DK1296970T3 - Fremgangsmåde til fremstilling af citalopram - Google Patents

Fremgangsmåde til fremstilling af citalopram

Info

Publication number: DK1296970T3
Authority: DK; Denmark
Prior art keywords: citalopram; preparation
Prior art date: 2000-05-12

Application number

DK01931469T

Other languages

Danish (da)

English (en)

Inventor

Hans Petersen

Robert Dancer

Original Assignee

Lundbeck & Co As H

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-05-12

Filing date

2001-05-10

Publication date

2008-07-14

2001-05-10 Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H

2008-07-14 Application granted granted Critical

2008-07-14 Publication of DK1296970T3 publication Critical patent/DK1296970T3/da

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
- C07D307/88—Benzo [c] furans; Hydrogenated benzo [c] furans with one oxygen atom directly attached in position 1 or 3

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Psychiatry (AREA)
Pain & Pain Management (AREA)
Bioinformatics & Cheminformatics (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Steroid Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Plural Heterocyclic Compounds (AREA)
Furan Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

DK01931469T 2000-05-12 2001-05-10 Fremgangsmåde til fremstilling af citalopram DK1296970T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DKPA200000783		2000-05-12
PCT/DK2001/000333 WO2001085712A1 (en)	2000-05-12	2001-05-10	Method for the preparation of citalopram

Publications (1)

Publication Number	Publication Date
DK1296970T3 true DK1296970T3 (da)	2008-07-14

Family

ID=8159493

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK01931469T DK1296970T3 (da)	2000-05-12	2001-05-10	Fremgangsmåde til fremstilling af citalopram

Country Status (30)

Country	Link
US (1)	US6660873B2 (ru)
EP (1)	EP1296970B1 (ru)
JP (1)	JP2003532721A (ru)
CN (1)	CN100422166C (ru)
AR (1)	AR032455A1 (ru)
AT (1)	ATE389645T1 (ru)
AU (2)	AU2001258239B2 (ru)
BG (1)	BG65820B1 (ru)
BR (1)	BR0110996A (ru)
CA (1)	CA2408292C (ru)
CZ (1)	CZ20024065A3 (ru)
DE (1)	DE60133280T2 (ru)
DK (1)	DK1296970T3 (ru)
EA (1)	EA005674B1 (ru)
ES (1)	ES2301541T3 (ru)
HK (1)	HK1056171A1 (ru)
HR (1)	HRP20020881A2 (ru)
HU (1)	HUP0301942A2 (ru)
IL (2)	IL152645A0 (ru)
IS (1)	IS2586B (ru)
MX (1)	MXPA02011125A (ru)
NO (1)	NO327963B1 (ru)
NZ (1)	NZ522475A (ru)
PL (1)	PL358144A1 (ru)
PT (1)	PT1296970E (ru)
SI (1)	SI1296970T1 (ru)
SK (1)	SK287035B6 (ru)
UA (1)	UA72039C2 (ru)
WO (1)	WO2001085712A1 (ru)
ZA (1)	ZA200208973B (ru)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ATE237604T1 (de)	1999-04-14	2003-05-15	Lundbeck & Co As H	Verfahren zur herstellung von citalopram
US6310222B1 (en) *	1999-11-01	2001-10-30	Sumika Fine Chemicals Co., Ltd.	Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate
US6433196B1 (en) *	2000-02-17	2002-08-13	Sumika Fine Chemicals Co., Ltd.	Production method of citalopram, intermediate therefor and production method of the intermediate
NL1017417C1 (nl)	2000-03-03	2001-03-16	Lundbeck & Co As H	Werkwijze voor de bereiding van Citalopram.
NL1017500C1 (nl)	2000-03-13	2001-04-26	Lundbeck & Co As H	Werkwijze voor de bereiding van Citalopram.
NZ521204A (en)	2000-03-13	2004-03-26	H	Stepwise alkylation of 5-substituted 1-(4-fluorophenyl)- 1,3-dihydroisobenzofurans for preparing citalopram, an anti depressant
AR032455A1 (es)	2000-05-12	2003-11-12	Lundbeck & Co As H	Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
IN192057B (ru) *	2001-07-19	2004-02-14	Ranbaxy Lab Ltd
TR200504022T1 (tr) *	2003-03-24	2006-08-21	Hetero Drugs Limited	(S)-sitalopram oksalatın yeni sıvı kristal formları.
WO2005042473A1 (en) *	2003-10-28	2005-05-12	Wockhardt Limited	Improved process for the manufacture of citalopram hydrobromide
US20050143350A1 (en) *	2003-11-19	2005-06-30	Seed John C.	Combination drug therapy to treat obesity
EP2141156A1 (en)	2004-08-23	2010-01-06	Sun Pharma Global FZE	Process for Preparation of Citalopram and Enantiomers

Family Cites Families (40)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1143702A (ru)	1965-03-18
GB1526331A (en) *	1976-01-14	1978-09-27	Kefalas As	Phthalanes
GB8419963D0 (en)	1984-08-06	1984-09-12	Lundbeck & Co As H	Intermediate compound and method
GB8814057D0 (en)	1988-06-14	1988-07-20	Lundbeck & Co As H	New enantiomers & their isolation
US5296507A (en)	1990-09-06	1994-03-22	H.Lundbeck A/S	Treatment of cerbrovascular disorders
DE19626659A1 (de)	1996-07-03	1998-01-08	Basf Ag	Verfahren zur Herstellung von Phthaliden
DE19627697A1 (de)	1996-07-10	1998-01-15	Basf Ag	Verfahren zur Herstellung von Phthaliden
ES2148120T3 (es)	1997-07-08	2002-01-16	Lundbeck & Co As H	Metodo para la preparacion de citalopram.
UA62985C2 (en) *	1997-11-10	2004-01-15	Lunnbeck As H	A method for the preparation of citalopram
ES2149734T3 (es)	1997-11-11	2003-02-16	Lundbeck & Co As H	Metodo para la preparacion de citalopram.
CN1129592C (zh)	1998-10-20	2003-12-03	H·隆德贝克有限公司	制备西酞普兰的方法
SI1140886T1 (en)	1998-12-23	2003-08-31	H. Lundbeck A/S	Method for the preparation of 5-cyanophthalide
AR022329A1 (es)	1999-01-29	2002-09-04	Lundbeck & Co As H	Metodo para la preparacion de 5-cianoftalida
ATE237604T1 (de)	1999-04-14	2003-05-15	Lundbeck & Co As H	Verfahren zur herstellung von citalopram
ITMI991579A1 (it)	1999-06-25	2001-01-15	Lundbeck & Co As H	Metodo per la preparazione di citalopram
ITMI991581A1 (it)	1999-06-25	2001-01-15	Lundbeck & Co As H	Metodo per la preparazione di citalopram
ITMI991486A1 (it)	1999-07-06	2001-01-06	Vis Farmaceutici S P A	Processo per la sintesi di citalopram
EP1228056B1 (en)	1999-10-25	2004-09-22	H. Lundbeck A/S	Method for the preparation of citalopram
US6310222B1 (en)	1999-11-01	2001-10-30	Sumika Fine Chemicals Co., Ltd.	Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate
AR026063A1 (es)	1999-11-01	2002-12-26	Lundbeck & Co As H	Metodo para la preparacion de 5-carboxiftalida.
EA004742B1 (ru)	1999-12-28	2004-08-26	Х.Лундбекк А/С	Способ получения циталопрама
JP2003519218A (ja)	1999-12-30	2003-06-17	ハー・ルンドベック・アクチエゼルスカベット	シタロプラムの製造方法
SI1254129T1 (en)	2000-01-14	2004-02-29	H. Lundbeck A/S	Method for the preparation of 5-cyanophthalide
IT1317729B1 (it)	2000-01-18	2003-07-15	Norpharma S P A	Procedimento per la preparazione della 5-carbossiftalide.
US6433196B1 (en)	2000-02-17	2002-08-13	Sumika Fine Chemicals Co., Ltd.	Production method of citalopram, intermediate therefor and production method of the intermediate
IES20010143A2 (en)	2000-02-24	2001-07-25	Lundbeck & Co As H	Method for the preparation of citalopram
NL1017415C1 (nl)	2000-02-24	2001-05-18	Lundbeck & Co As H	Werkwijze voor de bereiding van Citalopram.
NL1017417C1 (nl)	2000-03-03	2001-03-16	Lundbeck & Co As H	Werkwijze voor de bereiding van Citalopram.
GB0005477D0 (en)	2000-03-07	2000-04-26	Resolution Chemicals Limited	Process for the preparation of citalopram
CN1429219A (zh)	2000-03-13	2003-07-09	H·隆德贝克有限公司	制备西酞普兰的方法
GB2357762B (en)	2000-03-13	2002-01-30	Lundbeck & Co As H	Crystalline base of citalopram
NZ521204A (en)	2000-03-13	2004-03-26	H	Stepwise alkylation of 5-substituted 1-(4-fluorophenyl)- 1,3-dihydroisobenzofurans for preparing citalopram, an anti depressant
NL1017500C1 (nl)	2000-03-13	2001-04-26	Lundbeck & Co As H	Werkwijze voor de bereiding van Citalopram.
WO2001068630A1 (en)	2000-03-14	2001-09-20	H. Lundbeck A/S	Method for the preparation of citalopram
TR200202168T2 (tr)	2000-03-16	2002-12-23	H. Lundbeck A/S	5-Siyano-1-(4-Florofenil)-1,3-Dihidroizobenzofuranların preparasyon metodu
AR032455A1 (es)	2000-05-12	2003-11-12	Lundbeck & Co As H	Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
BR0106976A (pt)	2000-07-06	2002-07-23	Lundbeck & Co As H	Método para a preparação de citalopram
IL144816A (en)	2000-08-18	2005-09-25	Lundbeck & Co As H	Method for the preparation of citalopram
SG167655A1 (en)	2000-12-22	2011-01-28	Lundbeck & Co As H	Method for the preparation of pure citalopram
JP2003519121A (ja)	2000-12-28	2003-06-17	ハー・ルンドベック・アクチエゼルスカベット	純粋なシタロプラムの製造方法

2001
- 2001-05-07 AR ARP010102152A patent/AR032455A1/es active IP Right Grant
- 2001-05-10 EP EP01931469A patent/EP1296970B1/en not_active Expired - Lifetime
- 2001-05-10 WO PCT/DK2001/000333 patent/WO2001085712A1/en active IP Right Grant
- 2001-05-10 CN CNB018125859A patent/CN100422166C/zh not_active Expired - Fee Related
- 2001-05-10 ES ES01931469T patent/ES2301541T3/es not_active Expired - Lifetime
- 2001-05-10 MX MXPA02011125A patent/MXPA02011125A/es active IP Right Grant
- 2001-05-10 PL PL01358144A patent/PL358144A1/xx unknown
- 2001-05-10 EA EA200201211A patent/EA005674B1/ru not_active IP Right Cessation
- 2001-05-10 AU AU2001258239A patent/AU2001258239B2/en not_active Ceased
- 2001-05-10 BR BR0110996-0A patent/BR0110996A/pt not_active Application Discontinuation
- 2001-05-10 HU HU0301942A patent/HUP0301942A2/hu unknown
- 2001-05-10 AT AT01931469T patent/ATE389645T1/de not_active IP Right Cessation
- 2001-05-10 CA CA002408292A patent/CA2408292C/en not_active Expired - Fee Related
- 2001-05-10 SK SK1754-2002A patent/SK287035B6/sk not_active IP Right Cessation
- 2001-05-10 CZ CZ20024065A patent/CZ20024065A3/cs unknown
- 2001-05-10 PT PT01931469T patent/PT1296970E/pt unknown
- 2001-05-10 IL IL15264501A patent/IL152645A0/xx unknown
- 2001-05-10 NZ NZ522475A patent/NZ522475A/en unknown
- 2001-05-10 DK DK01931469T patent/DK1296970T3/da active
- 2001-05-10 DE DE60133280T patent/DE60133280T2/de not_active Expired - Fee Related
- 2001-05-10 AU AU5823901A patent/AU5823901A/xx active Pending
- 2001-05-10 JP JP2001582313A patent/JP2003532721A/ja not_active Withdrawn
- 2001-05-10 SI SI200130831T patent/SI1296970T1/sl unknown
- 2001-10-05 UA UA2002118821A patent/UA72039C2/uk unknown
2002
- 2002-10-31 IS IS6605A patent/IS2586B/is unknown
- 2002-11-04 IL IL152645A patent/IL152645A/en not_active IP Right Cessation
- 2002-11-05 ZA ZA200208973A patent/ZA200208973B/en unknown
- 2002-11-08 HR HRP20020881 patent/HRP20020881A2/hr not_active Application Discontinuation
- 2002-11-08 US US10/291,174 patent/US6660873B2/en not_active Expired - Fee Related
- 2002-11-12 NO NO20025423A patent/NO327963B1/no not_active IP Right Cessation
- 2002-12-03 BG BG107349A patent/BG65820B1/bg unknown
2003
- 2003-11-20 HK HK03108460.1A patent/HK1056171A1/xx not_active IP Right Cessation

Also Published As

Publication number	Publication date
EA200201211A1 (ru)	2003-04-24
ZA200208973B (en)	2003-11-05
HK1056171A1 (en)	2004-02-06
SK17542002A3 (sk)	2003-04-01
HUP0301942A2 (hu)	2003-09-29
EP1296970A1 (en)	2003-04-02
UA72039C2 (en)	2005-01-17
US20030134895A1 (en)	2003-07-17
ATE389645T1 (de)	2008-04-15
BG65820B1 (bg)	2010-01-29
IS2586B (is)	2010-02-15
ES2301541T3 (es)	2008-07-01
CN100422166C (zh)	2008-10-01
CA2408292A1 (en)	2001-11-15
AU2001258239B2 (en)	2005-12-08
EP1296970B1 (en)	2008-03-19
DE60133280T2 (de)	2009-04-16
NO20025423D0 (no)	2002-11-12
IL152645A (en)	2009-12-24
NO20025423L (no)	2002-11-12
NZ522475A (en)	2004-09-24
IS6605A (is)	2002-10-31
EA005674B1 (ru)	2005-04-28
DE60133280D1 (de)	2008-04-30
PT1296970E (pt)	2008-06-11
US6660873B2 (en)	2003-12-09
SK287035B6 (sk)	2009-10-07
SI1296970T1 (sl)	2008-08-31
NO327963B1 (no)	2009-10-26
BG107349A (bg)	2003-09-30
HRP20020881A2 (en)	2004-12-31
CZ20024065A3 (cs)	2003-03-12
BR0110996A (pt)	2003-03-18
PL358144A1 (en)	2004-08-09
AU5823901A (en)	2001-11-20
AR032455A1 (es)	2003-11-12
WO2001085712A1 (en)	2001-11-15
CA2408292C (en)	2009-11-10
IL152645A0 (en)	2003-06-24
CN1441795A (zh)	2003-09-10
MXPA02011125A (es)	2003-03-10
JP2003532721A (ja)	2003-11-05

Publication	Publication Date	Title
DK1173431T3 (da)	2003-08-04	Fremgangsmåde til fremstilling af citalopram
DK1105382T3 (da)	2002-05-27	Fremgangsmåde til fremstilling af citalopram
DK1159274T3 (da)	2003-07-21	Fremgangsmåde til fremstilling af citalopram
DK1296935T3 (da)	2009-06-22	Fremgangsmåde til fremstilling af substituerede octanoylamider
DK1309582T3 (da)	2005-03-14	Fremgangsmåde til fremstilling af citalopram
DK1123284T3 (da)	2003-04-28	Fremgangsmåde til fremstilling af citalopram
DK1181272T3 (da)	2002-12-30	Fremgangsmåde til fremstilling af rent citalopram
DK1181713T3 (da)	2005-01-31	Fremgangsmåde til fremstilling af rent citalopram
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CY2007029I2 (el)	2009-11-04	Μεθοδος για την παρασκευη υποκατεστημενων οκτανοϋλ-αμιδιων
DK1150966T3 (da)	2002-12-30	Fremgangsmåde til fremstilling af 5-cyanophthalid
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NO20040027L (no)	2004-01-05	Fremgangsmate for fremstillingen av escitalopram
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DK1228056T3 (da)	2005-01-24	Fremgangsmåde til fremstilling af citalopram
NO20021118D0 (no)	2002-03-06	Fremgangsmåte for fremstilling av citalopram
DK1392711T3 (da)	2014-06-10	Fremgangsmåde til fremstilling af xylose
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