EA201170300A1 - Кристаллические формы пиридинового производного - Google Patents
Кристаллические формы пиридинового производногоInfo
- Publication number
- EA201170300A1 EA201170300A1 EA201170300A EA201170300A EA201170300A1 EA 201170300 A1 EA201170300 A1 EA 201170300A1 EA 201170300 A EA201170300 A EA 201170300A EA 201170300 A EA201170300 A EA 201170300A EA 201170300 A1 EA201170300 A1 EA 201170300A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- crystal forms
- pyridine derivative
- solvate
- therapy
- compound
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5383—1,4-Oxazines, e.g. morpholine ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
Изобретение относится к 4-метилбензолсульфонатной соли соединения формулы (I)в кристаллической форме или ее сольвату, фармацевтическим препаратам, содержащим их, и их использованию в терапии, и способам их получения.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0814340.6A GB0814340D0 (en) | 2008-08-05 | 2008-08-05 | Anhydrous crystol form fo a pyridine derivative |
PCT/EP2009/060089 WO2010015626A1 (en) | 2008-08-05 | 2009-08-04 | Crystalline forms of a pyridine derivative |
Publications (1)
Publication Number | Publication Date |
---|---|
EA201170300A1 true EA201170300A1 (ru) | 2011-08-30 |
Family
ID=39767571
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201170300A EA201170300A1 (ru) | 2008-08-05 | 2009-08-04 | Кристаллические формы пиридинового производного |
Country Status (14)
Country | Link |
---|---|
US (1) | US8093242B2 (ru) |
EP (1) | EP2321324A1 (ru) |
JP (1) | JP2011529942A (ru) |
KR (1) | KR20110052686A (ru) |
CN (1) | CN102171219A (ru) |
AU (1) | AU2009279135B2 (ru) |
BR (1) | BRPI0917224A2 (ru) |
CA (1) | CA2733235A1 (ru) |
EA (1) | EA201170300A1 (ru) |
GB (1) | GB0814340D0 (ru) |
IL (1) | IL210777A0 (ru) |
MX (1) | MX2011001414A (ru) |
WO (1) | WO2010015626A1 (ru) |
ZA (1) | ZA201100426B (ru) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2440938T3 (es) * | 2009-08-27 | 2014-01-31 | Nerre Therapeutics Limited | Formas anhidrato de un derivado de piridina |
JP6902682B2 (ja) * | 2015-05-18 | 2021-07-14 | カンディー セラピューティクス リミテッド | 性ホルモン依存性疾患を治療するためのnk−1/nk−3受容体デュアルアンタゴニスト |
DK3765024T3 (da) | 2018-03-14 | 2024-02-12 | Kandy Therapeutics Ltd | Hidtil ukendt farmaceutisk formulering, som omfatter dobbelte nk-1/nk-3-receptor-antagonister |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2000514455A (ja) | 1996-07-17 | 2000-10-31 | メルク エンド カンパニー インコーポレーテッド | タキキニンアンタゴニストによるサーカディアンリズムの改変 |
ATE277905T1 (de) * | 1999-02-24 | 2004-10-15 | Hoffmann La Roche | 4-phenylpyridinderivate und deren verwendung als nk-1 rezeptorantagonisten |
AU7788500A (en) | 1999-10-25 | 2001-05-08 | Janssen Pharmaceutica N.V. | Use of substance p antagonists for influencing the circadian timing system |
GB0203022D0 (en) | 2002-02-08 | 2002-03-27 | Glaxo Group Ltd | Chemical compounds |
GB0203020D0 (en) | 2002-02-08 | 2002-03-27 | Glaxo Group Ltd | Chemical compounds |
TW200403058A (en) | 2002-04-19 | 2004-03-01 | Bristol Myers Squibb Co | Heterocyclo inhibitors of potassium channel function |
CN1852712B (zh) * | 2003-07-03 | 2010-06-09 | 弗·哈夫曼-拉罗切有限公司 | 用于治疗精神***症的双重nk1/nk3拮抗剂 |
ATE505472T1 (de) * | 2005-09-09 | 2011-04-15 | Glaxosmithkline Llc | Pyridinderivate und ihre verwendung bei der behandlung psychotischer erkrankungen |
-
2008
- 2008-08-05 GB GBGB0814340.6A patent/GB0814340D0/en not_active Ceased
-
2009
- 2009-08-04 CA CA2733235A patent/CA2733235A1/en not_active Abandoned
- 2009-08-04 EP EP09781468A patent/EP2321324A1/en not_active Withdrawn
- 2009-08-04 WO PCT/EP2009/060089 patent/WO2010015626A1/en active Application Filing
- 2009-08-04 AU AU2009279135A patent/AU2009279135B2/en not_active Ceased
- 2009-08-04 MX MX2011001414A patent/MX2011001414A/es unknown
- 2009-08-04 US US13/056,775 patent/US8093242B2/en active Active
- 2009-08-04 CN CN2009801393221A patent/CN102171219A/zh active Pending
- 2009-08-04 EA EA201170300A patent/EA201170300A1/ru unknown
- 2009-08-04 KR KR1020117005159A patent/KR20110052686A/ko not_active Application Discontinuation
- 2009-08-04 JP JP2011521561A patent/JP2011529942A/ja not_active Withdrawn
- 2009-08-04 BR BRPI0917224A patent/BRPI0917224A2/pt not_active IP Right Cessation
-
2011
- 2011-01-17 ZA ZA2011/00426A patent/ZA201100426B/en unknown
- 2011-01-20 IL IL210777A patent/IL210777A0/en unknown
Also Published As
Publication number | Publication date |
---|---|
JP2011529942A (ja) | 2011-12-15 |
IL210777A0 (en) | 2011-03-31 |
BRPI0917224A2 (pt) | 2015-11-24 |
CN102171219A (zh) | 2011-08-31 |
EP2321324A1 (en) | 2011-05-18 |
AU2009279135B2 (en) | 2012-09-13 |
US8093242B2 (en) | 2012-01-10 |
US20110136798A1 (en) | 2011-06-09 |
CA2733235A1 (en) | 2010-02-11 |
ZA201100426B (en) | 2012-03-28 |
MX2011001414A (es) | 2011-04-04 |
KR20110052686A (ko) | 2011-05-18 |
GB0814340D0 (en) | 2008-09-10 |
AU2009279135A1 (en) | 2010-02-11 |
WO2010015626A1 (en) | 2010-02-11 |
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