DK2298743T3 - p38-Kinaseinhibitorer på grundlag af en 5-leddet heterocyclisk ring - Google Patents

p38-Kinaseinhibitorer på grundlag af en 5-leddet heterocyclisk ring

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Publication number
DK2298743T3
DK2298743T3 DK10164367.4T DK10164367T DK2298743T3 DK 2298743 T3 DK2298743 T3 DK 2298743T3 DK 10164367 T DK10164367 T DK 10164367T DK 2298743 T3 DK2298743 T3 DK 2298743T3
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Prior art keywords
basis
kinase inhibitors
kinase
heterocyclic ring
membered heterocyclic
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Application number
DK10164367.4T
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English (en)
Inventor
Olga M Fryszman
Hengyuan Lang
Jiong Lan
Edcon Chang
Yunfeng Fang
Original Assignee
Novartis Ag
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Publication of DK2298743T3 publication Critical patent/DK2298743T3/da

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/10—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
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MY158162A (en) 2016-09-15
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JP2007521278A (ja) 2007-08-02
US20130172352A1 (en) 2013-07-04
JP4838121B2 (ja) 2011-12-14
IS2916B (is) 2014-12-15
US8242117B2 (en) 2012-08-14
PT1641764E (pt) 2011-10-27
SI1641764T1 (sl) 2011-11-30
US20050049288A1 (en) 2005-03-03
US20110071152A1 (en) 2011-03-24
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AU2004259662B2 (en) 2008-08-07
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US20120264801A1 (en) 2012-10-18
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