FI114475B - Menetelmä uusien terapeuttisesti käyttökelpoisten kinuklidiinijohdannaisten valmistamiseksi - Google Patents

Menetelmä uusien terapeuttisesti käyttökelpoisten kinuklidiinijohdannaisten valmistamiseksi Download PDF

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Publication number
FI114475B
FI114475B FI935297A FI935297A FI114475B FI 114475 B FI114475 B FI 114475B FI 935297 A FI935297 A FI 935297A FI 935297 A FI935297 A FI 935297A FI 114475 B FI114475 B FI 114475B
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FI
Finland
Prior art keywords
formula
methyl
azabicyclo
diphenylmethyl
methoxyphenyl
Prior art date
Application number
FI935297A
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English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI935297A (fi
FI935297A0 (fi
Inventor
Masami Nakane
Hiroshi Kondo
Kaoru Shimada
Iii John A Lowe
Terry J Rosen
Fimitaka Ito
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=24845673&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI114475(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of FI935297A publication Critical patent/FI935297A/fi
Publication of FI935297A0 publication Critical patent/FI935297A0/fi
Application granted granted Critical
Publication of FI114475B publication Critical patent/FI114475B/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Anesthesiology (AREA)
  • Psychiatry (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI935297A 1991-05-31 1993-11-29 Menetelmä uusien terapeuttisesti käyttökelpoisten kinuklidiinijohdannaisten valmistamiseksi FI114475B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US70840491A 1991-05-31 1991-05-31
US70840491 1991-05-31
US9203317 1992-04-28
PCT/US1992/003317 WO1992021677A1 (en) 1991-05-31 1992-04-28 bibNUCLIDINE DERIVATIVES

Publications (3)

Publication Number Publication Date
FI935297A FI935297A (fi) 1993-11-29
FI935297A0 FI935297A0 (fi) 1993-11-29
FI114475B true FI114475B (fi) 2004-10-29

Family

ID=24845673

Family Applications (1)

Application Number Title Priority Date Filing Date
FI935297A FI114475B (fi) 1991-05-31 1993-11-29 Menetelmä uusien terapeuttisesti käyttökelpoisten kinuklidiinijohdannaisten valmistamiseksi

Country Status (41)

Country Link
US (3) US5807867A (pl)
EP (1) EP0587723B1 (pl)
JP (2) JPH0733386B2 (pl)
KR (1) KR100214905B1 (pl)
CN (1) CN1048492C (pl)
AP (1) AP299A (pl)
AT (1) ATE135006T1 (pl)
AU (1) AU657552B2 (pl)
BG (1) BG61694B1 (pl)
BR (1) BR9206073A (pl)
CA (1) CA2102179C (pl)
CZ (1) CZ281403B6 (pl)
DE (4) DE122006000066I2 (pl)
DK (1) DK0587723T3 (pl)
EG (1) EG19944A (pl)
ES (1) ES2084361T3 (pl)
FI (1) FI114475B (pl)
GR (1) GR3019687T3 (pl)
GT (1) GT199200028A (pl)
HU (1) HU217548B (pl)
IE (1) IE72473B1 (pl)
IL (1) IL102008A (pl)
IS (1) IS1611B (pl)
LU (1) LU91293I2 (pl)
MA (1) MA22539A1 (pl)
MX (1) MX9202554A (pl)
NL (1) NL300250I2 (pl)
NO (2) NO302701B1 (pl)
NZ (2) NZ242956A (pl)
OA (1) OA09867A (pl)
PL (1) PL171379B1 (pl)
PT (1) PT100546B (pl)
RO (1) RO110499B1 (pl)
RU (1) RU2103269C1 (pl)
SK (1) SK390692A3 (pl)
TW (1) TW204349B (pl)
UA (1) UA27776C2 (pl)
UY (1) UY23422A1 (pl)
WO (1) WO1992021677A1 (pl)
YU (1) YU48995B (pl)
ZA (1) ZA923942B (pl)

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CA2102179C (en) 1998-10-27
BG61694B1 (bg) 1998-03-31
CZ281403B6 (cs) 1996-09-11
ZA923942B (en) 1993-11-29
PT100546B (pt) 1999-12-31
GT199200028A (es) 1993-11-20
IS3871A (is) 1992-12-02
DE122006000066I2 (de) 2007-12-06
AP9200384A0 (en) 1992-07-31
HU217548B (hu) 2000-02-28
IL102008A0 (en) 1992-12-30
DE69208877T2 (de) 1996-07-25
DE9290063U1 (de) 1994-02-24
CA2102179A1 (en) 1992-12-01
NZ270673A (en) 1997-07-27
CN1048492C (zh) 2000-01-19
FI935297A (fi) 1993-11-29
BR9206073A (pt) 1994-12-06
JPH0733386B2 (ja) 1995-04-12
LU91293I2 (fr) 2007-02-06
OA09867A (en) 1994-08-15
RU2103269C1 (ru) 1998-01-27
JPH06504292A (ja) 1994-05-19
ATE135006T1 (de) 1996-03-15
MA22539A1 (fr) 1992-12-31
NO2007003I2 (no) 2011-04-18
JPH07285965A (ja) 1995-10-31
MX9202554A (es) 1992-11-01
AU657552B2 (en) 1995-03-16
AP299A (en) 1994-01-14
YU56492A (sh) 1995-03-27
SK278788B6 (sk) 1998-02-04
DK0587723T3 (da) 1996-04-01
EG19944A (en) 1997-02-27
EP0587723A1 (en) 1994-03-23
IE72473B1 (en) 1997-04-23
PL171379B1 (en) 1997-04-30
NO934312D0 (no) 1993-11-29
AU1990192A (en) 1993-01-08
NL300250I1 (nl) 2007-02-01
US6222038B1 (en) 2001-04-24
WO1992021677A1 (en) 1992-12-10
NL300250I2 (nl) 2007-03-01
DE69208877D1 (de) 1996-04-11
NO934312L (no) 1993-11-29
US5807867A (en) 1998-09-15
US5939433A (en) 1999-08-17
TW204349B (pl) 1993-04-21
CZ390692A3 (en) 1994-02-16
JP2645225B2 (ja) 1997-08-25
ES2084361T3 (es) 1996-05-01
PT100546A (pt) 1993-08-31
FI935297A0 (fi) 1993-11-29
EP0587723B1 (en) 1996-03-06
HU9303393D0 (en) 1994-03-28
SK390692A3 (en) 1998-02-04
DE122006000066I1 (de) 2007-03-22
HUT70151A (en) 1995-09-28
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RO110499B1 (ro) 1996-01-30
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NZ242956A (en) 1995-06-27
BG98248A (bg) 1994-07-29
UY23422A1 (es) 1992-11-12
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CN1067428A (zh) 1992-12-30

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