IL158485A0 - Spiropyrazole compounds - Google Patents

Spiropyrazole compounds

Info

Publication number: IL158485A0
Authority: IL; Israel
Prior art keywords: spiropyrazole; compounds; spiropyrazole compounds; whereinz; compound
Prior art date: 2001-04-18

Application number

IL15848502A

Other languages

English (en)

Original Assignee

Euro Celtique Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-04-18

Filing date

2002-04-18

Publication date

2004-05-12

2002-04-18 Application filed by Euro Celtique Sa filed Critical Euro Celtique Sa

2004-05-12 Publication of IL158485A0 publication Critical patent/IL158485A0/xx

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/10—Spiro-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Neurosurgery (AREA)
Engineering & Computer Science (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Bioinformatics & Cheminformatics (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Dental Preparations (AREA)
Solid-Sorbent Or Filter-Aiding Compositions (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

IL15848502A 2001-04-18 2002-04-18 Spiropyrazole compounds IL158485A0 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US28467501P	2001-04-18	2001-04-18
PCT/US2002/012376 WO2002085355A1 (en)	2001-04-18	2002-04-18	Spiropyrazole compounds

Publications (1)

Publication Number	Publication Date
IL158485A0 true IL158485A0 (en)	2004-05-12

Family

ID=23091099

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
IL15848502A IL158485A0 (en)	2001-04-18	2002-04-18	Spiropyrazole compounds
IL158485A IL158485A (en)	2001-04-18	2003-10-19	Spiropyrazole compounds

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
IL158485A IL158485A (en)	2001-04-18	2003-10-19	Spiropyrazole compounds

Country Status (28)

Country	Link
US (2)	US6635653B2 (hu)
EP (1)	EP1385515B1 (hu)
JP (1)	JP4342181B2 (hu)
KR (1)	KR100628292B1 (hu)
CN (1)	CN1516584A (hu)
AT (1)	ATE403429T1 (hu)
AU (1)	AU2002311833B2 (hu)
BR (1)	BR0209127A (hu)
CA (1)	CA2444634C (hu)
CY (1)	CY1108454T1 (hu)
CZ (1)	CZ20032849A3 (hu)
DE (1)	DE60228071D1 (hu)
DK (1)	DK1385515T3 (hu)
ES (1)	ES2312584T3 (hu)
HK (1)	HK1062885A1 (hu)
HU (1)	HUP0401333A3 (hu)
IL (2)	IL158485A0 (hu)
MX (1)	MXPA03009604A (hu)
NO (1)	NO20034660L (hu)
NZ (1)	NZ528978A (hu)
PL (1)	PL367263A1 (hu)
PT (1)	PT1385515E (hu)
RU (1)	RU2299883C2 (hu)
SI (1)	SI1385515T1 (hu)
UA (1)	UA74439C2 (hu)
WO (1)	WO2002085355A1 (hu)
YU (1)	YU82403A (hu)
ZA (1)	ZA200308103B (hu)

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US20040242583A1 (en) *	2003-01-20	2004-12-02	Aventis Pharma Deutschland Gmbh	Pyrimido[5,4-e][1,2,4]triazine-5,7-diones, processes for preparing them and their use
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US20100009929A1 (en)	2004-03-29	2010-01-14	Cheng Jin Q	Compositions including triciribine and bortezomib and derivatives thereof and methods of use thereof
US20100009928A1 (en)	2004-03-29	2010-01-14	Cheng Jin Q	Compositions including triciribine and taxanes and methods of use thereof
US20100028339A1 (en) *	2004-03-29	2010-02-04	Cheng Jin Q	Compositions including triciribine and trastuzumab and methods of use thereof
US20100173864A1 (en)	2004-03-29	2010-07-08	Cheng Jin Q	Compositions including triciribine and one or more platinum compounds and methods of use thereof
PL2574341T3 (pl)	2004-03-29	2017-09-29	University Of South Florida	Efektywne leczenie guzów i raka fosforanem tricyrybiny
JP5078869B2 (ja)	2005-03-08	2012-11-21	ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ	ニューロキニン（ｎｋ１）拮抗物質としてのジアザ−スピロ−［４．４］−ノナン誘導体
CN1870631B (zh) *	2005-11-11	2010-04-14	华为技术有限公司	媒体网关的门控方法
US20080051380A1 (en)	2006-08-25	2008-02-28	Auerbach Alan H	Methods and compositions for treating cancer
CN103202840B (zh)	2006-11-28	2015-02-11	詹森药业有限公司	3-(3-氨基-2-(r)-羟基-丙基)-1-(4-氟-苯基)-8-(8-甲基-萘-1-基甲基)-1,3,8-三氮杂-螺[4.5]癸烷-4-酮的盐
SI2076506T1 (sl) *	2007-01-16	2011-01-31	Purdue Pharma Lp	Heterociklično substituirani piperidini kot ORL-1 ligandi
CN101679430B (zh)	2007-04-09	2013-12-25	詹森药业有限公司	用于治疗焦虑和抑郁症的作为orl-1受体的配体的1,3,8-三取代-1,3,8-三氮杂-螺[4.5]癸-4-酮衍生物
EP2433936A1 (en)	2007-08-31	2012-03-28	Purdue Pharma LP	Substituted-quinoxaline-type-piperidine compounds and the uses thereof
MX2011000872A (es)	2008-07-21	2011-07-29	Purdue Pharma Lp	Compuestos de piperidina puenteada tipo quinoxalina sustituida y los usos de los mismos.
UA107943C2 (en) *	2009-11-16	2015-03-10	Lilly Co Eli	Compounds of spiropiperidines as antagonists of the orl-1 receptors
AU2011346749A1 (en)	2010-12-22	2013-05-02	Purdue Pharma L.P.	Phosphorus-substituted quinoxaline-type piperidine compounds and uses thereof
US9290488B2 (en)	2011-12-01	2016-03-22	Purdue Pharma L.P.	Azetidine-substituted quinoxalines as opioid receptor like-1 modulators
US9085561B2 (en)	2012-07-30	2015-07-21	Purdue Pharma L.P.	Cyclic urea- or lactam-substituted quinoxaline-type piperidines as ORL-1 modulators
US9951038B2 (en)	2012-12-27	2018-04-24	Purdue Pharma L.P.	Quinazolin-4(3H)-one-type piperidine compounds and uses thereof
WO2014102592A2 (en)	2012-12-27	2014-07-03	Purdue Pharma L.P.	Oxime/substituted quinoxaline-type piperidine compounds and uses thereof
WO2014102588A2 (en)	2012-12-27	2014-07-03	Purdue Pharma L.P.	Indole and indoline-type piperidine compounds and uses thereof
WO2014102594A2 (en)	2012-12-27	2014-07-03	Purdue Pharma L.P.	Substituted benzimidazole-type piperidine compounds and uses thereof
WO2014102590A1 (en)	2012-12-27	2014-07-03	Purdue Pharma L.P.	Substituted piperidin-4-amino-type compounds and uses thereof
US20180028521A1 (en)	2016-07-29	2018-02-01	Janssen Pharmaceutica Nv	Methods of Treating Prostate Cancer
CN111825681A (zh) *	2020-07-07	2020-10-27	扬州大学	一种合成(e)-亚苄基螺吡唑吡咯嗪酮类化合物的方法

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2002
- 2002-04-18 AU AU2002311833A patent/AU2002311833B2/en not_active Ceased
- 2002-04-18 MX MXPA03009604A patent/MXPA03009604A/es active IP Right Grant
- 2002-04-18 HU HU0401333A patent/HUP0401333A3/hu unknown
- 2002-04-18 JP JP2002582928A patent/JP4342181B2/ja not_active Expired - Fee Related
- 2002-04-18 CN CNA028121767A patent/CN1516584A/zh active Pending
- 2002-04-18 RU RU2003133455/04A patent/RU2299883C2/ru not_active IP Right Cessation
- 2002-04-18 IL IL15848502A patent/IL158485A0/xx unknown
- 2002-04-18 CZ CZ20032849A patent/CZ20032849A3/cs unknown
- 2002-04-18 WO PCT/US2002/012376 patent/WO2002085355A1/en not_active Application Discontinuation
- 2002-04-18 PL PL02367263A patent/PL367263A1/xx not_active Application Discontinuation
- 2002-04-18 ES ES02739163T patent/ES2312584T3/es not_active Expired - Lifetime
- 2002-04-18 DK DK02739163T patent/DK1385515T3/da active
- 2002-04-18 SI SI200230748T patent/SI1385515T1/sl unknown
- 2002-04-18 YU YU82403A patent/YU82403A/sh unknown
- 2002-04-18 PT PT02739163T patent/PT1385515E/pt unknown
- 2002-04-18 AT AT02739163T patent/ATE403429T1/de active
- 2002-04-18 EP EP02739163A patent/EP1385515B1/en not_active Expired - Lifetime
- 2002-04-18 NZ NZ528978A patent/NZ528978A/en not_active IP Right Cessation
- 2002-04-18 KR KR1020037013821A patent/KR100628292B1/ko not_active IP Right Cessation
- 2002-04-18 DE DE60228071T patent/DE60228071D1/de not_active Expired - Lifetime
- 2002-04-18 CA CA2444634A patent/CA2444634C/en not_active Expired - Fee Related
- 2002-04-18 BR BRPI0209127-5A patent/BR0209127A/pt not_active Application Discontinuation
- 2002-04-18 US US10/126,506 patent/US6635653B2/en not_active Expired - Lifetime
- 2002-04-18 UA UA20031110381A patent/UA74439C2/uk unknown
2003
- 2003-06-19 US US10/601,174 patent/US20040087641A1/en not_active Abandoned
- 2003-10-17 ZA ZA200308103A patent/ZA200308103B/en unknown
- 2003-10-17 NO NO20034660A patent/NO20034660L/no not_active Application Discontinuation
- 2003-10-19 IL IL158485A patent/IL158485A/en not_active IP Right Cessation
2004
- 2004-08-03 HK HK04105726.6A patent/HK1062885A1/xx not_active IP Right Cessation
2008
- 2008-10-27 CY CY20081101206T patent/CY1108454T1/el unknown

Also Published As

Publication number	Publication date
CA2444634C (en)	2011-06-07
WO2002085355A1 (en)	2002-10-31
NO20034660L (no)	2003-12-17
CN1516584A (zh)	2004-07-28
US6635653B2 (en)	2003-10-21
MXPA03009604A (es)	2004-04-02
CA2444634A1 (en)	2002-10-31
RU2299883C2 (ru)	2007-05-27
AU2002311833B2 (en)	2005-04-28
HK1062885A1 (en)	2004-12-03
DE60228071D1 (de)	2008-09-18
ES2312584T3 (es)	2009-03-01
NO20034660D0 (no)	2003-10-17
EP1385515B1 (en)	2008-08-06
US20040087641A1 (en)	2004-05-06
US20030027834A1 (en)	2003-02-06
JP4342181B2 (ja)	2009-10-14
DK1385515T3 (da)	2008-10-27
EP1385515A1 (en)	2004-02-04
HUP0401333A2 (hu)	2004-10-28
ZA200308103B (en)	2004-10-18
ATE403429T1 (de)	2008-08-15
HUP0401333A3 (en)	2004-11-29
JP2004531531A (ja)	2004-10-14
CY1108454T1 (el)	2014-04-09
EP1385515A4 (en)	2004-06-30
NZ528978A (en)	2004-06-25
KR100628292B1 (ko)	2006-09-27
PT1385515E (pt)	2008-09-15
SI1385515T1 (sl)	2008-12-31
CZ20032849A3 (en)	2004-03-17
KR20040008159A (ko)	2004-01-28
PL367263A1 (en)	2005-02-21
UA74439C2 (uk)	2005-12-15
BR0209127A (pt)	2006-03-21
YU82403A (sh)	2006-08-17
IL158485A (en)	2009-09-01
RU2003133455A (ru)	2005-05-10

Publication	Publication Date	Title
HK1062885A1 (en)	2004-12-03	Spiropyrazole compounds
YU82303A (sh)	2006-03-03	Analozi nociceptina
RS51444B (sr)	2011-04-30	JEDINJENJA KOJA SADRŽE LAKTAM I NJIHOVI DERIVATI KAO INHIBITORI FAKTORA Xa
MY126559A (en)	2006-10-31	Fungicidal 2-methoxybenzophenones
MY134892A (en)	2007-12-31	Substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines and their use
DE60229736D1 (de)	2008-12-18	Spiroinden- und spiroindan-verbindungen
DE60214392D1 (de)	2006-10-12	1,4-disubstituierte benzokondensierte cycloalkyl harnstoffverbindungen
WO2003006425A3 (en)	2003-11-27	Novel compounds as anti-inflammatory, immunomodulatory and anti-proliferatory agents
GB0124627D0 (en)	2001-12-05	Novel compounds
MXPA02003977A (es)	2003-09-25	Inhibidores de adhesion de celula mediada por al°2.
MXPA04003886A (es)	2004-07-08	Tiofen- y tiazolsulfonamidas como agentes antineoplasticos.
MXPA03009602A (es)	2004-04-02	Analogos de nociceptina.
SE0004245D0 (sv)	2000-11-20	Novel compounds and their use
PT1975164E (pt)	2010-04-20	Compostos de octa-hidrobenzimidazolona utilizados como analgésicos
AU2003268342A8 (en)	2004-03-19	Antimicrobial compositions
EP1671948A4 (en)	2007-03-14	CINNAMOYL COMPOUND AND USE THEREOF
EP1671961A4 (en)	2009-04-01	CINNAMOYL COMPOUND AND USE THEREOF
MXPA05006450A (es)	2005-08-19	Nuevo derivado de 2,4-diamino-1,3,5-triazina.
ES2183709A1 (es)	2003-03-16	Composicion para el control de artropodos.
IL152632A0 (en)	2003-06-24	Trimethyldecenyl compounds
MXPA05003881A (es)	2005-10-05	Preparacion de compuestos triazospiro.
SE9901062D0 (sv)	1999-03-23	Use for conifer sapling protection
RS20050026A (en)	2007-08-03	Novel benzohydrazide derivatives as herbicides and desiccant compositions contaning them
IT1317718B1 (it)	2003-07-15	Benzilisotiouree ad attivita' fungicida.