PH11669A - Thienobenzo(1,5)diazepine derivatives and the pharmaceutical formulation thereof - Google Patents

Thienobenzo(1,5)diazepine derivatives and the pharmaceutical formulation thereof

Info

Publication number: PH11669A
Authority: PH; Philippines
Prior art keywords: thienobenzo; pharmaceutical formulation; diazepine derivatives; diazepine; derivatives
Prior art date: 1974-11-26

Application number

PH17788A

Inventor

D Tupper

J Chakrabarti

Original Assignee

Lilly Industries Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1974-11-26

Filing date

1975-11-21

Publication date

1978-05-19

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10459213&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PH11669(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1975-11-21 Application filed by Lilly Industries Ltd filed Critical Lilly Industries Ltd

1978-05-19 Publication of PH11669A publication Critical patent/PH11669A/en

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D333/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Neurology (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

PH17788A 1974-11-26 1975-11-21 Thienobenzo(1,5)diazepine derivatives and the pharmaceutical formulation thereof PH11669A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB51240/74A GB1533235A (en)	1974-11-26	1974-11-26	Benzodiazepine derivatives

Publications (1)

Publication Number	Publication Date
PH11669A true PH11669A (en)	1978-05-19

Family

ID=10459213

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
PH17788A PH11669A (en)	1974-11-26	1975-11-21	Thienobenzo(1,5)diazepine derivatives and the pharmaceutical formulation thereof
PH19480A PH24534A (en)	1974-11-26	1977-02-22	Benzothieno(1,5)diazepine intermediates

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
PH19480A PH24534A (en)	1974-11-26	1977-02-22	Benzothieno(1,5)diazepine intermediates

Country Status (30)

Country	Link
JP (1)	JPS6044314B2 (en)
AR (1)	AR221203A1 (en)
AT (1)	AT351547B (en)
AU (1)	AU506340B2 (en)
BE (1)	BE835932A (en)
BG (1)	BG29573A3 (en)
CA (1)	CA1075687A (en)
CH (2)	CH613454A5 (en)
CS (1)	CS236753B2 (en)
DD (1)	DD123343A5 (en)
DE (1)	DE2552403C2 (en)
DK (1)	DK146887C (en)
ES (1)	ES443011A1 (en)
FR (1)	FR2292479A1 (en)
GB (1)	GB1533235A (en)
HK (1)	HK58681A (en)
HU (1)	HU172493B (en)
IE (1)	IE42564B1 (en)
IL (1)	IL48502A (en)
KE (1)	KE3163A (en)
MY (1)	MY8200149A (en)
NL (1)	NL186088C (en)
NZ (1)	NZ179335A (en)
PH (2)	PH11669A (en)
PL (1)	PL100135B1 (en)
RO (1)	RO69912A (en)
SE (2)	SE421209B (en)
SU (2)	SU629879A3 (en)
YU (1)	YU298375A (en)
ZA (1)	ZA757344B (en)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IL62792A (en) *	1980-05-07	1985-02-28	Byk Gulden Lomberg Chem Fab	Acylated dihydrothienodiazepinone compounds,process for their preparation,and medicaments containing them
GB8819059D0 (en) *	1988-08-11	1988-09-14	Lilly Industries Ltd	Benzodiazepine compounds & their use as pharmaceuticals
GB9009229D0 (en)	1990-04-25	1990-06-20	Lilly Industries Ltd	Pharmaceutical compounds
TW268005B (en) *	1992-05-29	1996-01-11	Lilly Industries Ltd
JP3188715B2 (en) *	1995-11-01	2001-07-16	メルクエンドカンパニーインコーポレーテッド	Hexahydro-5-imino-1,4-heteroazepine derivatives as inhibitors of nitric oxide synthase
US6043358A (en)	1995-11-01	2000-03-28	Merck & Co., Inc.	Hexahydro-5-imino-1,4-heteroazepine derivatives as inhibitors of nitric oxide synthases
WO1999011647A1 (en)	1997-09-02	1999-03-11	Yoshitomi Pharmaceutical Industries, Ltd.	Fused thiophene compounds and medicinal use thereof
PL199016B1 (en) *	2002-06-20	2008-08-29	Adamed Sp Z Oo	Method of manufacture of alanzapine, new derivative of n-demethyl olanzapine and method of manufacture of new derivative of n-demethyl olanzapine
SI21270A (en)	2002-07-15	2004-02-29	Krka, Tovarna Zdravil, D.D., Novo Mesto	Crystal forms of olanzapine and procedures for their preparation
DE10301923B3 (en) *	2003-01-17	2004-09-16	Krka Tovarna Zdravil, D.D.	Process and intermediates for the production of olanzapine
EP1711503A1 (en) *	2004-01-27	2006-10-18	Synthon B.V.	Synthesis of olanzapine and intermediates thereof
AR048272A1 (en)	2004-03-18	2006-04-12	Lek Pharmaceuticals	SYNTHESIS OF 2 METHYL - 4- (4- METHYL -1- PIPERAZINIL) - 10 H- TIENO (2,3-B) (1,5) BENZODIAZEPIN AND ITS SALTS, METHODS FOR THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING IT AND ITS USE IN THE MANUFACTURE OF MEDICINES FOR THE TREATMENT OF MENTAL DISEASES.
ES2398694T3 (en) *	2004-06-30	2013-03-21	Athersys, Inc.	Substituted azepine derivatives as serotonin receptor modulators
EP2292624A1 (en)	2009-07-20	2011-03-09	LEK Pharmaceuticals d.d.	Process for the purification of olanzapine

1974
- 1974-11-25 SU SU742191705A patent/SU629879A3/en active
- 1974-11-26 GB GB51240/74A patent/GB1533235A/en not_active Expired
1975
- 1975-11-20 IL IL48502A patent/IL48502A/en unknown
- 1975-11-20 DK DK524175A patent/DK146887C/en active
- 1975-11-20 CA CA240,082A patent/CA1075687A/en not_active Expired
- 1975-11-21 AU AU86858/75A patent/AU506340B2/en not_active Expired
- 1975-11-21 PH PH17788A patent/PH11669A/en unknown
- 1975-11-22 DE DE2552403A patent/DE2552403C2/en not_active Expired
- 1975-11-24 CH CH1517275A patent/CH613454A5/en not_active IP Right Cessation
- 1975-11-24 SE SE7513185A patent/SE421209B/en not_active IP Right Cessation
- 1975-11-24 CH CH604478A patent/CH613455A5/en not_active IP Right Cessation
- 1975-11-24 ZA ZA757344A patent/ZA757344B/en unknown
- 1975-11-24 NZ NZ179335A patent/NZ179335A/en unknown
- 1975-11-25 IE IE2565/75A patent/IE42564B1/en unknown
- 1975-11-25 YU YU02983/75A patent/YU298375A/en unknown
- 1975-11-25 BE BE6045266A patent/BE835932A/en not_active IP Right Cessation
- 1975-11-25 JP JP50141080A patent/JPS6044314B2/en not_active Expired
- 1975-11-25 DD DD189666A patent/DD123343A5/xx unknown
- 1975-11-25 FR FR7535900A patent/FR2292479A1/en active Granted
- 1975-11-25 AR AR261340A patent/AR221203A1/en active
- 1975-11-25 RO RO7584018A patent/RO69912A/en unknown
- 1975-11-26 ES ES443011A patent/ES443011A1/en not_active Expired
- 1975-11-26 CS CS757991A patent/CS236753B2/en unknown
- 1975-11-26 HU HU75LI00000284A patent/HU172493B/en unknown
- 1975-11-26 PL PL1975184991A patent/PL100135B1/en unknown
- 1975-11-26 NL NLAANVRAGE7513833,A patent/NL186088C/en not_active IP Right Cessation
- 1975-11-26 AT AT898275A patent/AT351547B/en not_active IP Right Cessation
- 1975-11-26 BG BG7531601A patent/BG29573A3/en unknown
1976
- 1976-10-07 SU SU762406250A patent/SU626702A3/en active
1977
- 1977-02-22 PH PH19480A patent/PH24534A/en unknown
1978
- 1978-11-27 SE SE7812194A patent/SE429045B/en not_active IP Right Cessation
1981
- 1981-09-24 KE KE3163A patent/KE3163A/en unknown
- 1981-11-26 HK HK586/81A patent/HK58681A/en unknown
1982
- 1982-12-30 MY MY149/82A patent/MY8200149A/en unknown

Also Published As

Publication number	Publication date
CS236753B2 (en)	1985-05-15
SE7812194L (en)	1978-11-27
SU629879A3 (en)	1978-10-25
ES443011A1 (en)	1977-07-01
BE835932A (en)	1976-05-25
AT351547B (en)	1979-07-25
AU8685875A (en)	1977-05-26
IE42564L (en)	1976-05-26
HK58681A (en)	1981-12-04
DD123343A5 (en)	1976-12-12
FR2292479B1 (en)	1978-07-28
CH613455A5 (en)	1979-09-28
ATA898275A (en)	1979-01-15
JPS5176296A (en)	1976-07-01
IL48502A0 (en)	1976-01-30
AR221203A1 (en)	1981-01-15
DK524175A (en)	1976-05-27
DE2552403C2 (en)	1986-06-19
IL48502A (en)	1980-01-31
SE7513185L (en)	1976-05-27
JPS6044314B2 (en)	1985-10-02
BG29573A3 (en)	1980-12-12
KE3163A (en)	1981-10-16
NL186088B (en)	1990-04-17
SE421209B (en)	1981-12-07
RO69912A (en)	1980-08-15
GB1533235A (en)	1978-11-22
MY8200149A (en)	1982-12-31
FR2292479A1 (en)	1976-06-25
DK146887C (en)	1984-07-09
PH24534A (en)	1990-08-03
YU298375A (en)	1982-10-31
ZA757344B (en)	1976-11-24
AU506340B2 (en)	1979-12-20
HU172493B (en)	1978-09-28
PL100135B1 (en)	1978-09-30
NL186088C (en)	1990-09-17
SU626702A3 (en)	1978-09-30
NZ179335A (en)	1978-11-13
CA1075687A (en)	1980-04-15
CH613454A5 (en)	1979-09-28
DE2552403A1 (en)	1976-08-12
NL7513833A (en)	1976-05-31
IE42564B1 (en)	1980-09-10
SE429045B (en)	1983-08-08
DK146887B (en)	1984-01-30

Publication	Publication Date	Title
GR61176B (en)	1978-10-03	Pharmaceutical compositions and process for the preparation thereof
IL47625A (en)	1981-01-30	4-heterocyclyl-6,7-dialkoxyquin-azoline derivatives and pharmaceutical compositions containing them
IL53043A (en)	1982-01-31	N-heterocyclylalkyl-(1-aryloxy-2-hydroxy-3-amino-propane)derivatives,their preparation and pharmaceutical compositions containing them
NZ183150A (en)	1979-12-11	7-aminothiazolyl-iminoa-cetamido-cephalosporin derivatives and pharmaceutical compositions
PH11669A (en)	1978-05-19	Thienobenzo(1,5)diazepine derivatives and the pharmaceutical formulation thereof
IL49325A (en)	1979-11-30	8-aza-11-deoxy-pge1 derivatives,their preparation and pharmaceutical compositions containing them
NZ184755A (en)	1979-12-11	2-benzylpyrrolidine derivatives and pharmaceutical compositions
IL52717A (en)	1980-12-31	Derivatives of2-phenylamino-imidazoline-(2),their preparation and pharmaceutical compositions containing them
NZ185642A (en)	1980-09-12	Morphanthridine derivatives and pharmaceutical compositions
IL52857A (en)	1983-03-31	Oxo-benzopyrane derivatives,their preparation and pharmaceutical compositions containing them
NZ184103A (en)	1979-01-11	Fenzodioxole derivatives and pharmaceutical compositions
AU1306576A (en)	1977-10-20	Pharmaceutical formulation
NZ185539A (en)	1979-12-11	Cis-4a-aryl-2-substituted-2,3,4,4a,5,6,7,7a-octa hydro-1h-2-pyrindines and pharmaceutical compositions
NZ184185A (en)	1979-04-26	3,5,5-trimethylhexanoyl-ferrocene and pharmaceutical compositions
IL47335A0 (en)	1975-07-28	Hexahydro-diazepino-indole derivatives and the preparation thereof
IL51468A (en)	1981-01-30	17 -hydroxy- -d-homosteroid derivatives,their preparation and pharmaceutical compositions containing them
JPS52128364A (en)	1977-10-27	Novel corticoid * preparation thereof and antiiinflamatory pharmaceutical agent containing the same
IL49344A (en)	1979-05-31	2-substituted-7-halo-1,8-maphthyridine compounds,processesfor preparing the same and pharmaceutical compositions containing the same
NZ184367A (en)	1978-11-13	2-vinyl-chromone derivatives and pharmaceutical compositions
NZ185295A (en)	1980-04-28	9-chloroprednisolone derivatives and pharmaceutical compositions
PH10402A (en)	1977-03-07	1,4-dithino(2,3-c)pyrrole derivatives and pharmaceutical compositions containing the same
NZ182995A (en)	1979-10-25	5-substituted-indane-2-carboxylic acids,derivatives and pharmaceutical compositions
NZ185996A (en)	1980-04-28	6, 7-methylene-3-oxo-d-homo-17a-pregna-4, 16-dienes and pharmaceutical compositions
NZ183154A (en)	1978-09-25	1,3-dihydro-1-dimethylphosphinylalkyl-3-phenylspiro-(isobenzofuran) derivatives and pharmaceutical compositions
PH13123A (en)	1979-12-12	Hydrazinopyridazine derivatives and pharmaceutical compositions thereof