SK284408B6 - Chemické zlúčeniny s protizápalovou aktivitou obsahujúce indolovú skupinu, spôsob ich prípravy, použitie a farmaceutické kompozície, ktoré ich obsahujú - Google Patents

Chemické zlúčeniny s protizápalovou aktivitou obsahujúce indolovú skupinu, spôsob ich prípravy, použitie a farmaceutické kompozície, ktoré ich obsahujú Download PDF

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Publication number
SK284408B6
SK284408B6 SK167-2000A SK1672000A SK284408B6 SK 284408 B6 SK284408 B6 SK 284408B6 SK 1672000 A SK1672000 A SK 1672000A SK 284408 B6 SK284408 B6 SK 284408B6
Authority
SK
Slovakia
Prior art keywords
group
indole
carboxylic acid
dichlorobenzyl
alkyl
Prior art date
Application number
SK167-2000A
Other languages
English (en)
Slovak (sk)
Other versions
SK1672000A3 (en
Inventor
Andrew John Barker
Jason Grant Kettle
Alan Wellington Faull
Original Assignee
Astrazeneca Uk Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Uk Limited filed Critical Astrazeneca Uk Limited
Publication of SK1672000A3 publication Critical patent/SK1672000A3/sk
Publication of SK284408B6 publication Critical patent/SK284408B6/sk

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P39/00—General protective or antinoxious agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
SK167-2000A 1997-08-07 1998-08-04 Chemické zlúčeniny s protizápalovou aktivitou obsahujúce indolovú skupinu, spôsob ich prípravy, použitie a farmaceutické kompozície, ktoré ich obsahujú SK284408B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9716657.3A GB9716657D0 (en) 1997-08-07 1997-08-07 Chemical compounds
PCT/GB1998/002341 WO1999007351A2 (en) 1997-08-07 1998-08-04 Indole derivatives and their use as mcp-1 antagonists

Publications (2)

Publication Number Publication Date
SK1672000A3 SK1672000A3 (en) 2000-12-11
SK284408B6 true SK284408B6 (sk) 2005-03-04

Family

ID=10817097

Family Applications (1)

Application Number Title Priority Date Filing Date
SK167-2000A SK284408B6 (sk) 1997-08-07 1998-08-04 Chemické zlúčeniny s protizápalovou aktivitou obsahujúce indolovú skupinu, spôsob ich prípravy, použitie a farmaceutické kompozície, ktoré ich obsahujú

Country Status (28)

Country Link
US (2) US6441004B1 (pt)
EP (1) EP1003504B1 (pt)
JP (1) JP3863722B2 (pt)
KR (1) KR20010022318A (pt)
CN (1) CN1265591A (pt)
AT (1) ATE244007T1 (pt)
AU (1) AU745907C (pt)
BR (1) BR9811818A (pt)
CA (1) CA2297290A1 (pt)
CZ (1) CZ294600B6 (pt)
DE (1) DE69816091T2 (pt)
DK (1) DK1003504T3 (pt)
ES (1) ES2201517T3 (pt)
GB (1) GB9716657D0 (pt)
HK (1) HK1027979A1 (pt)
HR (1) HRP20000061A2 (pt)
HU (1) HUP0004301A3 (pt)
ID (1) ID23666A (pt)
IL (1) IL133989A0 (pt)
NO (1) NO20000573D0 (pt)
NZ (1) NZ502056A (pt)
PL (1) PL338948A1 (pt)
PT (1) PT1003504E (pt)
RU (1) RU2217142C2 (pt)
SK (1) SK284408B6 (pt)
TR (1) TR200000289T2 (pt)
WO (1) WO1999007351A2 (pt)
ZA (1) ZA987090B (pt)

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