MX2016008744A - Composiciones farmaceuticas que comprenden azd9291. - Google Patents

Composiciones farmaceuticas que comprenden azd9291.

Info

Publication number
MX2016008744A
MX2016008744A MX2016008744A MX2016008744A MX2016008744A MX 2016008744 A MX2016008744 A MX 2016008744A MX 2016008744 A MX2016008744 A MX 2016008744A MX 2016008744 A MX2016008744 A MX 2016008744A MX 2016008744 A MX2016008744 A MX 2016008744A
Authority
MX
Mexico
Prior art keywords
azd9291
pharmaceutical compositions
pharmaceutical
compositions
enamide
Prior art date
Application number
MX2016008744A
Other languages
English (en)
Other versions
MX367358B (es
Inventor
Wilson David
Finnie Cindy
Anthony Raw Steven
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=50191689&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2016008744(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of MX2016008744A publication Critical patent/MX2016008744A/es
Publication of MX367358B publication Critical patent/MX367358B/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente invención se relaciona con composiciones farmacéuticas adecuadas para la administración oral, y más particularmente con composiciones farmacéuticas, incluyendo composiciones de tabletas farmacéuticas, que contienen N-(2-{2-dimetilaminoetil-metilamino}-4-metoxi-5-{[4-(1-metilindol -3-il)pirimidin-2-il]amino}fenil)prop-2-enamida ("AZD9291 ") o una sal farmacéuticamente aceptable del mismo, en donde tales composiciones comprenden una cierta cantidad de celulosa microcristalina y al menos otro diluyente farmacéutico.
MX2016008744A 2014-01-02 2015-01-02 Composiciones farmaceuticas que comprenden azd9291. MX367358B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB1400034.3A GB201400034D0 (en) 2014-01-02 2014-01-02 Pharmaceutical Compositions comprising AZD9291
PCT/GB2015/050001 WO2015101791A1 (en) 2014-01-02 2015-01-02 Pharmaceutical compositions comprising azd9291

Publications (2)

Publication Number Publication Date
MX2016008744A true MX2016008744A (es) 2016-09-08
MX367358B MX367358B (es) 2019-08-16

Family

ID=50191689

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2016008744A MX367358B (es) 2014-01-02 2015-01-02 Composiciones farmaceuticas que comprenden azd9291.

Country Status (37)

Country Link
US (5) US10183020B2 (es)
EP (1) EP3089741B1 (es)
JP (1) JP6588915B2 (es)
KR (1) KR102336378B1 (es)
CN (2) CN114712362A (es)
AR (1) AR098989A1 (es)
AU (1) AU2015204218B2 (es)
CA (1) CA2933403C (es)
CL (1) CL2016001609A1 (es)
CR (1) CR20160310A (es)
CY (1) CY1124848T1 (es)
DK (1) DK3089741T3 (es)
DO (1) DOP2016000156A (es)
EA (1) EA034243B9 (es)
ES (1) ES2873226T3 (es)
GB (1) GB201400034D0 (es)
GT (1) GT201600142A (es)
HK (1) HK1225655A1 (es)
HR (1) HRP20210749T1 (es)
HU (1) HUE054344T2 (es)
IL (1) IL246186B (es)
LT (1) LT3089741T (es)
MX (1) MX367358B (es)
MY (1) MY183536A (es)
NI (1) NI201600098A (es)
NZ (1) NZ721298A (es)
PE (1) PE20161170A1 (es)
PH (1) PH12016501310A1 (es)
PL (1) PL3089741T3 (es)
PT (1) PT3089741T (es)
RS (1) RS61927B1 (es)
SG (1) SG11201605339QA (es)
SI (1) SI3089741T1 (es)
TW (1) TWI702953B (es)
UY (1) UY35933A (es)
WO (1) WO2015101791A1 (es)
ZA (1) ZA201605300B (es)

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GB201400034D0 (en) * 2014-01-02 2014-02-19 Astrazeneca Ab Pharmaceutical Compositions comprising AZD9291
EP3464275B1 (en) 2016-05-26 2024-05-08 Recurium IP Holdings, LLC Egfr inhibitor compounds
CN108057036B (zh) * 2016-11-07 2023-06-13 正大天晴药业集团股份有限公司 一种egfr抑制剂的固体药物组合物
CN107176954B (zh) * 2017-06-02 2019-01-11 无锡双良生物科技有限公司 一种egfr抑制剂的药用盐及其晶型、制备方法和应用
CN110013468B (zh) * 2018-01-09 2022-02-18 北京福元医药股份有限公司 一种azd9291氘代衍生物药物制剂
WO2019138346A1 (en) * 2018-01-10 2019-07-18 Alembic Pharmaceuticals Limited Pharmaceutical composition of osimertinib
KR20200119243A (ko) * 2018-02-12 2020-10-19 아스트라제네카 아베 비-소세포 폐암의 치료에 사용하기 위한 오시메르티닙
KR20210014621A (ko) * 2018-03-01 2021-02-09 아스트라제네카 에이비이 (2s)-n-｛(1s)-1-시아노-2-[4-(3-메틸-2-옥소-2,3-디하이드로-1,3-벤족사졸-5-일)페닐]에틸｝-1,4-옥사제판-2-카복스아미드를 포함하는 약학 조성물
JP7095108B2 (ja) * 2018-03-23 2022-07-04 ウーシー ショアンリャン バイオテクノロジー カンパニー，リミティド 医薬組成物、その製造方法及び使用
WO2020018547A1 (en) 2018-07-17 2020-01-23 Insmed Incorporated Certain (2s)-n-[(1s)-1-cyano-2-phenylethyl]-1,4-oxazepane-2-carboxamides for treating lupus nephritis
KR20200043618A (ko) * 2018-10-18 2020-04-28 주식회사유한양행 아미노피리미딘 유도체 또는 이의 염을 포함하는 경구투여용 약학 조성물
JP2022526159A (ja) 2019-03-29 2022-05-23 アストラゼネカ・アクチエボラーグ 非小細胞肺がんの治療に使用するためのオシメルチニブ
US20210161897A1 (en) 2019-11-12 2021-06-03 Astrazeneca Ab Epidermal growth factor receptor tyrosine kinase inhibitors for the treatment of cancer
CN114980883A (zh) 2020-01-20 2022-08-30 阿斯利康(瑞典)有限公司 用于治疗癌症的表皮生长因子受体酪氨酸激酶抑制剂
US20210369709A1 (en) 2020-05-27 2021-12-02 Astrazeneca Ab EGFR TKIs FOR USE IN THE TREATMENT OF NON-SMALL CELL LUNG CANCER
WO2023187037A1 (en) 2022-03-31 2023-10-05 Astrazeneca Ab Epidermal growth factor receptor (egfr) tyrosine kinase inhibitors in combination with an akt inhibitor for the treatment of cancer
WO2023209088A1 (en) 2022-04-28 2023-11-02 Astrazeneca Ab Bicyclic heteroaromatic compounds and their use in the treatment of cancer
WO2023209084A1 (en) 2022-04-28 2023-11-02 Astrazeneca Ab Condensed bicyclic heteroaromatic compounds and their use in the treatment of cancer
US20240116926A1 (en) 2022-04-28 2024-04-11 Astrazeneca Ab Heteroaromatic compounds
WO2023209090A1 (en) 2022-04-28 2023-11-02 Astrazeneca Ab Bicyclic heteroaromatic compounds and their application in the treatment of cancer
WO2024002938A1 (en) 2022-06-27 2024-01-04 Astrazeneca Ab Combinations involving epidermal growth factor receptor tyrosine kinase inhibitors for the treatment of cancer
WO2024008929A1 (en) 2022-07-08 2024-01-11 Astrazeneca Ab Epidermal growth factor receptor tyrosine kinase inhibitors in combination with hgf-receptor inhibitors for the treatment of cancer

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UA76325C2 (uk) 2002-02-26 2006-07-17 Астразенека Аб Лікарський препарат іресси, який містить водорозчинне похідне целюлози (варіанти), та спосіб його одержання
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CN105254616B (zh) * 2011-07-27 2017-10-17 阿斯利康(瑞典)有限公司 取代的n‑(2‑甲氧基‑5‑硝基苯基)嘧啶‑2‑胺化合物及其盐
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Also Published As

Publication number Publication date
US20200360378A1 (en) 2020-11-19
US20220395502A1 (en) 2022-12-15
EP3089741A1 (en) 2016-11-09
KR102336378B1 (ko) 2021-12-08
KR20160101720A (ko) 2016-08-25
DOP2016000156A (es) 2016-08-15
CA2933403C (en) 2022-03-29
LT3089741T (lt) 2021-06-10
JP2017501201A (ja) 2017-01-12
ES2873226T3 (es) 2021-11-03
PL3089741T3 (pl) 2021-09-27
DK3089741T3 (da) 2021-06-07
AU2015204218A1 (en) 2016-07-07
US20240189310A1 (en) 2024-06-13
WO2015101791A1 (en) 2015-07-09
EA034243B9 (ru) 2020-04-10
US10183020B2 (en) 2019-01-22
TW201609101A (zh) 2016-03-16
PE20161170A1 (es) 2016-11-24
EA201691242A1 (ru) 2016-12-30
EP3089741B1 (en) 2021-03-10
AU2015204218B2 (en) 2017-06-15
CN105848647B (zh) 2022-04-26
HUE054344T2 (hu) 2021-08-30
RS61927B1 (sr) 2021-06-30
HK1225655A1 (zh) 2017-09-15
IL246186A0 (en) 2016-07-31
US20160324854A1 (en) 2016-11-10
CY1124848T1 (el) 2022-11-25
EA034243B1 (ru) 2020-01-21
NZ721298A (en) 2017-10-27
CR20160310A (es) 2016-09-23
ZA201605300B (en) 2022-10-26
SI3089741T1 (sl) 2021-08-31
AR098989A1 (es) 2016-06-22
NI201600098A (es) 2016-12-20
CL2016001609A1 (es) 2016-12-09
HRP20210749T1 (hr) 2021-06-25
CA2933403A1 (en) 2015-07-09
TWI702953B (zh) 2020-09-01
IL246186B (en) 2020-07-30
JP6588915B2 (ja) 2019-10-09
CN114712362A (zh) 2022-07-08
UY35933A (es) 2015-07-31
MX367358B (es) 2019-08-16
SG11201605339QA (en) 2016-07-28
MY183536A (en) 2021-02-25
PH12016501310A1 (en) 2016-09-14
GT201600142A (es) 2019-08-12
CN105848647A (zh) 2016-08-10
PT3089741T (pt) 2021-06-11
GB201400034D0 (en) 2014-02-19
US20190111057A1 (en) 2019-04-18

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