EA201591340A1 - Модулятор андрогенного рецептора и его применения - Google Patents

Модулятор андрогенного рецептора и его применения

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Publication number
EA201591340A1
EA201591340A1 EA201591340A EA201591340A EA201591340A1 EA 201591340 A1 EA201591340 A1 EA 201591340A1 EA 201591340 A EA201591340 A EA 201591340A EA 201591340 A EA201591340 A EA 201591340A EA 201591340 A1 EA201591340 A1 EA 201591340A1
Authority
EA
Eurasian Patent Office
Prior art keywords
androgen receptor
modulator
applications
treatment
receptor modulator
Prior art date
Application number
EA201591340A
Other languages
English (en)
Other versions
EA035125B1 (ru
Inventor
Исан Чэнь
Джеффри Х. Хэджер
Эдна Чоу Маневал
Марк Р. Херберт
Николас Д. Смит
Original Assignee
Арагон Фармасьютикалз, Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=50029265&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA201591340(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Арагон Фармасьютикалз, Инк. filed Critical Арагон Фармасьютикалз, Инк.
Publication of EA201591340A1 publication Critical patent/EA201591340A1/ru
Publication of EA035125B1 publication Critical patent/EA035125B1/ru

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    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4025—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
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Abstract

В заявке описан модулятор андрогенного рецептора формулы (I)при лечении рака предстательной железы в комбинации с другими методами лечения и при лечении заболеваний или состояний, которые поддаются лечению модулятором андрогенного рецептора, а также фармацевтические композиции и лекарственные средства, включающие такое соединение.
EA201591340A 2013-01-15 2014-01-09 Способ лечения рака предстательной железы с использованием комбинации на основе модулятора андрогенного рецептора EA035125B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361752842P 2013-01-15 2013-01-15
PCT/US2014/010777 WO2014113260A1 (en) 2013-01-15 2014-01-09 Androgen receptor modulator and uses thereof

Publications (2)

Publication Number Publication Date
EA201591340A1 true EA201591340A1 (ru) 2015-12-30
EA035125B1 EA035125B1 (ru) 2020-04-29

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ID=50029265

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Application Number Title Priority Date Filing Date
EA201591340A EA035125B1 (ru) 2013-01-15 2014-01-09 Способ лечения рака предстательной железы с использованием комбинации на основе модулятора андрогенного рецептора
EA201991772A EA201991772A1 (ru) 2013-01-15 2014-01-09 Способ лечения рака предстательной железы с использованием комбинации на основе модулятора андрогенного рецептора

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