot Therapeutics Inc | Modulators of protein-coupled receptors - G |
EP3650440A4 (fr) | 2018-08-27 | 2020-11-25 | Scohia Pharma, Inc. | Composé d'ester benzoïque |
EP3856768A2 (fr) | 2018-09-24 | 2021-08-04 | Takeda Pharmaceutical Company Limited | Composés peptidiques agonistes du récepteur du gip et leurs utilisations |
WO2020067575A1 (fr) | 2018-09-24 | 2020-04-02 | Takeda Pharmaceutical Company Limited | Composés peptidiques agonistes du récepteur gip et leurs utilisations |
CN109250963B (zh) * | 2018-09-29 | 2021-07-16 | 福建省昊立建设工程有限公司 | 一种复合增韧混凝土及其制备方法 |
AR121649A1 (es) | 2020-03-25 | 2022-06-22 | Takeda Pharmaceuticals Co | Dosificación qw de compuestos peptídicos agonistas del receptor de gip y sus usos |
MX2022011816A (es) | 2020-03-25 | 2022-10-10 | Takeda Pharmaceuticals Co | Dosificacion qd de compuestos peptidicos agonistas del receptor de gip y sus usos. |
CN113563306B (zh) * | 2020-04-28 | 2022-07-01 | 新发药业有限公司 | 一种2-(4-苯氧基苯基)-6-(哌啶-4-)基烟酰胺的制备方法 |
KR20240007251A (ko) | 2021-05-13 | 2024-01-16 | 카모트 테라퓨틱스, 인크. | G-단백질 결합 수용체의 조절제 |
WO2023169456A1 (fr) | 2022-03-09 | 2023-09-14 | Gasherbrum Bio , Inc. | Agonistes hétérocycliques de glp-1 |
WO2023179542A1 (fr) | 2022-03-21 | 2023-09-28 | Gasherbrum Bio , Inc. | Dérivés de 5,8-dihydro-1,7-naphtyridine utiles en tant qu'agonistes de glp-1 pour le traitement du diabète |
WO2023198140A1 (fr) | 2022-04-14 | 2023-10-19 | Gasherbrum Bio, Inc. | Agonistes hétérocycliques de glp-1 |
Family Cites Families (21)
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FR2656610B1 (fr) | 1989-12-29 | 1992-05-07 | Sanofi Sa | Derives d'amino-2 phenyl-4 thiazole, leur procede de preparation et leur application therapeutique. |
AU683492B2 (en) | 1993-09-10 | 1997-11-13 | Eisai R&D Management Co., Ltd. | Bicyclic heterocyclic sulfonamide and sulfonic ester derivatives |
JP3545461B2 (ja) * | 1993-09-10 | 2004-07-21 | エーザイ株式会社 | 二環式ヘテロ環含有スルホンアミド誘導体 |
WO1997010224A1 (fr) | 1995-09-13 | 1997-03-20 | Takeda Chemical Industries, Ltd. | Composes de benzoxazepine, leur production et leur utilisation en tant qu'agent d'abaissement des niveaux de lipides |
NZ506329A (en) * | 1998-02-25 | 2004-01-30 | Inst Genetics Llc | Inhibitors of phospholipase enzymes |
JP4007743B2 (ja) | 1999-02-26 | 2007-11-14 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | 血管新生阻害剤 |
AR035016A1 (es) | 1999-08-25 | 2004-04-14 | Takeda Chemical Industries Ltd | Composicion de azol promotor de produccion/secrecion de neurotrofina, compuesto prodroga del mismo, composicion farmaceutica que lo comprende y uso del mismo para preparar esta ultima. |
GB0003636D0 (en) * | 2000-02-16 | 2000-04-05 | Smithkline Beecham Plc | Novel compounds |
EP1285651B1 (fr) | 2000-04-28 | 2010-09-01 | Takeda Pharmaceutical Company Limited | Antagonistes de l'hormone concentrant la melanine |
CA2408913A1 (fr) | 2000-05-16 | 2001-11-22 | Takeda Chemical Industries, Ltd. | Antagoniste de l'hormone de concentration de la melanine |
WO2004031179A1 (fr) * | 2002-10-03 | 2004-04-15 | F. Hoffmann-La Roche Ag | Indole-3-carboxamides servant d'activateurs de glucokinase (gk) |
EP1532980A1 (fr) * | 2003-11-24 | 2005-05-25 | Novo Nordisk A/S | Carboxamides d'indole n-heteroarylé et leurs analogues, utiles comme des activateurs de glucokinase pour le traitement de diabetes |
US7498445B2 (en) * | 2004-05-05 | 2009-03-03 | Renopharm Ltd. | Thiazole-based nitric oxide donors capable of releasing two or more nitric oxide molecules and uses thereof |
EP1632491A1 (fr) * | 2004-08-30 | 2006-03-08 | Laboratorios Del Dr. Esteve, S.A. | composes indole substitues et leur utilisation comme modulateurs du recepteur 5-ht6 |
EP2308839B1 (fr) | 2005-04-20 | 2017-03-01 | Takeda Pharmaceutical Company Limited | Composés hétérocycliques condensés |
WO2007037543A1 (fr) | 2005-09-29 | 2007-04-05 | Banyu Pharmaceutical Co., Ltd. | Dérivé de biarylamide |
US7799820B2 (en) | 2005-09-30 | 2010-09-21 | Banyu Pharmaceutical Co., Ltd. | 2-Heterocycle-substituted indole derivatives for treating diabetes and associated conditions |
EP2188291B1 (fr) | 2007-08-14 | 2012-09-19 | Bayer Pharma Aktiengesellschaft | Pyrimidines bicycliques condensées |
KR20100049589A (ko) | 2007-08-14 | 2010-05-12 | 바이엘 쉐링 파마 악티엔게젤샤프트 | 암 치료를 위한 융합된 이미다졸 |
RU2474579C2 (ru) | 2007-10-18 | 2013-02-10 | Янссен Фармацевтика Нв | Тризамещенные 1,2,4-триазолы |
JO2784B1 (en) | 2007-10-18 | 2014-03-15 | شركة جانسين فارماسوتيكا ان. في | 5,3,1 - Triazole substitute derivative |
-
2007
- 2007-10-18 KR KR1020097010151A patent/KR101444486B1/ko not_active IP Right Cessation
- 2007-10-18 MY MYPI20091549A patent/MY158052A/en unknown
- 2007-10-18 WO PCT/JP2007/070772 patent/WO2008050821A1/fr active Application Filing
- 2007-10-18 US US12/311,893 patent/US8410087B2/en not_active Expired - Fee Related
- 2007-10-18 ZA ZA200902585A patent/ZA200902585B/xx unknown
- 2007-10-18 CN CN2007800470664A patent/CN101573357B/zh not_active Expired - Fee Related
- 2007-10-18 TW TW096138971A patent/TWI460176B/zh not_active IP Right Cessation
- 2007-10-18 RU RU2009118602/04A patent/RU2454415C9/ru not_active IP Right Cessation
- 2007-10-18 BR BRPI0717722-4A patent/BRPI0717722A2/pt not_active IP Right Cessation
- 2007-10-18 AU AU2007310064A patent/AU2007310064B2/en not_active Ceased
- 2007-10-18 JP JP2009515658A patent/JP5260507B2/ja not_active Expired - Fee Related
- 2007-10-18 US US11/907,929 patent/US7652133B2/en not_active Expired - Fee Related
- 2007-10-18 CA CA2666973A patent/CA2666973C/fr not_active Expired - Fee Related
- 2007-10-18 MX MX2009003972A patent/MX2009003972A/es active IP Right Grant
- 2007-10-18 GE GEAP200711259A patent/GEP20115241B/en unknown
- 2007-10-18 EP EP07830506A patent/EP2074119A1/fr not_active Withdrawn
- 2007-10-18 UA UAA200904957A patent/UA97257C2/ru unknown
- 2007-10-18 EP EP12170280A patent/EP2508524A3/fr not_active Withdrawn
- 2007-10-18 NZ NZ576570A patent/NZ576570A/en not_active IP Right Cessation
- 2007-10-18 ME MEP-2009-118A patent/ME00681B/fr unknown
-
2008
- 2008-04-10 CL CL2008001017A patent/CL2008001017A1/es unknown
- 2008-04-16 PE PE2008000659A patent/PE20090884A1/es not_active Application Discontinuation
-
2009
- 2009-03-19 US US12/382,622 patent/US7777047B2/en not_active Expired - Fee Related
- 2009-03-19 US US12/382,623 patent/US7718798B2/en not_active Expired - Fee Related
- 2009-04-08 TN TNP2009000129A patent/TN2009000129A1/fr unknown
- 2009-04-16 IL IL198154A patent/IL198154A/en not_active IP Right Cessation
- 2009-04-24 CR CR10748A patent/CR10748A/es unknown
- 2009-05-13 MA MA31871A patent/MA30890B1/fr unknown
- 2009-05-14 EC EC2009009330A patent/ECSP099330A/es unknown
- 2009-05-19 NO NO20091948A patent/NO20091948L/no not_active Application Discontinuation
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MA29323B1 (fr) | Composes de l'acide pyridylacetique | |
MA31169B1 (fr) | Preparation solide comprenant de l'alogliptine et de la pioglitazone | |
MA30911B1 (fr) | Nouveaux derives de sulfonamide en tant qu'antagonistes de bradykinine | |
MA32171B1 (fr) | Compose heterocyclique | |
MA30228B1 (fr) | Pipéridinoylpyrrolidines agonistes du récepteur de mélanocortine de type 4 | |
MA29250B1 (fr) | Cyclohexylamides servant d'antagonistes des recepteurs de dopamine d3, d2 et de 5ht1a | |
TN2009000204A1 (fr) | Spirocetones servant d'inhibiteurs d'acetyl-coa-carboxylase | |
MA30456B1 (fr) | Nouveau dérivé de coumarine présentant une activité anti-tumorale. | |
MA32965B1 (fr) | Derives de sulfonamides | |
MA31710B1 (fr) | (carboxylalkylenephenyl)phényloxamides, procédés pour la production de ceux-ci et utilisation de ceux-ci en tant que medicament | |
MA31419B1 (fr) | Derives de pyridine | |
MA32164B1 (fr) | Derive heterocyclique fusionne et son utilisation | |
TNSN06358A1 (fr) | Methyl-aryl-ou-heteroaryl-amides substitues | |
MA30355B1 (fr) | Derives d'azabicyclo [3. 1. 0] hexyle utilises comme modulateurs des recepteurs de la dopamine d3 | |
MA29926B1 (fr) | Derives de pyrazine | |
TNSN07022A1 (fr) | Derives de pyridine | |
MA30999B1 (fr) | Composés. | |
MA30428B1 (fr) | Derives de dihydropyrazolopyrimidinones | |
MA34713B1 (fr) | Compose bicyclique | |
MA30142B1 (fr) | Agonistes du recepteur de neuropeptide-2 | |
MA27990A1 (fr) | Derives de piperazine pour le traitement d'infections par le vih | |
TNSN07275A1 (fr) | Derives de triazole substitues, servant d'antagonistes d'ocytocine | |
MA30351B1 (fr) | Composes de tetrahydropyridothienopyrimidine et leurs procedes d'utilisation |