DK1299104T3 - Orale opioidagonistformuleringer sikret mod forfalskning - Google Patents

Orale opioidagonistformuleringer sikret mod forfalskning

Info

Publication number
DK1299104T3
DK1299104T3 DK01909086T DK01909086T DK1299104T3 DK 1299104 T3 DK1299104 T3 DK 1299104T3 DK 01909086 T DK01909086 T DK 01909086T DK 01909086 T DK01909086 T DK 01909086T DK 1299104 T3 DK1299104 T3 DK 1299104T3
Authority
DK
Denmark
Prior art keywords
secured against
opioid agonist
against forgery
agonist formulations
oral opioid
Prior art date
Application number
DK01909086T
Other languages
English (en)
Inventor
Benjamin Oshlack
Curtis Wright
J David Haddox
Original Assignee
Euro Celtique Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22663996&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK1299104(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Euro Celtique Sa filed Critical Euro Celtique Sa
Application granted granted Critical
Publication of DK1299104T3 publication Critical patent/DK1299104T3/da

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5084—Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/485—Morphinan derivatives, e.g. morphine, codeine
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    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0043—Nose
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    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
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    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
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    • A61K9/1629—Organic macromolecular compounds
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    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
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    • A61K9/167—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface
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    • A61K9/1694—Processes resulting in granules or microspheres of the matrix type containing more than 5% of excipient
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    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
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    • A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • A61K9/2081—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets with microcapsules or coated microparticles according to A61K9/50
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    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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    • A61K9/4808—Preparations in capsules, e.g. of gelatin, of chocolate characterised by the form of the capsule or the structure of the filling; Capsules containing small tablets; Capsules with outer layer for immediate drug release
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    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
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    • A61K9/5005—Wall or coating material
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    • A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
    • A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
    • A61K9/7053—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
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    • A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
    • A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
    • A61K9/7053—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
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  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Emergency Medicine (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Otolaryngology (AREA)
  • Pain & Pain Management (AREA)
  • Addiction (AREA)
  • Optics & Photonics (AREA)
  • Inorganic Chemistry (AREA)
  • Physics & Mathematics (AREA)
  • Nanotechnology (AREA)
  • Toxicology (AREA)
  • Psychiatry (AREA)
  • Rheumatology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DK01909086T 2000-02-08 2001-02-08 Orale opioidagonistformuleringer sikret mod forfalskning DK1299104T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US18136900P 2000-02-08 2000-02-08
PCT/US2001/004346 WO2001058451A1 (en) 2000-02-08 2001-02-08 Tamper-resistant oral opioid agonist formulations

Publications (1)

Publication Number Publication Date
DK1299104T3 true DK1299104T3 (da) 2009-08-03

Family

ID=22663996

Family Applications (5)

Application Number Title Priority Date Filing Date
DK10011790.2T DK2283842T3 (da) 2000-02-08 2001-02-08 Orale opioid-agonist-formuleringer sikret mod forfalskning
DK09006024.5T DK2092936T3 (da) 2000-02-08 2001-02-08 Orale opioid-agonist-formuleringer sikret mod forfalskning
DK10011789.4T DK2277521T3 (da) 2000-02-08 2001-02-08 Orale opioid-agonist-formuleringer sikret mod forfalskning
DK01909086T DK1299104T3 (da) 2000-02-08 2001-02-08 Orale opioidagonistformuleringer sikret mod forfalskning
DK12167170.5T DK2517710T3 (da) 2000-02-08 2001-02-08 Orale opioid-agonist-formuleringer sikret mod forfalskning

Family Applications Before (3)

Application Number Title Priority Date Filing Date
DK10011790.2T DK2283842T3 (da) 2000-02-08 2001-02-08 Orale opioid-agonist-formuleringer sikret mod forfalskning
DK09006024.5T DK2092936T3 (da) 2000-02-08 2001-02-08 Orale opioid-agonist-formuleringer sikret mod forfalskning
DK10011789.4T DK2277521T3 (da) 2000-02-08 2001-02-08 Orale opioid-agonist-formuleringer sikret mod forfalskning

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK12167170.5T DK2517710T3 (da) 2000-02-08 2001-02-08 Orale opioid-agonist-formuleringer sikret mod forfalskning

Country Status (35)

Country Link
US (15) US6696088B2 (da)
EP (6) EP1299104B1 (da)
JP (10) JP2003522144A (da)
KR (2) KR20020071032A (da)
CN (3) CN1423559A (da)
AP (1) AP1665A (da)
AT (1) ATE431145T1 (da)
AU (2) AU776904B2 (da)
BG (1) BG65828B1 (da)
BR (2) BRPI0108380B8 (da)
CA (1) CA2400567C (da)
CY (2) CY1109270T1 (da)
CZ (1) CZ299991B6 (da)
DE (1) DE60138706D1 (da)
DK (5) DK2283842T3 (da)
EA (1) EA004876B1 (da)
EE (1) EE05171B1 (da)
ES (5) ES2539945T3 (da)
GE (1) GEP20053614B (da)
HK (3) HK1051487A1 (da)
HU (2) HUP0204163A2 (da)
IL (5) IL151057A0 (da)
ME (1) MEP48308A (da)
MX (2) MXPA02007690A (da)
NO (2) NO324717B1 (da)
NZ (1) NZ520554A (da)
OA (1) OA12215A (da)
PL (1) PL210845B1 (da)
PT (6) PT1299104E (da)
RS (1) RS50407B (da)
SI (5) SI2092936T1 (da)
SK (1) SK287107B6 (da)
TW (1) TWI292317B (da)
UA (1) UA79069C2 (da)
WO (2) WO2001058447A1 (da)

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