EA200400816A1 - Замещенные аналоги хиназолин-4-иламина в качестве модуляторов капсаицина - Google Patents

Замещенные аналоги хиназолин-4-иламина в качестве модуляторов капсаицина

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Publication number
EA200400816A1
EA200400816A1 EA200400816A EA200400816A EA200400816A1 EA 200400816 A1 EA200400816 A1 EA 200400816A1 EA 200400816 A EA200400816 A EA 200400816A EA 200400816 A EA200400816 A EA 200400816A EA 200400816 A1 EA200400816 A1 EA 200400816A1
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Prior art keywords
capsaicin
modulators
hinazolin
ilamine
analogues
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EA200400816A
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English (en)
Inventor
Раджагопал Бактхаваткхалам
Чарлз А. Блам
Харри Л. Брилманн
Тимоти М. Колдуэлл
Стефан Де Ломбер
Кевин Дж. Ходжеттс
Тэйянг Юн
Ксяожанг Женг
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Ньюроджин Корпорейшн
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Application filed by Ньюроджин Корпорейшн filed Critical Ньюроджин Корпорейшн
Publication of EA200400816A1 publication Critical patent/EA200400816A1/ru

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Abstract

В общем, данное изобретение относится к замещенным аналогам хиназолин-4-иламина, которые являются модуляторами капсаициновых рецепторов, и к применению таких соединений для лечения состояний, связанных с активацией капсаициновых рецепторов. Данное изобретение относится также к использованию таких соединений в качестве зондов для детектирования и локализирования капсаициновых рецепторов.Отчет о международном поиске был опубликован 2003.09.04.
EA200400816A 2002-01-17 2003-01-17 Замещенные аналоги хиназолин-4-иламина в качестве модуляторов капсаицина EA200400816A1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US34992002P 2002-01-17 2002-01-17
US35052702P 2002-01-22 2002-01-22
PCT/US2003/001563 WO2003062209A2 (en) 2002-01-17 2003-01-17 Substituted quinazolin-4-ylamine analogues as modulators of capsaicin

Publications (1)

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EA200400816A1 true EA200400816A1 (ru) 2005-02-24

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EA200400816A EA200400816A1 (ru) 2002-01-17 2003-01-17 Замещенные аналоги хиназолин-4-иламина в качестве модуляторов капсаицина

Country Status (15)

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US (3) US7074799B2 (ru)
EP (1) EP1471910A2 (ru)
JP (1) JP2005526714A (ru)
KR (1) KR20040085151A (ru)
CN (1) CN1627944A (ru)
BR (1) BR0306982A (ru)
CA (1) CA2473796A1 (ru)
EA (1) EA200400816A1 (ru)
HU (1) HUP0500200A2 (ru)
MX (1) MXPA04006882A (ru)
NO (1) NO20043411L (ru)
PL (1) PL371587A1 (ru)
RS (1) RS63204A (ru)
TW (1) TW200406390A (ru)
WO (1) WO2003062209A2 (ru)

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