FI870113A - Menetelmä uusien terapeuttisesti käyttökelpoisten 4,5,6-substioitujenN-(substituoitu-fenyyli)-2-pyrimidiiniamiinien valmistamiseksi - Google Patents

Menetelmä uusien terapeuttisesti käyttökelpoisten 4,5,6-substioitujenN-(substituoitu-fenyyli)-2-pyrimidiiniamiinien valmistamiseksi Download PDF

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Publication number
FI870113A
FI870113A FI870113A FI870113A FI870113A FI 870113 A FI870113 A FI 870113A FI 870113 A FI870113 A FI 870113A FI 870113 A FI870113 A FI 870113A FI 870113 A FI870113 A FI 870113A
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FI
Finland
Prior art keywords
substituted
phenyl
pyrimidineamines
preparation
therapeutically useful
Prior art date
Application number
FI870113A
Other languages
English (en)
Swedish (sv)
Other versions
FI91150C (fi
FI91150B (fi
FI870113A0 (fi
Inventor
Lawrence Wayne Torley
Bernard D Johnson
John Paul Dusza
Original Assignee
American Cyanamid Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=25224278&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI870113(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by American Cyanamid Co filed Critical American Cyanamid Co
Publication of FI870113A0 publication Critical patent/FI870113A0/fi
Publication of FI870113A publication Critical patent/FI870113A/fi
Application granted granted Critical
Publication of FI91150B publication Critical patent/FI91150B/fi
Publication of FI91150C publication Critical patent/FI91150C/fi

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/14Antitussive agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
FI870113A 1986-01-13 1987-01-13 Menetelmä uusien terapeuttisesti käyttökelpoisten 4,5,6-substioitujenN-(substituoitu-fenyyli)-2-pyrimidiiniamiinien valmistamiseksi FI91150C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US81795186A 1986-01-13 1986-01-13
US81795186 1986-01-13

Publications (4)

Publication Number Publication Date
FI870113A0 FI870113A0 (fi) 1987-01-13
FI870113A true FI870113A (fi) 1987-07-14
FI91150B FI91150B (fi) 1994-02-15
FI91150C FI91150C (fi) 1994-05-25

Family

ID=25224278

Family Applications (1)

Application Number Title Priority Date Filing Date
FI870113A FI91150C (fi) 1986-01-13 1987-01-13 Menetelmä uusien terapeuttisesti käyttökelpoisten 4,5,6-substioitujenN-(substituoitu-fenyyli)-2-pyrimidiiniamiinien valmistamiseksi

Country Status (18)

Country Link
EP (1) EP0233461B2 (fi)
JP (1) JPH0780857B2 (fi)
KR (1) KR900004693B1 (fi)
AT (1) ATE135699T1 (fi)
AU (2) AU591223B2 (fi)
BR (1) BR1100989A (fi)
CA (1) CA1320201C (fi)
DE (1) DE3751742T3 (fi)
DK (1) DK171251B1 (fi)
ES (1) ES2087056T3 (fi)
FI (1) FI91150C (fi)
GR (1) GR3019455T3 (fi)
HU (1) HU198708B (fi)
IE (1) IE74202B1 (fi)
NZ (1) NZ218924A (fi)
PH (1) PH25056A (fi)
SG (1) SG47583A1 (fi)
ZA (1) ZA87219B (fi)

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Also Published As

Publication number Publication date
IE74202B1 (en) 1997-07-16
DE3751742T2 (de) 1996-11-21
GR3019455T3 (en) 1996-06-30
FI91150C (fi) 1994-05-25
KR870007154A (ko) 1987-08-17
ZA87219B (en) 1987-08-26
SG47583A1 (en) 1998-04-17
DK171251B1 (da) 1996-08-12
AU5057890A (en) 1990-07-26
NZ218924A (en) 1990-04-26
AU6751887A (en) 1987-07-16
EP0233461A2 (en) 1987-08-26
ES2087056T3 (es) 1996-07-16
DK15187D0 (da) 1987-01-13
JPH0780857B2 (ja) 1995-08-30
AU591223B2 (en) 1989-11-30
EP0233461A3 (en) 1988-05-25
FI91150B (fi) 1994-02-15
EP0233461B1 (en) 1996-03-20
DE3751742D1 (de) 1996-04-25
HUT43582A (en) 1987-11-30
FI870113A0 (fi) 1987-01-13
BR1100989A (pt) 1999-11-09
CA1320201C (en) 1993-07-13
EP0233461B2 (en) 2002-05-29
HU198708B (en) 1989-11-28
DK15187A (da) 1987-07-14
ATE135699T1 (de) 1996-04-15
DE3751742T3 (de) 2002-11-21
PH25056A (en) 1991-01-28
IE870074L (en) 1987-07-13
KR900004693B1 (ko) 1990-07-02
AU621461B2 (en) 1992-03-12
JPS62223177A (ja) 1987-10-01

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Owner name: AMERICAN CYANAMID COMPANY