PT831829E - Derivados de pirimidina heterociclicos de aneis fundidos - Google Patents

Derivados de pirimidina heterociclicos de aneis fundidos

Info

Publication number
PT831829E
PT831829E PT95924027T PT95924027T PT831829E PT 831829 E PT831829 E PT 831829E PT 95924027 T PT95924027 T PT 95924027T PT 95924027 T PT95924027 T PT 95924027T PT 831829 E PT831829 E PT 831829E
Authority
PT
Portugal
Prior art keywords
heterocyclics
fused rings
pyrimidine derivatives
pyrimidine
derivatives
Prior art date
Application number
PT95924027T
Other languages
English (en)
Inventor
Mikel P Moyer
Lee D Arnold
Susan B Sobolov-Jaynes
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of PT831829E publication Critical patent/PT831829E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/26Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32Nitrogen atom
PT95924027T 1995-06-07 1995-06-07 Derivados de pirimidina heterociclicos de aneis fundidos PT831829E (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
PCT/US1995/007881 WO1996040142A1 (en) 1995-06-07 1995-06-07 Heterocyclic ring-fused pyrimidine derivatives
HU9601559A HUP9601559A3 (en) 1995-06-07 1996-06-06 Heterocyclic ring-fused pyrimidine derivatives, pharmaceutical compositions containing the same and intermediates

Publications (1)

Publication Number Publication Date
PT831829E true PT831829E (pt) 2003-12-31

Family

ID=89994036

Family Applications (1)

Application Number Title Priority Date Filing Date
PT95924027T PT831829E (pt) 1995-06-07 1995-06-07 Derivados de pirimidina heterociclicos de aneis fundidos

Country Status (32)

Country Link
EP (1) EP0831829B1 (pt)
JP (1) JP3290666B2 (pt)
CN (1) CN1141298A (pt)
AP (1) AP637A (pt)
AR (1) AR002746A1 (pt)
AT (1) ATE247469T1 (pt)
AU (1) AU5479196A (pt)
BR (1) BR9602695A (pt)
CA (1) CA2223081C (pt)
CO (1) CO4440628A1 (pt)
CZ (1) CZ164196A3 (pt)
DE (1) DE69531558T2 (pt)
DK (1) DK0831829T3 (pt)
ES (1) ES2203642T3 (pt)
FI (1) FI974443A (pt)
HR (1) HRP960269A2 (pt)
HU (1) HUP9601559A3 (pt)
IL (1) IL118487A0 (pt)
MA (1) MA26409A1 (pt)
MX (1) MX9709867A (pt)
NO (1) NO962386L (pt)
NZ (1) NZ286755A (pt)
OA (1) OA10460A (pt)
PL (1) PL314641A1 (pt)
PT (1) PT831829E (pt)
RU (1) RU2136683C1 (pt)
SG (1) SG45483A1 (pt)
SI (1) SI9600184A (pt)
SK (1) SK72996A3 (pt)
TR (1) TR199600474A2 (pt)
WO (1) WO1996040142A1 (pt)
ZA (1) ZA964725B (pt)

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HUP9601559A3 (en) 1997-07-28
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TR199600474A2 (tr) 1996-12-21
MA26409A1 (fr) 2004-12-20
EP0831829B1 (en) 2003-08-20
SG45483A1 (en) 1998-01-16
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AP637A (en) 1998-04-08
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AR002746A1 (es) 1998-04-29

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