MA28478B1 - Derive du benzimidazole et ses utilisations - Google Patents
Derive du benzimidazole et ses utilisationsInfo
- Publication number
- MA28478B1 MA28478B1 MA29333A MA29333A MA28478B1 MA 28478 B1 MA28478 B1 MA 28478B1 MA 29333 A MA29333 A MA 29333A MA 29333 A MA29333 A MA 29333A MA 28478 B1 MA28478 B1 MA 28478B1
- Authority
- MA
- Morocco
- Prior art keywords
- benzimidazole derivative
- benzimidazole
- derivative
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4245—Oxadiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Diabetes (AREA)
- Heart & Thoracic Surgery (AREA)
- Neurosurgery (AREA)
- Cardiology (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Epidemiology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Urology & Nephrology (AREA)
- Hospice & Palliative Care (AREA)
- Vascular Medicine (AREA)
- Psychiatry (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pyrrole Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2004048928 | 2004-02-25 | ||
US11/031,057 US7157584B2 (en) | 2004-02-25 | 2005-01-07 | Benzimidazole derivative and use thereof |
Publications (1)
Publication Number | Publication Date |
---|---|
MA28478B1 true MA28478B1 (fr) | 2007-03-01 |
Family
ID=34858222
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MA29333A MA28478B1 (fr) | 2004-02-25 | 2006-09-22 | Derive du benzimidazole et ses utilisations |
Country Status (33)
Country | Link |
---|---|
US (3) | US7157584B2 (fr) |
EP (3) | EP2119715B1 (fr) |
JP (2) | JP4256852B2 (fr) |
KR (1) | KR101080029B1 (fr) |
CN (2) | CN100503605C (fr) |
AR (2) | AR047972A1 (fr) |
AT (2) | ATE370136T1 (fr) |
AU (1) | AU2005214271B8 (fr) |
BR (2) | BR122012009489B8 (fr) |
CA (1) | CA2557538C (fr) |
CY (5) | CY1107008T1 (fr) |
DE (3) | DE602005002030T2 (fr) |
DK (3) | DK1857457T3 (fr) |
ES (3) | ES2293552T3 (fr) |
HK (2) | HK1098472A1 (fr) |
HR (3) | HRP20070510T3 (fr) |
HU (1) | HUS1200008I1 (fr) |
IL (1) | IL177533A (fr) |
LU (1) | LU91962I2 (fr) |
MA (1) | MA28478B1 (fr) |
ME (2) | ME01643B (fr) |
MY (1) | MY142807A (fr) |
NL (1) | NL300802I2 (fr) |
NO (2) | NO332344B1 (fr) |
NZ (1) | NZ549755A (fr) |
PL (3) | PL1857457T3 (fr) |
PT (3) | PT2119715E (fr) |
RS (3) | RS52376B (fr) |
RU (2) | RU2501798C2 (fr) |
SI (3) | SI1718641T1 (fr) |
TW (1) | TWI336702B (fr) |
WO (1) | WO2005080384A2 (fr) |
ZA (1) | ZA200607241B (fr) |
Families Citing this family (80)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7157584B2 (en) * | 2004-02-25 | 2007-01-02 | Takeda Pharmaceutical Company Limited | Benzimidazole derivative and use thereof |
JP4966202B2 (ja) | 2004-12-24 | 2012-07-04 | スピニフェクス ファーマシューティカルズ ピーティーワイ リミテッド | 治療または予防のための方法 |
JP4465469B2 (ja) * | 2005-02-21 | 2010-05-19 | 国立大学法人佐賀大学 | 循環器病マーカーとしてのインターロイキン13 |
KR20070116648A (ko) * | 2005-03-30 | 2007-12-10 | 다케다 야쿠힌 고교 가부시키가이샤 | 벤즈이미다졸 유도체 및 안지오텐신 ⅱ 길항제로서의 용도 |
JP5047156B2 (ja) * | 2006-02-27 | 2012-10-10 | 武田薬品工業株式会社 | 医薬パッケージ |
WO2007097452A1 (fr) * | 2006-02-27 | 2007-08-30 | Takeda Pharmaceutical Company Limited | Emballage-coque à usage médical |
CA2646379C (fr) | 2006-03-20 | 2014-12-23 | The University Of Queensland | Methode de traitement prophylactique ou therapeutique |
US20090308780A1 (en) * | 2006-09-25 | 2009-12-17 | Takeda Pharmaceutical Company Limited | Medicinal package |
CN101677961B (zh) * | 2007-03-28 | 2012-10-17 | 武田药品工业株式会社 | 包含苯并咪唑-7-羧酸酯衍生物和pH控制剂的固体药物组合物 |
JP2009062296A (ja) * | 2007-09-05 | 2009-03-26 | Fujifilm Corp | カルボン酸エステル化合物の製造方法 |
EP2253318B1 (fr) * | 2008-03-13 | 2014-08-06 | Daiichi Sankyo Company, Limited | Amélioration de la solubilité d'une préparation contenant de l'olmésartan médoxomil |
NZ590948A (en) * | 2008-07-31 | 2012-06-29 | Takeda Pharmaceutical | Solid pharmaceutical composition comprising a diuretic, ph control agent and an oxadiazole |
AR073380A1 (es) | 2008-09-25 | 2010-11-03 | Takeda Pharmaceutical | Composicion farmaceutica solida. comprimido multicapa |
MX2011004258A (es) * | 2008-10-22 | 2011-06-01 | Merck Sharp & Dohme | Derivados de bencimidazol ciclicos novedosos utiles como agentes anti-diabeticos. |
WO2010075347A2 (fr) | 2008-12-23 | 2010-07-01 | Takeda Pharmaceutical Company Limited | Méthode de traitement de l'hypertension avec au moins un agent bloquant les récepteurs d'angiotensine ii et de la chlorthalidone |
US20110009347A1 (en) * | 2009-07-08 | 2011-01-13 | Yin Liang | Combination therapy for the treatment of diabetes |
MX339570B (es) | 2010-05-11 | 2016-05-31 | Janssen Pharmaceutica Nv | Formulaciones farmaceuticas que comprenden derivados de 1-(beta-d-glucopiranosil)-2-tienil-metilbenceno como inhibidores de transportadores de glucosa dependientes de sodio. |
WO2012090043A1 (fr) * | 2010-12-29 | 2012-07-05 | Jubilant Life Sciences Limited | Nouvelles formes à l'état solide d'azilsartan médoxomil et leur procédé de préparation |
JP5981940B2 (ja) | 2011-01-20 | 2016-08-31 | ジエンス ハンセン ファーマセウティカル カンパニー リミテッド | アジルサルタン有機アミン塩、その製造方法及び使用 |
US9233955B2 (en) | 2011-02-08 | 2016-01-12 | Jubilant Life Sciences, Ltd. | Process for the preparation of azilsartan medoxomil |
CN102138899B (zh) * | 2011-03-18 | 2013-08-21 | 海南本创医药科技有限公司 | 阿齐沙坦酯脂质体固体制剂 |
EA028946B1 (ru) | 2011-04-13 | 2018-01-31 | Янссен Фармацевтика Нв | Способ получения соединений для применения в качестве ингибиторов sglt2 |
CN102827153B (zh) * | 2011-06-14 | 2016-10-05 | 江苏豪森药业集团有限公司 | 阿齐沙坦的晶型及其制备方法 |
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WO2013042066A1 (fr) * | 2011-09-20 | 2013-03-28 | Ranbaxy Laboratories Limited | Procédé de préparation d'azilsartan médoxomil |
WO2013042067A1 (fr) | 2011-09-20 | 2013-03-28 | Ranbaxy Laboratories Limited | Procédé de préparation d'un sel de potassium de l'azilsartan médoxomil |
WO2013088384A2 (fr) | 2011-12-15 | 2013-06-20 | Jubilant Life Sciences Limited | Formes à l'état solide d'azilsartan et d'azilsartan médoxomil monopotassique et leur procédé de préparation |
US20130158080A1 (en) | 2011-12-15 | 2013-06-20 | Takeda Pharmaceuticals U.S.A., Inc. | Methods for treating hypertension in black patients |
WO2013104342A1 (fr) * | 2012-01-14 | 2013-07-18 | Sunshine Lake Pharma Co., Ltd. | Formes cristallines de l'azilsartan médoxomil potassique et préparation et utilisations de celles-ci |
EP2814826A1 (fr) * | 2012-02-02 | 2014-12-24 | Ranbaxy Laboratories Limited | Procédé de préparation d'azilsartan médoxomil ou de ses sels pharmaceutiquement acceptables |
WO2013124748A1 (fr) * | 2012-02-20 | 2013-08-29 | Alembic Pharmaceuticals Limited | Nouveaux polymorphes d'azilsartan médoxomil potassique |
CZ2012274A3 (cs) * | 2012-04-19 | 2013-10-30 | Zentiva, K.S. | Zpusob prípravy vysoce cisté draselné soli azilsartanu medoxomilu |
WO2013186792A2 (fr) * | 2012-06-11 | 2013-12-19 | Msn Laboratories Limited | Procédé de préparation de 2-éthoxy-1-{[2'-(5-oxo-4,5-dihydro-1,2,4- oxadiazol-3-yl)biphényl-4-yl]méthyl}-lh-benzimidazole-7-carboxylate de (5-méthyl-2-oxo-l,3-dioxol-4-yl)méthyle et de ses sels |
WO2014009969A2 (fr) * | 2012-07-09 | 2014-01-16 | Hetero Research Foundation | Nouveaux polymorphes d'azilsartan |
WO2014020381A1 (fr) * | 2012-08-01 | 2014-02-06 | Alembic Pharmaceuticals Limited | Forme cristalline inédite d'azilsartan médoxomil potassique |
US9314753B2 (en) | 2012-08-27 | 2016-04-19 | Stempeutics Research Private Limited | Multi plane mixer and separator (MPMS) system |
CZ305318B6 (cs) * | 2012-09-26 | 2015-07-29 | Zentiva, K.S. | Způsob přípravy vysoce čisté draselné soli azilsartanu medoxomilu |
WO2014049512A2 (fr) | 2012-09-26 | 2014-04-03 | Lupin Limited | Nouveau procédé de préparation d'azilsartan médoxomil |
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IN2015DN03071A (fr) * | 2012-10-09 | 2015-10-02 | Avery Dennison Corp | |
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WO2015051546A1 (fr) * | 2013-10-12 | 2015-04-16 | 杭州领业医药科技有限公司 | Formes cristallines de l'ester d'azilsartan et leur procédé de préparation |
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CZ2014702A3 (cs) | 2014-10-15 | 2016-04-27 | Zentiva, K.S. | Způsob přípravy vysoce čistého azilsartanu |
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US20200179369A1 (en) * | 2015-07-29 | 2020-06-11 | Takeda Gmbh | Treatment of diabetic nephropathy |
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JP6856365B2 (ja) * | 2016-11-30 | 2021-04-07 | 株式会社トクヤマ | アジルサルタンの製造方法 |
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EP3461822B1 (fr) * | 2016-07-11 | 2022-11-02 | Wuhan LL Science And Technology Development Co., Ltd. | Forme cristalline de composé chimique, son procédé de préparation, sa composition et son application |
RU2623082C1 (ru) * | 2016-07-11 | 2017-06-21 | Государственное бюджетное образовательное учреждение высшего профессионального образования "Курский государственный медицинский университет" Министерства здравоохранения Российской Федерации | Способ коррекции артериальной ригидности у больных ревматоидным артритом |
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WO2018064945A1 (fr) * | 2016-10-08 | 2018-04-12 | 武汉朗来科技发展有限公司 | Composition pharmaceutique |
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CN110237071B (zh) * | 2018-03-09 | 2022-03-22 | 武汉朗来科技发展有限公司 | 药物制剂及其应用 |
CN110237072B (zh) * | 2018-03-09 | 2022-03-25 | 武汉朗来科技发展有限公司 | 药物组合物的制备方法 |
US11081240B2 (en) | 2018-06-14 | 2021-08-03 | Astrazeneca Uk Limited | Methods for treatment of hypertension with an angiotensin II receptor blocker pharmaceutical composition |
WO2019241519A1 (fr) * | 2018-06-14 | 2019-12-19 | Astrazeneca Uk Limited | Méthodes de diminution de la tension artérielle avec une composition pharmaceutique de blocage de canal calcique de type dihydropyridine |
WO2020101450A1 (fr) | 2018-11-16 | 2020-05-22 | 엠에프씨 주식회사 | Composés dérivés d'azilsartan, leurs intermédiaires, leur procédé de préparation et composition pharmaceutique les comprenant |
WO2020166710A1 (fr) | 2019-02-15 | 2020-08-20 | 国立大学法人東北大学 | Dérivé de 1, 3-dioxolane |
KR102220011B1 (ko) | 2020-05-15 | 2021-02-25 | 대봉엘에스 주식회사 | 친환경 용매를 이용한 아질사탄의 제조방법 및 이에 관한 핵심 중간체 화합물 |
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