ZA200303794B - Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same. - Google Patents

Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same.

Info

Publication number: ZA200303794B
Authority: ZA; South Africa
Prior art keywords: preparation; compositions containing; containing same; piperidine derivatives; heterocyclylalkyl piperidine
Prior art date: 2000-11-15

Application number

ZA200303794A

Inventor

Eric Bacque

Youssef El-Ahmad

Philippe Hubert

Serge Mignani

Michel Tabart

Jean-Christophe Carry

Michel Evers

Jean-Luc Malleron

Guy Pantel

Fabrice Viviani

Original Assignee

Aventis Pharma Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-11-15

Filing date

2003-05-15

Publication date

2004-06-29

2003-05-15 Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa

2004-06-29 Publication of ZA200303794B publication Critical patent/ZA200303794B/en

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

ZA200303794A 2000-11-15 2003-05-15 Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same. ZA200303794B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR0014738A FR2816618B1 (en)	2000-11-15	2000-11-15	HETEROCYCLYLALCOYL PIPERIDINE DERIVATIVES, THEIR PREPARATION AND THE COMPOSITIONS CONTAINING THEM

Publications (1)

Publication Number	Publication Date
ZA200303794B true ZA200303794B (en)	2004-06-29

Family

ID=8856503

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA200303794A ZA200303794B (en)	2000-11-15	2003-05-15	Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same.

Country Status (28)

Country	Link
EP (2)	EP1695964A1 (en)
JP (1)	JP2004514661A (en)
KR (1)	KR100849608B1 (en)
CN (1)	CN1483031A (en)
AR (1)	AR034006A1 (en)
AT (1)	ATE337311T1 (en)
AU (2)	AU2002218365B2 (en)
BG (1)	BG107793A (en)
BR (1)	BR0115312A (en)
CA (1)	CA2429311A1 (en)
CZ (1)	CZ20031316A3 (en)
DE (1)	DE60122567T2 (en)
DK (1)	DK1337529T3 (en)
EA (1)	EA200300568A1 (en)
EE (1)	EE200300207A (en)
ES (1)	ES2271119T3 (en)
FR (1)	FR2816618B1 (en)
HR (1)	HRP20030379A2 (en)
HU (1)	HUP0303758A3 (en)
IL (1)	IL155841A0 (en)
NO (2)	NO20032187L (en)
PL (1)	PL363004A1 (en)
PT (1)	PT1337529E (en)
SK (1)	SK5822003A3 (en)
TN (1)	TNSN01160A1 (en)
WO (1)	WO2002040474A2 (en)
YU (1)	YU46803A (en)
ZA (1)	ZA200303794B (en)

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DE60125373T2 (en)	2000-07-26	2007-10-18	Smithkline Beecham P.L.C., Brentford	AMINOPIPERIDINE CHINOLINE AND ITS AZAISOSTERIC ANALOGUE WITH ANTIBACTERIAL EFFECT
GB0101577D0 (en)	2001-01-22	2001-03-07	Smithkline Beecham Plc	Compounds
GB0112834D0 (en)	2001-05-25	2001-07-18	Smithkline Beecham Plc	Medicaments
GB0112836D0 (en)	2001-05-25	2001-07-18	Smithkline Beecham Plc	Medicaments
GB0118238D0 (en) *	2001-07-26	2001-09-19	Smithkline Beecham Plc	Medicaments
WO2003064431A2 (en)	2002-01-29	2003-08-07	Glaxo Group Limited	Aminopiperidine compounds, process for their preparation, and pharmaceutical compositions containing them
EP2181996A1 (en)	2002-01-29	2010-05-05	Glaxo Group Limited	Aminopiperidine derivatives
AR040336A1 (en)	2002-06-26	2005-03-30	Glaxo Group Ltd	PIPERIDINE COMPOUND, USE OF THE SAME FOR THE MANUFACTURE OF A MEDICINAL PRODUCT, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT AND PROCEDURE TO PREPARE SUCH COMPOUND
AR040335A1 (en)	2002-06-26	2005-03-30	Glaxo Group Ltd	CYCLLOHEXAN OR CYCLHEXENE COMPOUND, USE OF THE SAME TO PREPARE A MEDICINAL PRODUCT, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT, PROCEDURE AND INTERMEDIATE COMPOUNDS OF UTILITY TO PREPARE SUCH COMPOUND
FR2842807A1 (en) *	2002-07-23	2004-01-30	Aventis Pharma Sa	QUINOLYL PROPYL PIPERIDINE DERIVATIVES, PROCESS AND PREPARATION INTERMEDIATES AND COMPOSITIONS COMPRISING THE SAME
GB0217294D0 (en) *	2002-07-25	2002-09-04	Glaxo Group Ltd	Medicaments
FR2844270B1 (en)	2002-09-11	2006-05-19	Aventis Pharma Sa	QUINOLYL PROPYL PIPERIDINE DERIVATIVES, THEIR PROCESS AND PREPARATION INTERMEDIATES AND THE COMPOSITIONS CONTAINING THEM
FR2844268B1 (en)	2002-09-11	2004-10-22	Aventis Pharma Sa	QUINOLYL PROPYL PIPERIDINE DERIVATIVES, PROCESSES AND INTERMEDIATES FOR THEIR PREPARATION, AND COMPOSITIONS CONTAINING THEM
DE10256405A1 (en) *	2002-12-02	2004-06-17	Morphochem Aktiengesellschaft für kombinatorische Chemie	New 4-substituted quinoline derivatives, useful for treating bacterial infections, optionally including additional ring nitrogens
JP4704755B2 (en)	2002-11-05	2011-06-22	グラクソスミスクライン・リミテッド・ライアビリティ・カンパニー	Antibacterial agent
EP1567520B1 (en)	2002-12-04	2008-10-15	Glaxo Group Limited	Quinolines and nitrogenated derivatives thereof and their use as antibacterial agents
FR2852954B1 (en) *	2003-03-28	2006-07-14	Aventis Pharma Sa	QUINOLINE-4-SUBSTITUTED DERIVATIVES, METHODS AND PREPARATION INTERMEDIATES THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
US7232833B2 (en)	2003-03-28	2007-06-19	Novexel	4-substituted quinoline derivatives, method and intermediates for their preparation and pharmaceutical compositions containing them
FR2862301B1 (en) *	2003-11-17	2007-12-21	Aventis Pharma Sa	NEW PROCESS FOR THE PREPARATION OF 3-FLUORINATED QUINOLINES
FR2867472B1 (en) *	2004-03-12	2008-07-18	Aventis Pharma Sa	QUINOLINE-4-SUBSTITUTED DERIVATIVES, METHODS AND PREPARATION INTERMEDIATES THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
WO2006081178A2 (en)	2005-01-25	2006-08-03	Glaxo Group Limited	Antibacterial agents
US7605169B2 (en)	2005-01-25	2009-10-20	Glaxo Group Limited	Antibacterial agents
JP2008528587A (en)	2005-01-25	2008-07-31	グラクソグループリミテッド	Antibacterial agent
EP1846418A4 (en)	2005-01-25	2009-12-23	Glaxo Group Ltd	Antibacterial agents
JP2008531709A (en)	2005-03-01	2008-08-14	ワイス	Cinnoline compounds and their use as liver X receptor modulators
MY150958A (en) *	2005-06-16	2014-03-31	Astrazeneca Ab	Compounds for the treatment of multi-drug resistant bacterial infections
CA2635126A1 (en)	2006-01-26	2007-08-02	Actelion Pharmaceuticals Ltd	Tetrahydropyrane antibiotics
WO2007115947A1 (en)	2006-04-06	2007-10-18	Glaxo Group Limited	Pyrrolo-quinoxalinone derivatives as antibacterials
EP1992628A1 (en)	2007-05-18	2008-11-19	Glaxo Group Limited	Derivatives and analogs of N-ethylquinolones and N-ethylazaquinolones
ATE520687T1 (en)	2007-06-15	2011-09-15	Actelion Pharmaceuticals Ltd	3-AMINO-6-(1-AMINO-ETHYL)-TETRAHYDROPYRANDERIVA E
EP2080761A1 (en)	2008-01-18	2009-07-22	Glaxo Group Limited	Compounds
WO2010043714A1 (en)	2008-10-17	2010-04-22	Glaxo Group Limited	Tricyclic nitrogen compounds used as antibacterials
EP2379554B1 (en)	2009-01-15	2015-11-11	Glaxo Group Limited	Naphthyridin-2(1h)-one compounds useful as antibacterials
JP6389174B2 (en) *	2012-08-15	2018-09-12	グラクソグループリミテッドＧｌａｘｏＧｒｏｕｐＬｉｍｉｔｅｄ	Chemical method
EA031589B1 (en)	2014-08-22	2019-01-31	Глэксосмитклайн Интеллекчуал Проперти Дивелопмент Лимитед	Tricyclic nitrogen containing compounds for treating neisseria gonorrhoea infection
WO2016138988A1 (en) *	2015-03-02	2016-09-09	University Of Copenhagen	Piperazine inhibitors of bacterial gyrase and topoisomerase iv
UY36851A (en)	2015-08-16	2017-03-31	Glaxosmithkline Ip Dev Ltd	COMPOUNDS FOR USE IN ANTIBACTERIAL APPLICATIONS

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
NL7908031A (en)	1979-11-01	1981-06-01	Acf Chemiefarma Nv	NEW QUINOLINE DERIVATIVES AND PHARMACEUTICAL PREPARATIONS CONTAINING SUCH A COMPOUND AND METHOD FOR PREPARING THESE COMPOUNDS.
JPH0239546A (en)	1988-07-29	1990-02-08	Origin Electric Co Ltd	Manufacture of hybrid integrated circuit
AU623474B2 (en)	1989-01-16	1992-05-14	Laboratoire Roger Bellon	New benzo(1,8)naphthyridine derivatives, their preparation and compositions containing them
ES2201674T3 (en) *	1998-01-26	2004-03-16	Smithkline Beecham Plc	DERIVATIVES OF QUINOLINA WITH ANTIBACTERIAL PROPERTIES.
AU2437900A (en) *	1999-01-20	2000-08-07	Smithkline Beecham Plc	Piperidinylquinolines as protein tyrosine kinase inhibitors
FR2852954B1 (en) *	2003-03-28	2006-07-14	Aventis Pharma Sa	QUINOLINE-4-SUBSTITUTED DERIVATIVES, METHODS AND PREPARATION INTERMEDIATES THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

2000
- 2000-11-15 FR FR0014738A patent/FR2816618B1/en not_active Expired - Fee Related
2001
- 2001-11-13 AR ARP010105289A patent/AR034006A1/en unknown
- 2001-11-14 ES ES01996538T patent/ES2271119T3/en not_active Expired - Lifetime
- 2001-11-14 EA EA200300568A patent/EA200300568A1/en unknown
- 2001-11-14 EP EP06010725A patent/EP1695964A1/en not_active Withdrawn
- 2001-11-14 AU AU2002218365A patent/AU2002218365B2/en not_active Ceased
- 2001-11-14 CN CNA018210996A patent/CN1483031A/en active Pending
- 2001-11-14 KR KR1020037006600A patent/KR100849608B1/en not_active IP Right Cessation
- 2001-11-14 YU YU46803A patent/YU46803A/en unknown
- 2001-11-14 EP EP01996538A patent/EP1337529B1/en not_active Expired - Lifetime
- 2001-11-14 PL PL01363004A patent/PL363004A1/en not_active Application Discontinuation
- 2001-11-14 AT AT01996538T patent/ATE337311T1/en not_active IP Right Cessation
- 2001-11-14 PT PT01996538T patent/PT1337529E/en unknown
- 2001-11-14 JP JP2002543484A patent/JP2004514661A/en active Pending
- 2001-11-14 CZ CZ20031316A patent/CZ20031316A3/en unknown
- 2001-11-14 EE EEP200300207A patent/EE200300207A/en unknown
- 2001-11-14 BR BR0115312-9A patent/BR0115312A/en not_active Application Discontinuation
- 2001-11-14 DE DE60122567T patent/DE60122567T2/en not_active Expired - Fee Related
- 2001-11-14 AU AU1836502A patent/AU1836502A/en active Pending
- 2001-11-14 TN TNTNSN01160A patent/TNSN01160A1/en unknown
- 2001-11-14 HU HU0303758A patent/HUP0303758A3/en unknown
- 2001-11-14 DK DK01996538T patent/DK1337529T3/en active
- 2001-11-14 IL IL15584101A patent/IL155841A0/en unknown
- 2001-11-14 WO PCT/FR2001/003559 patent/WO2002040474A2/en active IP Right Grant
- 2001-11-14 SK SK582-2003A patent/SK5822003A3/en unknown
- 2001-11-14 CA CA002429311A patent/CA2429311A1/en not_active Abandoned
2003
- 2003-05-09 BG BG107793A patent/BG107793A/en unknown
- 2003-05-13 HR HR20030379A patent/HRP20030379A2/en not_active Application Discontinuation
- 2003-05-14 NO NO20032187A patent/NO20032187L/en unknown
- 2003-05-15 ZA ZA200303794A patent/ZA200303794B/en unknown
2007
- 2007-04-25 NO NO20072142A patent/NO20072142L/en not_active Application Discontinuation

Also Published As

Publication number	Publication date
WO2002040474A3 (en)	2002-10-31
BR0115312A (en)	2003-09-23
NO20072142L (en)	2007-04-25
EA200300568A1 (en)	2003-12-25
FR2816618A1 (en)	2002-05-17
SK5822003A3 (en)	2004-06-08
BG107793A (en)	2004-08-31
EP1337529A2 (en)	2003-08-27
HRP20030379A2 (en)	2005-04-30
PT1337529E (en)	2006-12-29
KR20030060934A (en)	2003-07-16
KR100849608B1 (en)	2008-07-31
DE60122567T2 (en)	2007-08-23
CA2429311A1 (en)	2002-05-23
ES2271119T3 (en)	2007-04-16
CZ20031316A3 (en)	2003-10-15
EP1337529B1 (en)	2006-08-23
AU1836502A (en)	2002-05-27
DK1337529T3 (en)	2006-12-18
WO2002040474A2 (en)	2002-05-23
PL363004A1 (en)	2004-11-15
YU46803A (en)	2006-05-25
JP2004514661A (en)	2004-05-20
AU2002218365B2 (en)	2007-07-05
EE200300207A (en)	2003-08-15
FR2816618B1 (en)	2002-12-27
HUP0303758A3 (en)	2009-08-28
HUP0303758A2 (en)	2004-03-01
IL155841A0 (en)	2003-12-23
NO20032187L (en)	2003-06-26
AR034006A1 (en)	2004-01-21
NO20032187D0 (en)	2003-05-14
EP1695964A1 (en)	2006-08-30
CN1483031A (en)	2004-03-17
TNSN01160A1 (en)	2005-11-10
ATE337311T1 (en)	2006-09-15
DE60122567D1 (en)	2006-10-05

Publication	Publication Date	Title
ZA200303794B (en)	2004-06-29	Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same.
ZA200206905B (en)	2003-08-26	Azetidine derivatives, preparation thereof and pharmaceutical compositions containing same.
IL151209A0 (en)	2003-04-10	Pharmaceutical compositions containing 3-aminoazetidine derivatives, novel derivatives and their preparation
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HUP0400636A3 (en)	2004-09-28	Pharmaceutical compositions containing azetidine derivatives, novel azetidine derivatives and preparation thereof
AU2001237526A1 (en)	2001-11-22	Pharmaceutical compositions containing 3-amino-azetidine derivatives, novel derivatives and preparation thereof
HK1036935A1 (en)	2002-01-25	Pharmaceutical compositions.
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