HK1174334A1 - Compounds that inhibit (block) bitter taste in compositions and use thereof () - Google Patents

Compounds that inhibit (block) bitter taste in compositions and use thereof ()

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Publication number
HK1174334A1
HK1174334A1 HK13101711.1A HK13101711A HK1174334A1 HK 1174334 A1 HK1174334 A1 HK 1174334A1 HK 13101711 A HK13101711 A HK 13101711A HK 1174334 A1 HK1174334 A1 HK 1174334A1
Authority
HK
Hong Kong
Prior art keywords
inhibit
compositions
compounds
block
bitter taste
Prior art date
Application number
HK13101711.1A
Other languages
English (en)
Chinese (zh)
Inventor
Xiaodong Li
Vincent Darmohusodo
Melissa Arellano
Victor Selchau
Brett Weylan Ching
Donald S Karanewsky
Paul Brust
Jing Ling
Wen Zhao
Chad Priest
Andrew Patron
Catherine Tachdjian
Hong Xu
Qing Li
Alexey Pronin
Guy Servant
Lan Zhang
Thomas Brady
Original Assignee
Senomyx Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Senomyx Inc filed Critical Senomyx Inc
Publication of HK1174334A1 publication Critical patent/HK1174334A1/xx

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/15—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C311/16—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to hydrogen atoms or to an acyclic carbon atom
    • C07C311/17—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to hydrogen atoms or to an acyclic carbon atom to an acyclic carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23L—FOODS, FOODSTUFFS, OR NON-ALCOHOLIC BEVERAGES, NOT COVERED BY SUBCLASSES A21D OR A23B-A23J; THEIR PREPARATION OR TREATMENT, e.g. COOKING, MODIFICATION OF NUTRITIVE QUALITIES, PHYSICAL TREATMENT; PRESERVATION OF FOODS OR FOODSTUFFS, IN GENERAL
    • A23L27/00—Spices; Flavouring agents or condiments; Artificial sweetening agents; Table salts; Dietetic salt substitutes; Preparation or treatment thereof
    • A23L27/86—Addition of bitterness inhibitors
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    • A61K8/4933—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom having sulfur as an exocyclic substituent, e.g. pyridinethione
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    • A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
    • A61K8/494—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with more than one nitrogen as the only hetero atom
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    • A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
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    • A61K8/4973—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with oxygen as the only hetero atom
    • A61K8/498—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with oxygen as the only hetero atom having 6-membered rings or their condensed derivatives, e.g. coumarin
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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CA2696995A1 (fr) 2009-02-26
EP2195656A2 (fr) 2010-06-16
US20090274632A1 (en) 2009-11-05
CL2008002473A1 (es) 2009-03-27
KR101558193B1 (ko) 2015-10-12
TW200912306A (en) 2009-03-16
RU2010110557A (ru) 2011-09-27
EP2195656A4 (fr) 2011-10-19
KR20100076949A (ko) 2010-07-06
BRPI0815634B1 (pt) 2024-01-09
KR101599715B1 (ko) 2016-03-08
RU2522456C2 (ru) 2014-07-10
CN104130247A (zh) 2014-11-05
CN101828111B (zh) 2014-07-23
EP2487169B1 (fr) 2015-05-20
CN104130247B (zh) 2018-06-01
US8148544B2 (en) 2012-04-03
CA2982520A1 (fr) 2009-02-26
US20110207937A1 (en) 2011-08-25
CZ2010180A3 (cs) 2010-10-13
US7939671B2 (en) 2011-05-10
WO2009025793A3 (fr) 2009-05-14
ES2545121T3 (es) 2015-09-08
MX2010001995A (es) 2010-06-09
CN101828111A (zh) 2010-09-08
AU2008289485B2 (en) 2014-08-14
TWI482967B (zh) 2015-05-01
KR20150034819A (ko) 2015-04-03
NZ583350A (en) 2012-03-30
AU2008289485A1 (en) 2009-02-26
EP2487169A1 (fr) 2012-08-15
CA2696995C (fr) 2017-11-21
WO2009025793A8 (fr) 2009-07-30
BRPI0815634A2 (pt) 2015-02-18
RO128637A2 (ro) 2013-07-30
HUE025137T2 (en) 2016-01-28
WO2009025793A2 (fr) 2009-02-26
US20130183252A1 (en) 2013-07-18

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