FR2735777B1 - Derives de 4-phenylaminothiazole, leur procede de preparation et les compositions pharmaceutiques les contenant - Google Patents
Derives de 4-phenylaminothiazole, leur procede de preparation et les compositions pharmaceutiques les contenantInfo
- Publication number
- FR2735777B1 FR2735777B1 FR9507437A FR9507437A FR2735777B1 FR 2735777 B1 FR2735777 B1 FR 2735777B1 FR 9507437 A FR9507437 A FR 9507437A FR 9507437 A FR9507437 A FR 9507437A FR 2735777 B1 FR2735777 B1 FR 2735777B1
- Authority
- FR
- France
- Prior art keywords
- preparation
- pharmaceutical compositions
- compositions containing
- phenylaminothiazole
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
- A61P5/04—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin for decreasing, blocking or antagonising the activity of the hypothalamic hormones
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
Priority Applications (23)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9507437A FR2735777B1 (fr) | 1995-06-21 | 1995-06-21 | Derives de 4-phenylaminothiazole, leur procede de preparation et les compositions pharmaceutiques les contenant |
PL96324202A PL324202A1 (en) | 1995-06-21 | 1996-06-18 | Derivatives of 4-phenylaminothiazole, method of obtaining them and pharmaceutic compositions containing such derivatives |
TR97/01654T TR199701654T1 (xx) | 1995-06-21 | 1996-06-18 | 4-Fenilaminotiyazol t�revleri. |
EP96922946A EP0833822A1 (fr) | 1995-06-21 | 1996-06-18 | Derives de 4-phenylaminothiazole, leur procede de preparation et les compositions pharmaceutiques les contenant |
KR1019970709640A KR19990028325A (ko) | 1995-06-21 | 1996-06-18 | 치환된 4-페닐아미노티아졸, 이의 제조방법 및 이를 포함하는약학적 조성물 |
AU63627/96A AU710300B2 (en) | 1995-06-21 | 1996-06-18 | Substituted 4-phenylaminothiazoles, their process for preparation and the pharmaceutical compositions containing them |
JP9503616A JP3067807B2 (ja) | 1995-06-21 | 1996-06-18 | 4−フェニルアミノチアゾール誘導体、その製造方法、および該誘導体を含有してなる医薬組成物 |
CZ974103A CZ410397A3 (cs) | 1995-06-21 | 1996-06-18 | Deriváty 4-fenylaminothiazolu, způsob jejich přípravy a farmaceutické přípravky, které je obsahují |
US08/945,098 US5880135A (en) | 1995-06-21 | 1996-06-18 | Substituted 4-phenylaminothiazoles, their process of preparation and the pharmaceutical compositions containing them |
EE9700333A EE9700333A (et) | 1995-06-21 | 1996-06-18 | Substitueeritud 4-fenüülaminotiasoolid, nende valmistamise meetod ja neid sisaldavad farmakoloogilised kompositsioonid |
HU9900056A HUP9900056A2 (hu) | 1995-06-21 | 1996-06-18 | Szubsztituált 4-fenil-amino-tiazol-származékok, eljárás előállításukra és ilyen vegyületeket tartalmazó gyógyászati készítmények |
SK1711-97A SK171197A3 (en) | 1995-06-21 | 1996-06-18 | 4-phenylaminothiazole derivatives, method for preparing same, and pharmaceutical compositions containing said derivatives |
NZ312157A NZ312157A (en) | 1995-06-21 | 1996-06-18 | 4-phenylaminothiazole derivatives, method for preparing same, and pharmaceutical compositions containing said derivatives |
PCT/FR1996/000941 WO1997000868A1 (fr) | 1995-06-21 | 1996-06-18 | Derives de 4-phenylaminothiazole, leur procede de preparation et les compositions pharmaceutiques les contenant |
RU98100764A RU2146253C1 (ru) | 1995-06-21 | 1996-06-18 | Производные 4-фениламинотиазола, способы их получения и фармацевтическая композиция |
BR9609420A BR9609420A (pt) | 1995-06-21 | 1996-06-18 | Derivados de 4-fenilaminotiazol seu processo de preparação e as composições farmacêuticas contendo os mesmos |
IL12229396A IL122293A0 (en) | 1995-06-21 | 1996-06-18 | Substituted 4-phenylaminothiazoles their preparation and pharmaceutical compositions containing them |
CA002222266A CA2222266A1 (fr) | 1995-06-21 | 1996-06-18 | Derives de 4-phenylaminothiazole, leur procede de preparation et les compositions pharmaceutiques les contenant |
ZA9605294A ZA965294B (en) | 1995-06-21 | 1996-06-21 | Substituted 4-phenylaminothiazoles, their process of preparation and the pharmaceutical compositions containing them. |
TW085107427A TW416952B (en) | 1995-06-21 | 1996-07-17 | Substituted 4-phenyl-2-aminothiazoles capable of antgonizing the effects of corticotropin releasing factor (CRF) and their process of preparation |
IS4635A IS4635A (is) | 1995-06-21 | 1997-12-16 | 4-fenýlamínóþíasólafleiður, aðferð við að framleiða þær og lyfjablöndur sem innihalda þær |
MXPA/A/1997/010378A MXPA97010378A (en) | 1995-06-21 | 1997-12-18 | Derivatives of 4-finilaminotiazol, its process of preparation and the pharmaceutical compositions that contains them |
NO975987A NO975987L (no) | 1995-06-21 | 1997-12-19 | 4-Fenylaminotiazol-derivater, fremgangsmåte for fremstilling av disse og farmasöytiske blandinger inneholdende nevnte derivater |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9507437A FR2735777B1 (fr) | 1995-06-21 | 1995-06-21 | Derives de 4-phenylaminothiazole, leur procede de preparation et les compositions pharmaceutiques les contenant |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2735777A1 FR2735777A1 (fr) | 1996-12-27 |
FR2735777B1 true FR2735777B1 (fr) | 1997-09-12 |
Family
ID=9480235
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR9507437A Expired - Lifetime FR2735777B1 (fr) | 1995-06-21 | 1995-06-21 | Derives de 4-phenylaminothiazole, leur procede de preparation et les compositions pharmaceutiques les contenant |
Country Status (22)
Country | Link |
---|---|
US (1) | US5880135A (fr) |
EP (1) | EP0833822A1 (fr) |
JP (1) | JP3067807B2 (fr) |
KR (1) | KR19990028325A (fr) |
AU (1) | AU710300B2 (fr) |
BR (1) | BR9609420A (fr) |
CA (1) | CA2222266A1 (fr) |
CZ (1) | CZ410397A3 (fr) |
EE (1) | EE9700333A (fr) |
FR (1) | FR2735777B1 (fr) |
HU (1) | HUP9900056A2 (fr) |
IL (1) | IL122293A0 (fr) |
IS (1) | IS4635A (fr) |
NO (1) | NO975987L (fr) |
NZ (1) | NZ312157A (fr) |
PL (1) | PL324202A1 (fr) |
RU (1) | RU2146253C1 (fr) |
SK (1) | SK171197A3 (fr) |
TR (1) | TR199701654T1 (fr) |
TW (1) | TW416952B (fr) |
WO (1) | WO1997000868A1 (fr) |
ZA (1) | ZA965294B (fr) |
Families Citing this family (29)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6124289A (en) * | 1996-07-24 | 2000-09-26 | Dupont Pharmaceuticals Co. | Azolo triazines and pyrimidines |
US6191131B1 (en) | 1997-07-23 | 2001-02-20 | Dupont Pharmaceuticals Company | Azolo triazines and pyrimidines |
US6313124B1 (en) | 1997-07-23 | 2001-11-06 | Dupont Pharmaceuticals Company | Tetrazine bicyclic compounds |
US7094782B1 (en) | 1996-07-24 | 2006-08-22 | Bristol-Myers Squibb Company | Azolo triazines and pyrimidines |
US6060478A (en) * | 1996-07-24 | 2000-05-09 | Dupont Pharmaceuticals | Azolo triazines and pyrimidines |
FR2754258B1 (fr) | 1996-10-08 | 1998-12-31 | Sanofi Sa | Derives d'aminothiazole, leur procede de preparation et les compositions pharmaceutiques les contenant |
US6187777B1 (en) * | 1998-02-06 | 2001-02-13 | Amgen Inc. | Compounds and methods which modulate feeding behavior and related diseases |
CN1217945C (zh) | 1998-11-12 | 2005-09-07 | 纽罗克里恩生物科学有限公司 | Crf受体拮抗剂以及与其有关的方法 |
ATE240958T1 (de) | 1998-11-12 | 2003-06-15 | Neurocrine Biosciences Inc | Crf rezeptor-antagonisten und darauf bezogene methoden |
US6531475B1 (en) * | 1998-11-12 | 2003-03-11 | Neurocrine Biosciences, Inc. | CRF receptor antagonists and methods relating thereto |
FR2796380B3 (fr) * | 1999-07-15 | 2001-08-17 | Sanofi Synthelabo | Nouveaux derives d'aminothiazoles, leur preparation et les compositions pharmaceutiques les contenant |
FR2819508B1 (fr) * | 2001-01-12 | 2005-01-21 | Sod Conseils Rech Applic | Derives de 2-arylimino-2, 3-dihydorthiazoles, leurs procedes de preparation et leur utilisation therapeutiques |
US6432989B1 (en) * | 1999-08-27 | 2002-08-13 | Pfizer Inc | Use of CRF antagonists to treat circadian rhythm disorders |
CO5271670A1 (es) * | 1999-10-29 | 2003-04-30 | Pfizer Prod Inc | Antagonistas del factor de liberacion de corticitropina y composiciones relacionadas |
WO2001062718A1 (fr) * | 2000-02-25 | 2001-08-30 | Japan Tobacco, Inc. | Dérivé de benzamide et utilisation de celui-ci |
EP1149583A3 (fr) * | 2000-04-13 | 2001-11-14 | Pfizer Products Inc. | Combinaison des antagonistes de la facteur de la liberation de la corticotropin et des secrétagogues de l hormone de croissance |
DE10045650A1 (de) * | 2000-09-15 | 2002-03-28 | Wuerth Adolf Gmbh & Co Kg | Kunststoffdübel |
US7153871B2 (en) | 2001-01-22 | 2006-12-26 | Memory Pharmaceuticals Corporation | Phosphodiesterase 4 inhibitors, including aminoindazole and aminobenzofuran analogs |
US7205320B2 (en) | 2001-01-22 | 2007-04-17 | Memory Pharmaceuticals Corp. | Phosphodiesterase 4 inhibitors |
EP1423113A4 (fr) * | 2001-08-13 | 2007-04-18 | Phenex Pharmaceuticals Ag | Composes de liaison au recepteur nucleaire nr1h4 |
CA2492907A1 (fr) | 2002-07-19 | 2004-01-29 | Memory Pharmaceuticals Corporation | Inhibiteurs de phosphodiesterase 4 comprenant des analogues de diphenylamine et d'aniline n-substitues |
MXPA05000825A (es) * | 2002-07-19 | 2005-08-29 | Memory Pharm Corp | Compuestos de 6-amino-1h-indazol y 4-aminobenzofurano como inhibidores de fosfodiesterasa 4. |
WO2004046113A2 (fr) * | 2002-11-19 | 2004-06-03 | Memory Pharmaceuticals Corporation | Inhibiteurs de la phosphodiesterase 4 |
US20090048255A1 (en) * | 2003-07-21 | 2009-02-19 | Schumacher Richard A | Phosphodiesterase 4 inhibitors, including n-substituted aniline and diphenylamine analogs |
MY141255A (en) * | 2003-12-11 | 2010-03-31 | Memory Pharm Corp | Phosphodiesterase 4 inhibitors, including n-substituted diarylamine analogs |
ES2389062T3 (es) * | 2006-01-18 | 2012-10-22 | Amgen, Inc | Compuestos de tiazol como inhibidores de proteína cinasa B (PKB) |
US8252333B2 (en) | 2006-01-26 | 2012-08-28 | Jorge Cueto-Garcia | Biodegradable, non-toxic biological adhesive for use in abdominal surgery |
US20100029689A1 (en) * | 2008-07-02 | 2010-02-04 | Memory Pharmaceuticals Corporation | Phosphodiesterase 4 inhibitors |
WO2015166370A1 (fr) | 2014-04-28 | 2015-11-05 | Pfizer Inc. | Composés hétéroaromatiques et leur utilisation en tant que ligands de la dopamine d1 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2612187B1 (fr) * | 1987-03-12 | 1989-07-21 | Sanofi Sa | Derives du thiazole actifs sur le systeme cholinergique, leur procede de preparation et compositions pharmaceutiques en contenant |
FR2656610B1 (fr) * | 1989-12-29 | 1992-05-07 | Sanofi Sa | Derives d'amino-2 phenyl-4 thiazole, leur procede de preparation et leur application therapeutique. |
FR2692893B1 (fr) * | 1992-06-24 | 1994-09-02 | Sanofi Elf | Dérivés alkylamino ramifiés du thiazole, leurs procédés de préparation et les compositions pharmaceutiques qui les contiennent. |
-
1995
- 1995-06-21 FR FR9507437A patent/FR2735777B1/fr not_active Expired - Lifetime
-
1996
- 1996-06-18 EP EP96922946A patent/EP0833822A1/fr not_active Withdrawn
- 1996-06-18 TR TR97/01654T patent/TR199701654T1/xx unknown
- 1996-06-18 EE EE9700333A patent/EE9700333A/xx unknown
- 1996-06-18 NZ NZ312157A patent/NZ312157A/en unknown
- 1996-06-18 PL PL96324202A patent/PL324202A1/xx unknown
- 1996-06-18 KR KR1019970709640A patent/KR19990028325A/ko active IP Right Grant
- 1996-06-18 HU HU9900056A patent/HUP9900056A2/hu unknown
- 1996-06-18 WO PCT/FR1996/000941 patent/WO1997000868A1/fr not_active Application Discontinuation
- 1996-06-18 IL IL12229396A patent/IL122293A0/xx unknown
- 1996-06-18 RU RU98100764A patent/RU2146253C1/ru active
- 1996-06-18 CA CA002222266A patent/CA2222266A1/fr not_active Abandoned
- 1996-06-18 SK SK1711-97A patent/SK171197A3/sk unknown
- 1996-06-18 BR BR9609420A patent/BR9609420A/pt not_active Application Discontinuation
- 1996-06-18 AU AU63627/96A patent/AU710300B2/en not_active Ceased
- 1996-06-18 JP JP9503616A patent/JP3067807B2/ja not_active Expired - Lifetime
- 1996-06-18 US US08/945,098 patent/US5880135A/en not_active Expired - Fee Related
- 1996-06-18 CZ CZ974103A patent/CZ410397A3/cs unknown
- 1996-06-21 ZA ZA9605294A patent/ZA965294B/xx unknown
- 1996-07-17 TW TW085107427A patent/TW416952B/zh active
-
1997
- 1997-12-16 IS IS4635A patent/IS4635A/is unknown
- 1997-12-19 NO NO975987A patent/NO975987L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
CA2222266A1 (fr) | 1997-01-09 |
AU710300B2 (en) | 1999-09-16 |
NO975987D0 (no) | 1997-12-19 |
AU6362796A (en) | 1997-01-22 |
TR199701654T1 (xx) | 1998-05-21 |
NO975987L (no) | 1998-02-19 |
PL324202A1 (en) | 1998-05-11 |
TW416952B (en) | 2001-01-01 |
ZA965294B (en) | 1997-12-22 |
EE9700333A (et) | 1998-06-15 |
IL122293A0 (en) | 1998-04-05 |
IS4635A (is) | 1997-12-16 |
NZ312157A (en) | 1999-04-29 |
CZ410397A3 (cs) | 1998-04-15 |
HUP9900056A2 (hu) | 1999-05-28 |
MX9710378A (es) | 1998-07-31 |
WO1997000868A1 (fr) | 1997-01-09 |
EP0833822A1 (fr) | 1998-04-08 |
FR2735777A1 (fr) | 1996-12-27 |
JPH10511693A (ja) | 1998-11-10 |
KR19990028325A (ko) | 1999-04-15 |
SK171197A3 (en) | 1998-08-05 |
RU2146253C1 (ru) | 2000-03-10 |
BR9609420A (pt) | 1999-05-18 |
JP3067807B2 (ja) | 2000-07-24 |
US5880135A (en) | 1999-03-09 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
TP | Transmission of property |