TW337986B - Pyrazolo(1.5a) pyrimidines, their preparation and their use - Google Patents

Pyrazolo(1.5a) pyrimidines, their preparation and their use

Info

Publication number: TW337986B
Authority: TW; Taiwan
Prior art keywords: noch3; alkyl; hydrogen; pyrazolo; h3co
Prior art date: 1995-05-09

Application number

TW085105501A

Other languages

English (en)

Inventor

Benoit Remy

Grote Thomas

Bayer Herbert

Muller Bernd

Oberdorff Klaus

Original Assignee

Basf Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-05-09

Filing date

1996-05-09

Publication date

1998-08-11

1996-05-09 Application filed by Basf Ag filed Critical Basf Ag

1998-08-11 Application granted granted Critical

1998-08-11 Publication of TW337986B publication Critical patent/TW337986B/zh

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system

Landscapes

Life Sciences & Earth Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Environmental Sciences (AREA)
Engineering & Computer Science (AREA)
Dentistry (AREA)
General Health & Medical Sciences (AREA)
Wood Science & Technology (AREA)
Zoology (AREA)
Plant Pathology (AREA)
Pest Control & Pesticides (AREA)
Agronomy & Crop Science (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Plural Heterocyclic Compounds (AREA)

TW085105501A 1995-05-09 1996-05-09 Pyrazolo(1.5a) pyrimidines, their preparation and their use TW337986B (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE19516843		1995-05-09
DE19602072		1996-01-20

Publications (1)

Publication Number	Publication Date
TW337986B true TW337986B (en)	1998-08-11

Family

ID=26014970

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
TW085105501A TW337986B (en)	1995-05-09	1996-05-09	Pyrazolo(1.5a) pyrimidines, their preparation and their use

Country Status (14)

Country	Link
US (1)	US5902773A (zh)
EP (1)	EP0824533B1 (zh)
JP (1)	JPH11506428A (zh)
KR (1)	KR19990008451A (zh)
CN (1)	CN1183783A (zh)
AT (1)	ATE208778T1 (zh)
AU (1)	AU700001B2 (zh)
BR (1)	BR9608100A (zh)
CA (1)	CA2217778A1 (zh)
DE (1)	DE59608203D1 (zh)
HU (1)	HUP9801135A2 (zh)
IL (1)	IL118167A0 (zh)
TW (1)	TW337986B (zh)
WO (1)	WO1996035690A1 (zh)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE19731153A1 (de) *	1997-07-21	1999-01-28	Basf Ag	2-(Pyrazolyl- und Triazolyl-3'-oxymethylen)-phenyl-isoxazolone und -triazolone, Verfahren zu ihrer Herstellung und ihre Verwendung
AU3953799A (en) *	1998-05-28	1999-12-13	Sumitomo Chemical Company, Limited	Pyrazolopyrimidine compounds and utilization thereof
US6552026B2 (en)	1999-06-14	2003-04-22	Basf Aktiengesellschaft	6-phenyl-pyrazolopyrimidines
US20020061897A1 (en)	2000-03-30	2002-05-23	Elliott Richard L.	Neuropeptide Y antagonists
US7067520B2 (en) *	2000-11-17	2006-06-27	Ishihara Sangyo Kaisha, Ltd.	Preventive or therapeutic medicines for diabetes containing fused-heterocyclic compounds or their salts
AU2002359160A1 (en) *	2001-12-20	2003-07-09	Biovitrum Ab	PIPAZOLO (1,5-a) PYRIMIDINE DERIVATIVES AS MODULATORS OF PPAR
WO2004082383A1 (en) *	2003-03-17	2004-09-30	Basf Aktiengesellschaft	Use of triazolopyrimidines for combating nematode diseases of plants
DE10357569A1 (de) *	2003-12-10	2005-07-07	Bayer Cropscience Ag	Pyrazolopyrimidine
JP5463034B2 (ja) *	2005-05-20	2014-04-09	アラントス・フアーマシユーテイカルズ・ホールデイング・インコーポレイテツド	ピリミジン若しくはトリアジン縮合二環式メタロプロテアーゼ阻害薬
US20070155738A1 (en) *	2005-05-20	2007-07-05	Alantos Pharmaceuticals, Inc.	Heterobicyclic metalloprotease inhibitors
PL1973545T3 (pl)	2005-12-23	2013-05-31	Ariad Pharma Inc	Bicykliczne Związki Heteroarylowe
CN101967149B (zh) *	2009-07-28	2013-01-16	北京师范大学	18F取代硝基标记的吡唑并[1,5-a]嘧啶类化合物及制备和应用
US9309250B2 (en)	2011-06-22	2016-04-12	Vertex Pharmaceuticals Incorporated	Substituted pyrrolo[2,3-b]pyrazines as ATR kinase inhibitors
DK2941432T3 (en)	2012-12-07	2018-06-14	Vertex Pharma	2-amino-6-fluoro-N- (5-fluoro-4- (4- (4- (oxetan-3-yl) piperazine-1-carbonyl) piperidin-1-yl) pyridine-3-yl) pyrazolo [ 1,5ALPHA] PYRIMIDIN-3-CARBOXAMIDE AS ATR-KINASE INHIBITOR
JP2016512815A (ja)	2013-03-15	2016-05-09	バーテックスファーマシューティカルズインコーポレイテッドＶｅｒｔｅｘＰｈａｒｍａｃｅｕｔｉｃａｌｓＩｎｃｏｒｐｏｒａｔｅｄ	Ａｔｒキナーゼの阻害剤として有用な縮合ピラゾロピリミジン誘導体
WO2014143241A1 (en)	2013-03-15	2014-09-18	Vertex Pharmaceuticals Incorporated	Compounds useful as inhibitors of atr kinase
JP2016512816A (ja)	2013-03-15	2016-05-09	バーテックスファーマシューティカルズインコーポレイテッドＶｅｒｔｅｘＰｈａｒｍａｃｅｕｔｉｃａｌｓＩｎｃｏｒｐｏｒａｔｅｄ	Ａｔｒキナーゼの阻害剤として有用な化合物
US10160760B2 (en)	2013-12-06	2018-12-25	Vertex Pharmaceuticals Incorporated	Compounds useful as inhibitors of ATR kinase
SG11201610197XA (en)	2014-06-05	2017-01-27	Vertex Pharma	Radiolabelled derivatives of a 2-amino-6-fluoro-n-[5-fluoro-pyridin-3-yl]- pyrazolo[1,5-a]pyrimidin-3-carboxamide compound useful as atr kinase inhibitor, the preparation of said compound and different solid forms thereof
RS59054B1 (sr)	2014-06-17	2019-08-30	Vertex Pharma	Postupak za lečenje raka korišćenjem kombinacije chk1 i atr inhibitora
US11464774B2 (en)	2015-09-30	2022-10-11	Vertex Pharmaceuticals Incorporated	Method for treating cancer using a combination of DNA damaging agents and ATR inhibitors
MA46092A (fr)	2016-08-31	2021-04-21	Agios Pharmaceuticals Inc	Inhibiteurs de processus métaboliques cellulaires

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8617648D0 (en) *	1986-07-18	1986-08-28	Ici Plc	Fungicides
US4877738A (en) *	1986-07-25	1989-10-31	Wisconsin Alumni Research Foundation	Biological control of damping off and root rot and inoculum preparation therefor
ATE82268T1 (de) *	1987-02-09	1992-11-15	Ici Plc	Schimmelbekaempfungsmittel.
DE3825043A1 (de) *	1988-07-20	1990-02-15	Schering Ag	3-methylsulfonyl-pyrazolo(1,5-a)pyrimidin-sulfonsaeureamide, verfahren zu ihrer herstellung und ihre verwendung als mittel mit herbizider, pflanzenwuchsregulierender und fungizider wirkung
DK0629609T3 (da) *	1989-05-17	1996-12-23	Shionogi & Co	Fremgangsmåde til fremstilling af alkoxyiminoacetamidderivater og et mellemprodukt dertil

1996
- 1996-04-26 CA CA002217778A patent/CA2217778A1/en not_active Abandoned
- 1996-04-26 CN CN96193780A patent/CN1183783A/zh active Pending
- 1996-04-26 EP EP96913532A patent/EP0824533B1/de not_active Expired - Lifetime
- 1996-04-26 BR BR9608100A patent/BR9608100A/pt not_active Application Discontinuation
- 1996-04-26 JP JP8533705A patent/JPH11506428A/ja active Pending
- 1996-04-26 AT AT96913532T patent/ATE208778T1/de not_active IP Right Cessation
- 1996-04-26 KR KR1019970707981A patent/KR19990008451A/ko active IP Right Grant
- 1996-04-26 US US08/945,609 patent/US5902773A/en not_active Expired - Fee Related
- 1996-04-26 DE DE59608203T patent/DE59608203D1/de not_active Expired - Lifetime
- 1996-04-26 AU AU56484/96A patent/AU700001B2/en not_active Ceased
- 1996-04-26 HU HU9801135A patent/HUP9801135A2/hu unknown
- 1996-04-26 WO PCT/EP1996/001774 patent/WO1996035690A1/de active IP Right Grant
- 1996-05-07 IL IL11816796A patent/IL118167A0/xx unknown
- 1996-05-09 TW TW085105501A patent/TW337986B/zh active

Also Published As

Publication number	Publication date
ATE208778T1 (de)	2001-11-15
IL118167A0 (en)	1996-09-12
CN1183783A (zh)	1998-06-03
AU5648496A (en)	1996-11-29
DE59608203D1 (de)	2001-12-20
HUP9801135A2 (hu)	1998-08-28
EP0824533A1 (de)	1998-02-25
WO1996035690A1 (de)	1996-11-14
KR19990008451A (ko)	1999-01-25
US5902773A (en)	1999-05-11
JPH11506428A (ja)	1999-06-08
BR9608100A (pt)	1999-02-23
CA2217778A1 (en)	1996-11-14
AU700001B2 (en)	1998-12-17
EP0824533B1 (de)	2001-11-14

Publication	Publication Date	Title
TW337986B (en)	1998-08-11	Pyrazolo(1.5a) pyrimidines, their preparation and their use
IL119461A (en)	2000-02-29	4,7-disubstituted -7H-pyrrolo ¬2, 3-d¾pyrimidines
TW328086B (en)	1998-03-11	Biphenylamides, compositions comprising them and the preparation and use thereof
IL123293A0 (en)	1998-09-24	Piperidine derivatives their preparation and use
MY111201A (en)	1999-09-30	New imidazopyridines
WO1993000330A3 (en)	1993-03-04	Azanorbornane derivatives
AP2002002637A0 (en)	2002-09-30	Novel piperazine
UA66801C2 (uk)	2004-06-15	Триазоло[4,5-d]піримідинові сполуки, спосіб їх одержання (варіанти), фармацевтична композиція на їх основі та спосіб лікування порушень агрегації тромбоцитів
TW334435B (en)	1998-06-21	Bicyclic amines
TW234120B (zh)	1994-11-11
TW347387B (en)	1998-12-11	Piperidine derivatives
ZA9710796B (en)	1998-06-12	Oxyiminopregnanecarbolactones.
HUP0001802A2 (hu)	2001-05-28	Pirazin-származékok, eljárás előállításukra és a vegyületeket tartalmazó gyógyászati készítmények
MX9709240A (es)	1998-03-31	Fenilpiridazinonas.
GB9300763D0 (en)	1993-03-03	Chemical compound
CA2045359A1 (en)	1991-12-30	1-indolyalkyl-4-(alkoxypyrimidinyl)piperazines
PL338181A1 (en)	2000-10-09	Novel chemical compounds
TR200002380T2 (tr)	2001-03-21	Yeni triazolo (4,5-d) pirimidin bileşikleri
ZA982137B (en)	1999-09-13	Cycloalkylalkanecarboxamides and their preparation and use.
AU2392392A (en)	1993-02-23	Novel benzopyrido piperylidene compounds, compositions, methods of manufacture and methods of use
GB9123967D0 (en)	1992-01-02	New compound and its preparation
TW334430B (en)	1998-06-21	Preparation process for benzoyl derivatives and its intermediates
NZ326675A (en)	2000-01-28	Oxazoline arthropodicides
IL111966A0 (en)	1995-03-15	4-Benzoylisoxazole derivatives, their preparation and herbicidal compositions containing them
SE9802574D0 (sv)	1998-07-17	Novel compounds