RO69912A - Procedeu pentru prepararea unor tieno (1,5) benzodiazepine - Google Patents

Procedeu pentru prepararea unor tieno (1,5) benzodiazepine

Info

Publication number: RO69912A
Authority: RO; Romania
Prior art keywords: tieno; benzodiazepines; preparation
Prior art date: 1974-11-26

Application number

RO7584018A

Other languages

English (en)

French (fr)

Inventor

Jiban K Chakrabarti

David E Tupper

Original Assignee

Lilly Industries Ltd,Gb

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1974-11-26

Filing date

1975-11-25

Publication date

1980-08-15

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10459213&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=RO69912(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1975-11-25 Application filed by Lilly Industries Ltd,Gb filed Critical Lilly Industries Ltd,Gb

1980-08-15 Publication of RO69912A publication Critical patent/RO69912A/ro

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D333/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

RO7584018A 1974-11-26 1975-11-25 Procedeu pentru prepararea unor tieno (1,5) benzodiazepine RO69912A (ro)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB51240/74A GB1533235A (en)	1974-11-26	1974-11-26	Benzodiazepine derivatives

Publications (1)

Publication Number	Publication Date
RO69912A true RO69912A (ro)	1980-08-15

Family

ID=10459213

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
RO7584018A RO69912A (ro)	1974-11-26	1975-11-25	Procedeu pentru prepararea unor tieno (1,5) benzodiazepine

Country Status (30)

Country	Link
JP (1)	JPS6044314B2 (ro)
AR (1)	AR221203A1 (ro)
AT (1)	AT351547B (ro)
AU (1)	AU506340B2 (ro)
BE (1)	BE835932A (ro)
BG (1)	BG29573A3 (ro)
CA (1)	CA1075687A (ro)
CH (2)	CH613455A5 (ro)
CS (1)	CS236753B2 (ro)
DD (1)	DD123343A5 (ro)
DE (1)	DE2552403C2 (ro)
DK (1)	DK146887C (ro)
ES (1)	ES443011A1 (ro)
FR (1)	FR2292479A1 (ro)
GB (1)	GB1533235A (ro)
HK (1)	HK58681A (ro)
HU (1)	HU172493B (ro)
IE (1)	IE42564B1 (ro)
IL (1)	IL48502A (ro)
KE (1)	KE3163A (ro)
MY (1)	MY8200149A (ro)
NL (1)	NL186088C (ro)
NZ (1)	NZ179335A (ro)
PH (2)	PH11669A (ro)
PL (1)	PL100135B1 (ro)
RO (1)	RO69912A (ro)
SE (2)	SE421209B (ro)
SU (2)	SU629879A3 (ro)
YU (1)	YU298375A (ro)
ZA (1)	ZA757344B (ro)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IL62792A (en) *	1980-05-07	1985-02-28	Byk Gulden Lomberg Chem Fab	Acylated dihydrothienodiazepinone compounds,process for their preparation,and medicaments containing them
GB8819059D0 (en) *	1988-08-11	1988-09-14	Lilly Industries Ltd	Benzodiazepine compounds & their use as pharmaceuticals
GB9009229D0 (en)	1990-04-25	1990-06-20	Lilly Industries Ltd	Pharmaceutical compounds
NZ247703A (en) *	1992-05-29	1995-07-26	Lilly Industries Ltd	Thienobenzdiazepine derivatives and medicaments thereof
CA2234641A1 (en) *	1995-11-01	1997-05-09	Merck & Co., Inc.	Hexahydro-5-imino-1,4-heteroazepine derivatives as inhibitors of nitric oxide synthases
US6043358A (en)	1995-11-01	2000-03-28	Merck & Co., Inc.	Hexahydro-5-imino-1,4-heteroazepine derivatives as inhibitors of nitric oxide synthases
HUP0003718A3 (en)	1997-09-02	2002-11-28	Welfide Corp	Fused thiophene derivatives, use thereof and pharmaceutical compositions containing them
PL199016B1 (pl) *	2002-06-20	2008-08-29	Adamed Sp Z Oo	Sposób wytwarzania olanzapiny
SI21270A (sl)	2002-07-15	2004-02-29	Krka, Tovarna Zdravil, D.D., Novo Mesto	Kristalne oblike olanzapina in postopki za njihovo pripravo
DE10301923B3 (de) *	2003-01-17	2004-09-16	Krka Tovarna Zdravil, D.D.	Verfahren und Zwischenprodukte zur Herstellung von Olanzapin
AR047460A1 (es) *	2004-01-27	2006-01-18	Synthon Bv	Proceso para la fabricacion de acetato de 2-metil-4-(4-metil-1-piperazinil)-10h-tieno[2,3-b][1,5]benzodiazepina (acetato de olanzapina)
AR048272A1 (es)	2004-03-18	2006-04-12	Lek Pharmaceuticals	Sintesis de 2 metil - 4- (4- metil -1- piperazinil) - 10 h- tieno ( 2,3-b) (1,5) benzodiazepina y sus sales, metodos para su preparacion, composiciones farmaceuticas que la contienen y su uso en la fabricacion de medicamentos para el tratamiento de enfermedades mentales.
CN1980710B (zh) *	2004-06-30	2013-06-12	阿特西斯公司	作为5-羟色胺受体调节剂的取代的氮杂环庚烯衍生物
EP2292624A1 (en)	2009-07-20	2011-03-09	LEK Pharmaceuticals d.d.	Process for the purification of olanzapine

1974
- 1974-11-25 SU SU742191705A patent/SU629879A3/ru active
- 1974-11-26 GB GB51240/74A patent/GB1533235A/en not_active Expired
1975
- 1975-11-20 DK DK524175A patent/DK146887C/da active
- 1975-11-20 IL IL48502A patent/IL48502A/xx unknown
- 1975-11-20 CA CA240,082A patent/CA1075687A/en not_active Expired
- 1975-11-21 PH PH17788A patent/PH11669A/en unknown
- 1975-11-21 AU AU86858/75A patent/AU506340B2/en not_active Expired
- 1975-11-22 DE DE2552403A patent/DE2552403C2/de not_active Expired
- 1975-11-24 CH CH604478A patent/CH613455A5/xx not_active IP Right Cessation
- 1975-11-24 CH CH1517275A patent/CH613454A5/xx not_active IP Right Cessation
- 1975-11-24 ZA ZA757344A patent/ZA757344B/xx unknown
- 1975-11-24 SE SE7513185A patent/SE421209B/xx not_active IP Right Cessation
- 1975-11-24 NZ NZ179335A patent/NZ179335A/xx unknown
- 1975-11-25 AR AR261340A patent/AR221203A1/es active
- 1975-11-25 YU YU02983/75A patent/YU298375A/xx unknown
- 1975-11-25 DD DD189666A patent/DD123343A5/xx unknown
- 1975-11-25 FR FR7535900A patent/FR2292479A1/fr active Granted
- 1975-11-25 JP JP50141080A patent/JPS6044314B2/ja not_active Expired
- 1975-11-25 IE IE2565/75A patent/IE42564B1/en unknown
- 1975-11-25 RO RO7584018A patent/RO69912A/ro unknown
- 1975-11-25 BE BE6045266A patent/BE835932A/xx not_active IP Right Cessation
- 1975-11-26 HU HU75LI00000284A patent/HU172493B/hu unknown
- 1975-11-26 ES ES443011A patent/ES443011A1/es not_active Expired
- 1975-11-26 BG BG7531601A patent/BG29573A3/xx unknown
- 1975-11-26 AT AT898275A patent/AT351547B/de not_active IP Right Cessation
- 1975-11-26 PL PL1975184991A patent/PL100135B1/pl unknown
- 1975-11-26 CS CS757991A patent/CS236753B2/cs unknown
- 1975-11-26 NL NLAANVRAGE7513833,A patent/NL186088C/xx not_active IP Right Cessation
1976
- 1976-10-07 SU SU762406250A patent/SU626702A3/ru active
1977
- 1977-02-22 PH PH19480A patent/PH24534A/en unknown
1978
- 1978-11-27 SE SE7812194A patent/SE429045B/sv not_active IP Right Cessation
1981
- 1981-09-24 KE KE3163A patent/KE3163A/xx unknown
- 1981-11-26 HK HK586/81A patent/HK58681A/xx unknown
1982
- 1982-12-30 MY MY149/82A patent/MY8200149A/xx unknown

Also Published As

Publication number	Publication date
CH613454A5 (en)	1979-09-28
AR221203A1 (es)	1981-01-15
IE42564L (en)	1976-05-26
AU506340B2 (en)	1979-12-20
NL7513833A (nl)	1976-05-31
PH11669A (en)	1978-05-19
IE42564B1 (en)	1980-09-10
SE7513185L (sv)	1976-05-27
PH24534A (en)	1990-08-03
JPS6044314B2 (ja)	1985-10-02
DD123343A5 (ro)	1976-12-12
FR2292479A1 (fr)	1976-06-25
SE421209B (sv)	1981-12-07
ZA757344B (en)	1976-11-24
IL48502A0 (en)	1976-01-30
YU298375A (en)	1982-10-31
NZ179335A (en)	1978-11-13
KE3163A (en)	1981-10-16
SE7812194L (sv)	1978-11-27
DK146887B (da)	1984-01-30
DE2552403C2 (de)	1986-06-19
DK524175A (da)	1976-05-27
AT351547B (de)	1979-07-25
MY8200149A (en)	1982-12-31
CH613455A5 (en)	1979-09-28
HK58681A (en)	1981-12-04
SU626702A3 (ru)	1978-09-30
SE429045B (sv)	1983-08-08
CS236753B2 (en)	1985-05-15
DK146887C (da)	1984-07-09
NL186088B (nl)	1990-04-17
JPS5176296A (en)	1976-07-01
HU172493B (hu)	1978-09-28
NL186088C (nl)	1990-09-17
FR2292479B1 (ro)	1978-07-28
PL100135B1 (pl)	1978-09-30
BE835932A (fr)	1976-05-25
IL48502A (en)	1980-01-31
CA1075687A (en)	1980-04-15
ATA898275A (de)	1979-01-15
GB1533235A (en)	1978-11-22
ES443011A1 (es)	1977-07-01
AU8685875A (en)	1977-05-26
SU629879A3 (ru)	1978-10-25
DE2552403A1 (de)	1976-08-12
BG29573A3 (en)	1980-12-12

Publication	Publication Date	Title
RO70051A (ro)	1980-12-30	Procedeu pentru prepararea unor 2-tetrahidrofurfuril-6,7-benzomorfani
RO72736A (ro)	1982-09-09	Procedeu pentru prepararea unor 2-tetrahidrofurfuril-6,7-benzomorfani-5,9-beta-disubstituiti
RO68142A (ro)	1981-08-30	Procedeu pentru prepararea unor 4-fenilpiperidine
RO65454A (ro)	1980-01-15	Procedeu pentru prepararea unor calcone substituite
RO69608A (ro)	1982-07-06	Procedeu pentru prepararea unor 1,2-benzizotiazol-3-one
RO69912A (ro)	1980-08-15	Procedeu pentru prepararea unor tieno (1,5) benzodiazepine
RO68145A (ro)	1980-01-15	Procedeu pentru prepararea unor 3,4-dihidro-2h-1,2-benzo-tiazincarboxamide
BE838823A (fr)	1976-08-23	Procede pour la preparation de 1,2,5-dihydroxycholecalciferol
RO66914A (ro)	1981-07-30	Procedeu pentru prepararea de pirido-benzodiazepinone
RO64606A (fr)	1979-01-15	Procede pour la preparation des 6-methylergolines-8,8-disubstituees
RO67193A (fr)	1979-06-15	Procede pour la preparation du 2,2,6,6-tetramethyle-4-piperydone
RO63021A (fr)	1978-05-15	Procede pour la preparation des 3-fluorcephalosporines
RO64281A (fr)	1979-07-15	Procede pour la preparation des 6-methyle-8-methylergolines substituees
RO76667A (ro)	1981-04-30	Procedeu pentru prepararea unor 2,4-dialchilamino-6-clor-5-triazine
FR2303798A1 (fr)	1976-10-08	Procede pour la preparation de (3r, 3'r)-zeaxanthene
RO68749A (ro)	1980-01-15	Procedeu pentru prepararea 2-aminoimidazolilor
BE826343A (fr)	1975-09-08	Procede de preparation de s-triazolo(3,4- bbenzothiazoles
RO66020A (ro)	1980-06-15	Procedeu pentru prepararea unor 3-piperazinoizochinoline
RO70232A (ro)	1982-04-12	Procedeu pentru prepararea unor 4-pirazoli-4h-1,2,4-triazolil
RO72516A (ro)	1982-02-26	Procedeu pentru prepararea unor chinoxalin-1,4-dioxizi
BE809494A (fr)	1974-07-08	Procede pour la preparation de 1,4-dioxanne
RO68650A (ro)	1980-04-15	Procedeu pentru prepararea unor imidazol-(1,2-a)s-triazine
BE835855A (fr)	1976-05-24	Procede de preparation de nouvelles 7,7 -diphenyl - hexahydro - 1,4 - oxazepines
FR2286198A1 (fr)	1976-04-23	Procede pour la preparation d'agglomeres
FR2283150A1 (fr)	1976-03-26	Procede pour la preparation d'hydroxy-11b alkyl-18 oestranes