NO20032187L - Heterocyklylalkylpiperidinderivater, deres fremstilling samt preparater inneholdende forbindelsene - Google Patents

Heterocyklylalkylpiperidinderivater, deres fremstilling samt preparater inneholdende forbindelsene

Info

Publication number: NO20032187L
Authority: NO; Norway
Prior art keywords: compounds; preparation; preparations containing; heterocyclylalkylpiperidine derivatives; heterocyclylalkylpiperidine
Prior art date: 2000-11-15

Application number

NO20032187A

Other languages

English (en)

Other versions

NO20032187D0 (no

Inventor

Eric Bacque

Jean-Christophe Carry

Youssef El-Ahmad

Michel Evers

Philippe Hubert

Jean-Luc Malleron

Serge Mignani

Guy Pantel

Michel Tabart

Fabrice Viviani

Original Assignee

Aventis Pharma Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-11-15

Filing date

2003-05-14

Publication date

2003-06-26

2003-05-14 Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa

2003-05-14 Publication of NO20032187D0 publication Critical patent/NO20032187D0/no

2003-06-26 Publication of NO20032187L publication Critical patent/NO20032187L/no

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

NO20032187A 2000-11-15 2003-05-14 Heterocyklylalkylpiperidinderivater, deres fremstilling samt preparater inneholdende forbindelsene NO20032187L (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR0014738A FR2816618B1 (fr)	2000-11-15	2000-11-15	Derives heterocyclylalcoyl piperidine, leur preparation et les compositions qui les contiennent
PCT/FR2001/003559 WO2002040474A2 (fr)	2000-11-15	2001-11-14	Derives heterocyclylalcoyl piperidine et leur application comme antimicrobiens

Publications (2)

Publication Number	Publication Date
NO20032187D0 NO20032187D0 (no)	2003-05-14
NO20032187L true NO20032187L (no)	2003-06-26

Family

ID=8856503

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
NO20032187A NO20032187L (no)	2000-11-15	2003-05-14	Heterocyklylalkylpiperidinderivater, deres fremstilling samt preparater inneholdende forbindelsene
NO20072142A NO20072142L (no)	2000-11-15	2007-04-25	Mellomprodukter for fremstilling av heterocyklylalkylpiperidinderivater og forbindelser for fremstilling av disse

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
NO20072142A NO20072142L (no)	2000-11-15	2007-04-25	Mellomprodukter for fremstilling av heterocyklylalkylpiperidinderivater og forbindelser for fremstilling av disse

Country Status (28)

Country	Link
EP (2)	EP1695964A1 (no)
JP (1)	JP2004514661A (no)
KR (1)	KR100849608B1 (no)
CN (1)	CN1483031A (no)
AR (1)	AR034006A1 (no)
AT (1)	ATE337311T1 (no)
AU (2)	AU2002218365B2 (no)
BG (1)	BG107793A (no)
BR (1)	BR0115312A (no)
CA (1)	CA2429311A1 (no)
CZ (1)	CZ20031316A3 (no)
DE (1)	DE60122567T2 (no)
DK (1)	DK1337529T3 (no)
EA (1)	EA200300568A1 (no)
EE (1)	EE200300207A (no)
ES (1)	ES2271119T3 (no)
FR (1)	FR2816618B1 (no)
HR (1)	HRP20030379A2 (no)
HU (1)	HUP0303758A3 (no)
IL (1)	IL155841A0 (no)
NO (2)	NO20032187L (no)
PL (1)	PL363004A1 (no)
PT (1)	PT1337529E (no)
SK (1)	SK5822003A3 (no)
TN (1)	TNSN01160A1 (no)
WO (1)	WO2002040474A2 (no)
YU (1)	YU46803A (no)
ZA (1)	ZA200303794B (no)

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DE60125373T2 (de)	2000-07-26	2007-10-18	Smithkline Beecham P.L.C., Brentford	Aminopiperidin chinoline und ihre azaisosteren analoga mit antibakterieller wirkung
GB0101577D0 (en)	2001-01-22	2001-03-07	Smithkline Beecham Plc	Compounds
GB0112834D0 (en)	2001-05-25	2001-07-18	Smithkline Beecham Plc	Medicaments
GB0112836D0 (en)	2001-05-25	2001-07-18	Smithkline Beecham Plc	Medicaments
GB0118238D0 (en) *	2001-07-26	2001-09-19	Smithkline Beecham Plc	Medicaments
WO2003064431A2 (en)	2002-01-29	2003-08-07	Glaxo Group Limited	Aminopiperidine compounds, process for their preparation, and pharmaceutical compositions containing them
EP2181996A1 (en)	2002-01-29	2010-05-05	Glaxo Group Limited	Aminopiperidine derivatives
AR040336A1 (es)	2002-06-26	2005-03-30	Glaxo Group Ltd	Compuesto de piperidina, uso del mismo para la fabricacion de un medicamento, composicion farmaceutica que lo comprende y procedimiento para preparar dicho compuesto
AR040335A1 (es)	2002-06-26	2005-03-30	Glaxo Group Ltd	Compuesto de ciclohexano o ciclohexeno, uso del mismo para preparar un medicamento, composicion farmaceutica que lo comprende, procedimiento y compuestos intermediarios de utilidad para preparar dicho compuesto
FR2842807A1 (fr) *	2002-07-23	2004-01-30	Aventis Pharma Sa	Derives de la quinolyl propyl piperidine, procede et intermediaires de preparation et compositions les renfermant
GB0217294D0 (en) *	2002-07-25	2002-09-04	Glaxo Group Ltd	Medicaments
FR2844270B1 (fr)	2002-09-11	2006-05-19	Aventis Pharma Sa	Derives de la quinolyl propyl piperidine, leur procede et intermediaires de preparation et les compositions qui les contiennent
FR2844268B1 (fr)	2002-09-11	2004-10-22	Aventis Pharma Sa	Derives de la quinolyl propyl piperidine, leurs procedes et intermediaires de preparation et les compositions qui les contiennent
DE10256405A1 (de) *	2002-12-02	2004-06-17	Morphochem Aktiengesellschaft für kombinatorische Chemie	Neue Verbindungen, die Topoisomerase IV inhibieren
JP4704755B2 (ja)	2002-11-05	2011-06-22	グラクソスミスクライン・リミテッド・ライアビリティ・カンパニー	抗菌剤
EP1567520B1 (en)	2002-12-04	2008-10-15	Glaxo Group Limited	Quinolines and nitrogenated derivatives thereof and their use as antibacterial agents
FR2852954B1 (fr) *	2003-03-28	2006-07-14	Aventis Pharma Sa	Derives de quinoleines-4-substituees, leurs procede et intermediaires de preparation et les compositions pharmaceutiques qui les contiennent
US7232833B2 (en)	2003-03-28	2007-06-19	Novexel	4-substituted quinoline derivatives, method and intermediates for their preparation and pharmaceutical compositions containing them
FR2862301B1 (fr) *	2003-11-17	2007-12-21	Aventis Pharma Sa	Nouveau procede de preparation de quinoleines 3-fluorees
FR2867472B1 (fr) *	2004-03-12	2008-07-18	Aventis Pharma Sa	Derives de quinoleines-4-substituees, leurs procede et intermediaires de preparation et les compositions pharmaceutiques qui les contiennent
WO2006081178A2 (en)	2005-01-25	2006-08-03	Glaxo Group Limited	Antibacterial agents
US7605169B2 (en)	2005-01-25	2009-10-20	Glaxo Group Limited	Antibacterial agents
JP2008528587A (ja)	2005-01-25	2008-07-31	グラクソグループリミテッド	抗菌剤
EP1846418A4 (en)	2005-01-25	2009-12-23	Glaxo Group Ltd	ANTIBACTERIAL ACTIVE SUBSTANCES
JP2008531709A (ja)	2005-03-01	2008-08-14	ワイス	シンノリン化合物および肝臓ｘ受容体調節物質としてのそれらの使用
MY150958A (en) *	2005-06-16	2014-03-31	Astrazeneca Ab	Compounds for the treatment of multi-drug resistant bacterial infections
CA2635126A1 (en)	2006-01-26	2007-08-02	Actelion Pharmaceuticals Ltd	Tetrahydropyrane antibiotics
WO2007115947A1 (en)	2006-04-06	2007-10-18	Glaxo Group Limited	Pyrrolo-quinoxalinone derivatives as antibacterials
EP1992628A1 (en)	2007-05-18	2008-11-19	Glaxo Group Limited	Derivatives and analogs of N-ethylquinolones and N-ethylazaquinolones
ATE520687T1 (de)	2007-06-15	2011-09-15	Actelion Pharmaceuticals Ltd	3-amino-6-(1-amino-ethyl)-tetrahydropyranderiva e
EP2080761A1 (en)	2008-01-18	2009-07-22	Glaxo Group Limited	Compounds
WO2010043714A1 (en)	2008-10-17	2010-04-22	Glaxo Group Limited	Tricyclic nitrogen compounds used as antibacterials
EP2379554B1 (en)	2009-01-15	2015-11-11	Glaxo Group Limited	Naphthyridin-2(1h)-one compounds useful as antibacterials
JP6389174B2 (ja) *	2012-08-15	2018-09-12	グラクソグループリミテッドＧｌａｘｏＧｒｏｕｐＬｉｍｉｔｅｄ	化学的方法
EA031589B1 (ru)	2014-08-22	2019-01-31	Глэксосмитклайн Интеллекчуал Проперти Дивелопмент Лимитед	Трициклические азотсодержащие соединения для лечения инфекции, вызываемой neisseria gonorrhoeae
WO2016138988A1 (en) *	2015-03-02	2016-09-09	University Of Copenhagen	Piperazine inhibitors of bacterial gyrase and topoisomerase iv
UY36851A (es)	2015-08-16	2017-03-31	Glaxosmithkline Ip Dev Ltd	Compuestos para uso en aplicaciones antibacterianas

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
NL7908031A (nl)	1979-11-01	1981-06-01	Acf Chemiefarma Nv	Nieuwe chinolinederivaten en farmaceutische preparaten die een dergelijke verbinding bevatten, alsmede werk- wijze voor het bereiden van deze verbindingen.
JPH0239546A (ja)	1988-07-29	1990-02-08	Origin Electric Co Ltd	混成集積回路の製造方法
AU623474B2 (en)	1989-01-16	1992-05-14	Laboratoire Roger Bellon	New benzo(1,8)naphthyridine derivatives, their preparation and compositions containing them
ES2201674T3 (es) *	1998-01-26	2004-03-16	Smithkline Beecham Plc	Derivados de quinolina con propiedades antibacterianas.
AU2437900A (en) *	1999-01-20	2000-08-07	Smithkline Beecham Plc	Piperidinylquinolines as protein tyrosine kinase inhibitors
FR2852954B1 (fr) *	2003-03-28	2006-07-14	Aventis Pharma Sa	Derives de quinoleines-4-substituees, leurs procede et intermediaires de preparation et les compositions pharmaceutiques qui les contiennent

2000
- 2000-11-15 FR FR0014738A patent/FR2816618B1/fr not_active Expired - Fee Related
2001
- 2001-11-13 AR ARP010105289A patent/AR034006A1/es unknown
- 2001-11-14 ES ES01996538T patent/ES2271119T3/es not_active Expired - Lifetime
- 2001-11-14 EA EA200300568A patent/EA200300568A1/ru unknown
- 2001-11-14 EP EP06010725A patent/EP1695964A1/fr not_active Withdrawn
- 2001-11-14 AU AU2002218365A patent/AU2002218365B2/en not_active Ceased
- 2001-11-14 CN CNA018210996A patent/CN1483031A/zh active Pending
- 2001-11-14 KR KR1020037006600A patent/KR100849608B1/ko not_active IP Right Cessation
- 2001-11-14 YU YU46803A patent/YU46803A/sh unknown
- 2001-11-14 EP EP01996538A patent/EP1337529B1/fr not_active Expired - Lifetime
- 2001-11-14 PL PL01363004A patent/PL363004A1/xx not_active Application Discontinuation
- 2001-11-14 AT AT01996538T patent/ATE337311T1/de not_active IP Right Cessation
- 2001-11-14 PT PT01996538T patent/PT1337529E/pt unknown
- 2001-11-14 JP JP2002543484A patent/JP2004514661A/ja active Pending
- 2001-11-14 CZ CZ20031316A patent/CZ20031316A3/cs unknown
- 2001-11-14 EE EEP200300207A patent/EE200300207A/xx unknown
- 2001-11-14 BR BR0115312-9A patent/BR0115312A/pt not_active Application Discontinuation
- 2001-11-14 DE DE60122567T patent/DE60122567T2/de not_active Expired - Fee Related
- 2001-11-14 AU AU1836502A patent/AU1836502A/xx active Pending
- 2001-11-14 TN TNTNSN01160A patent/TNSN01160A1/fr unknown
- 2001-11-14 HU HU0303758A patent/HUP0303758A3/hu unknown
- 2001-11-14 DK DK01996538T patent/DK1337529T3/da active
- 2001-11-14 IL IL15584101A patent/IL155841A0/xx unknown
- 2001-11-14 WO PCT/FR2001/003559 patent/WO2002040474A2/fr active IP Right Grant
- 2001-11-14 SK SK582-2003A patent/SK5822003A3/sk unknown
- 2001-11-14 CA CA002429311A patent/CA2429311A1/en not_active Abandoned
2003
- 2003-05-09 BG BG107793A patent/BG107793A/bg unknown
- 2003-05-13 HR HR20030379A patent/HRP20030379A2/hr not_active Application Discontinuation
- 2003-05-14 NO NO20032187A patent/NO20032187L/no unknown
- 2003-05-15 ZA ZA200303794A patent/ZA200303794B/xx unknown
2007
- 2007-04-25 NO NO20072142A patent/NO20072142L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
WO2002040474A3 (fr)	2002-10-31
BR0115312A (pt)	2003-09-23
NO20072142L (no)	2007-04-25
EA200300568A1 (ru)	2003-12-25
FR2816618A1 (fr)	2002-05-17
SK5822003A3 (en)	2004-06-08
BG107793A (bg)	2004-08-31
EP1337529A2 (fr)	2003-08-27
HRP20030379A2 (en)	2005-04-30
PT1337529E (pt)	2006-12-29
ZA200303794B (en)	2004-06-29
KR20030060934A (ko)	2003-07-16
KR100849608B1 (ko)	2008-07-31
DE60122567T2 (de)	2007-08-23
CA2429311A1 (en)	2002-05-23
ES2271119T3 (es)	2007-04-16
CZ20031316A3 (cs)	2003-10-15
EP1337529B1 (fr)	2006-08-23
AU1836502A (en)	2002-05-27
DK1337529T3 (da)	2006-12-18
WO2002040474A2 (fr)	2002-05-23
PL363004A1 (en)	2004-11-15
YU46803A (sh)	2006-05-25
JP2004514661A (ja)	2004-05-20
AU2002218365B2 (en)	2007-07-05
EE200300207A (et)	2003-08-15
FR2816618B1 (fr)	2002-12-27
HUP0303758A3 (en)	2009-08-28
HUP0303758A2 (hu)	2004-03-01
IL155841A0 (en)	2003-12-23
AR034006A1 (es)	2004-01-21
NO20032187D0 (no)	2003-05-14
EP1695964A1 (fr)	2006-08-30
CN1483031A (zh)	2004-03-17
TNSN01160A1 (fr)	2005-11-10
ATE337311T1 (de)	2006-09-15
DE60122567D1 (de)	2006-10-05

Publication	Publication Date	Title
NO20032187D0 (no)	2003-05-14	Heterocyklylalkylpiperidinderivater, deres fremstilling samt preparater inneholdende forbindelsene
NO20024175D0 (no)	2002-09-02	Azetidinderivater, deres fremstilling og farmasöytiske forbindelser inneholdende de samme
NO20010013L (no)	2001-03-01	Svovelsubstituerte sulfonylaminokarboksylsyre N-arylamider, deres fremstilling og anvendelse samt farmasöytiske preparater inneholdende forbindelsene
NO20032438D0 (no)	2003-05-28	Orto- og metasubstituerte bis-arylforbindelser, deres fremstilling og anvendelse samt farmasöytiske preparater inneholdende forbindelsene
NO20011216L (no)	2001-05-09	Azetidinderivater, deres fremstilling og medikamenter inneholdende forbindelsene
NO324250B1 (no)	2007-09-17	Diazabicykliske forbindelser, farmasoytiske sammensetninger omfattende disse samt deres anvendelse
NO20032735L (no)	2003-08-06	Difenylazetidinonderivater, fremgangsmåte for deres fremstilling, legemidler som inneholder disse forbindelsene samt deres anvendelse
NL1015859A1 (nl)	2001-07-27	Farmaceutische preparaten.
NO20015156L (no)	2001-12-18	5-pyridyl-1,3-azolforbindelser, deres fremstilling og anvendelse
IS6040A (is)	2001-08-07	Valdekoxib efnablöndur
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NO20023400L (no)	2002-09-09	Nye forbindelser med hypolidemisk og hypokolesteremisk virkning, deres fremstilling samt preparater inneholdendeforbindelsene
DK1073672T3 (da)	2003-12-08	Antipicornavirale forbindelser, deres fremstilling og anvendelse
NO20016247L (no)	2002-02-08	Streptograminderivater, deres fremstilling samt preparater inneholdende derivatene
DK1118610T3 (da)	2002-12-16	Benzensulfonamid-derivater, fremgangsmåde til fremstilling heraf samt farmaceutiske sammensætninger indeholdende derivaterne
DE59908817D1 (de)	2004-04-15	Wässrige zubereitungen
NO20024590L (no)	2002-09-25	Farmasöytiske preparater inneholdende oligosakkarider, de nye oligosakkarider samt deres fremstilling
DK1137644T3 (da)	2003-12-08	Benzofuranderivater, deres fremstilling samt anvendelse
NO20014692L (no)	2001-11-30	3-amidinobenzensulfonamidderivater, medisinske sammensetninger inneholdende slike samt intermediater vedfremstillingen derav