TW200602058A - Fused pyrazolo pyrimidine and pyrazolo pyrimidinone derivatives - Google Patents
Fused pyrazolo pyrimidine and pyrazolo pyrimidinone derivativesInfo
- Publication number
- TW200602058A TW200602058A TW094105812A TW94105812A TW200602058A TW 200602058 A TW200602058 A TW 200602058A TW 094105812 A TW094105812 A TW 094105812A TW 94105812 A TW94105812 A TW 94105812A TW 200602058 A TW200602058 A TW 200602058A
- Authority
- TW
- Taiwan
- Prior art keywords
- pyrazolo
- fused
- pyrimidine
- pyrimidinone derivatives
- compounds
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/16—Central respiratory analeptics
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
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- A—HUMAN NECESSITIES
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- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US54858304P | 2004-02-27 | 2004-02-27 |
Publications (1)
Publication Number | Publication Date |
---|---|
TW200602058A true TW200602058A (en) | 2006-01-16 |
Family
ID=34919377
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TW094105812A TW200602058A (en) | 2004-02-27 | 2005-02-25 | Fused pyrazolo pyrimidine and pyrazolo pyrimidinone derivatives |
Country Status (16)
Country | Link |
---|---|
US (1) | US7435731B2 (zh) |
EP (1) | EP1737865A1 (zh) |
JP (1) | JP2007523938A (zh) |
KR (1) | KR100843526B1 (zh) |
CN (1) | CN1926139A (zh) |
AR (1) | AR048302A1 (zh) |
AU (1) | AU2005219525B2 (zh) |
BR (1) | BRPI0508036A (zh) |
CA (1) | CA2557575A1 (zh) |
CO (1) | CO5721008A2 (zh) |
IL (1) | IL177569A (zh) |
NO (1) | NO20064015L (zh) |
RU (1) | RU2006134020A (zh) |
TW (1) | TW200602058A (zh) |
WO (1) | WO2005085249A1 (zh) |
ZA (1) | ZA200606921B (zh) |
Families Citing this family (101)
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KR100844864B1 (ko) * | 2004-02-27 | 2008-07-09 | 에프. 호프만-라 로슈 아게 | 헤테로아릴-융합 피라졸로 유도체 |
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CA2575430A1 (en) * | 2004-08-03 | 2006-02-16 | Merck & Co., Inc. | 1,3-disubstituted heteroaryl nmda/nr2b antagonists |
US9512125B2 (en) | 2004-11-19 | 2016-12-06 | The Regents Of The University Of California | Substituted pyrazolo[3.4-D] pyrimidines as anti-inflammatory agents |
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EP2557080A1 (en) | 2006-04-04 | 2013-02-13 | The Regents of The University of California | Method for identifying pI3-kinase antagonists |
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TW200831085A (en) * | 2006-12-13 | 2008-08-01 | Merck & Co Inc | Non-nucleoside reverse transcriptase inhibitors |
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EP2123654A4 (en) | 2006-12-28 | 2011-05-11 | Taisho Pharmaceutical Co Ltd | pyrazolopyrimidine compound |
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WO2008104473A2 (en) * | 2007-02-28 | 2008-09-04 | F. Hoffmann-La Roche Ag | Pyrazolopyriidine derivatives and their use as kinase inhibitors |
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- 2005-02-24 KR KR1020067017111A patent/KR100843526B1/ko not_active IP Right Cessation
- 2005-02-24 CA CA002557575A patent/CA2557575A1/en not_active Abandoned
- 2005-02-24 JP JP2007500149A patent/JP2007523938A/ja active Pending
- 2005-02-24 CN CNA2005800063442A patent/CN1926139A/zh active Pending
- 2005-02-24 BR BRPI0508036-3A patent/BRPI0508036A/pt not_active IP Right Cessation
- 2005-02-24 RU RU2006134020/04A patent/RU2006134020A/ru not_active Application Discontinuation
- 2005-02-24 EP EP05707608A patent/EP1737865A1/en not_active Withdrawn
- 2005-02-24 WO PCT/EP2005/001936 patent/WO2005085249A1/en active Application Filing
- 2005-02-25 TW TW094105812A patent/TW200602058A/zh unknown
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US20050197340A1 (en) | 2005-09-08 |
CN1926139A (zh) | 2007-03-07 |
IL177569A0 (en) | 2006-12-10 |
RU2006134020A (ru) | 2008-04-10 |
ZA200606921B (en) | 2008-08-27 |
KR100843526B1 (ko) | 2008-07-03 |
BRPI0508036A (pt) | 2007-07-17 |
CA2557575A1 (en) | 2005-09-15 |
WO2005085249A1 (en) | 2005-09-15 |
NO20064015L (no) | 2006-11-23 |
US7435731B2 (en) | 2008-10-14 |
CO5721008A2 (es) | 2007-01-31 |
IL177569A (en) | 2012-08-30 |
JP2007523938A (ja) | 2007-08-23 |
AU2005219525A1 (en) | 2005-09-15 |
AU2005219525B2 (en) | 2011-08-18 |
KR20060114019A (ko) | 2006-11-03 |
AR048302A1 (es) | 2006-04-19 |
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