UY34632A - Compuestos de oxazolidin- 2- ona y usos de los mismos - Google Patents

Compuestos de oxazolidin- 2- ona y usos de los mismos

Info

Publication number
UY34632A
UY34632A UY0001034632A UY34632A UY34632A UY 34632 A UY34632 A UY 34632A UY 0001034632 A UY0001034632 A UY 0001034632A UY 34632 A UY34632 A UY 34632A UY 34632 A UY34632 A UY 34632A
Authority
UY
Uruguay
Prior art keywords
oxazolidin
same
ona
compounds
ona compounds
Prior art date
Application number
UY0001034632A
Other languages
English (en)
Inventor
Furet Pascal
Robin Alec Fairhurst
Caravatti Giorgio
Frederic Stauffer
Frank Hans Seiler
Mccarthy Clive
Rueeger Heinrich
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48142031&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY34632(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of UY34632A publication Critical patent/UY34632A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Abstract

La presente invención se relaciona con compuestos de pirimidina oxazolidin- 2-ona sustituidos que actúan como inhibidores de la PI3K (fosfatidilinositol- 5 3- quinasa), así como también composiciones farmacéuticas de los mismos, métodos para su fabricación y usos para el tratamiento de condiciones, enfermedades y trastornos dependientes de PI3K.
UY0001034632A 2012-02-24 2013-02-21 Compuestos de oxazolidin- 2- ona y usos de los mismos UY34632A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261602954P 2012-02-24 2012-02-24
US201261736707P 2012-12-13 2012-12-13

Publications (1)

Publication Number Publication Date
UY34632A true UY34632A (es) 2013-05-31

Family

ID=48142031

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001034632A UY34632A (es) 2012-02-24 2013-02-21 Compuestos de oxazolidin- 2- ona y usos de los mismos

Country Status (31)

Country Link
US (2) US8865894B2 (es)
EP (1) EP2817307B1 (es)
JP (1) JP6154404B2 (es)
KR (1) KR101640698B1 (es)
CN (1) CN104144926B (es)
AP (1) AP2014007835A0 (es)
AR (1) AR090121A1 (es)
AU (1) AU2013223713C1 (es)
BR (1) BR112014020672B1 (es)
CA (1) CA2865372A1 (es)
CO (1) CO7051028A2 (es)
CR (1) CR20140397A (es)
DO (1) DOP2014000194A (es)
EA (1) EA026031B1 (es)
ES (1) ES2598118T3 (es)
GE (1) GEP20156389B (es)
GT (1) GT201400178A (es)
HK (1) HK1199643A1 (es)
IL (1) IL233936A (es)
MX (1) MX353341B (es)
NI (1) NI201400089A (es)
NZ (1) NZ629198A (es)
PE (1) PE20142456A1 (es)
PH (1) PH12014501900A1 (es)
PL (1) PL2817307T3 (es)
PT (1) PT2817307T (es)
SG (1) SG11201404794XA (es)
TW (1) TW201339155A (es)
UY (1) UY34632A (es)
WO (1) WO2013124826A1 (es)
ZA (1) ZA201405446B (es)

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US9296733B2 (en) 2012-11-12 2016-03-29 Novartis Ag Oxazolidin-2-one-pyrimidine derivative and use thereof for the treatment of conditions, diseases and disorders dependent upon PI3 kinases
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JOP20200094A1 (ar) 2014-01-24 2017-06-16 Dana Farber Cancer Inst Inc جزيئات جسم مضاد لـ pd-1 واستخداماتها
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TWI714525B (zh) 2014-03-24 2021-01-01 瑞士商諾華公司 用於治療細菌感染之單內醯胺（ｍｏｎｏｂａｃｔａｍ）有機化合物
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CN114920840A (zh) 2014-10-14 2022-08-19 诺华股份有限公司 针对pd-l1的抗体分子及其用途
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JP7433910B2 (ja) 2017-06-22 2024-02-20 ノバルティス アーゲー Ｃｄ７３に対する抗体分子及びその使用
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