DK1194426T3 - Benzofuranderivater - Google Patents

Benzofuranderivater

Info

Publication number: DK1194426T3
Authority: DK; Denmark
Prior art keywords: benzofuran
Prior art date: 1999-07-10

Application number

DK00949229T

Other languages

English (en)

Inventor

Andreas Bathe

Henning Boettcher

Bernd Helfert

Original Assignee

Merck Patent Gmbh

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-07-10

Filing date

2000-06-29

Publication date

2004-12-20

2000-06-29 Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh

2004-12-20 Application granted granted Critical

2004-12-20 Publication of DK1194426T3 publication Critical patent/DK1194426T3/da

Links

IANQTJSKSUMEQM-UHFFFAOYSA-N 1-benzofuran Chemical compound C1=CC=C2OC=CC2=C1 IANQTJSKSUMEQM-UHFFFAOYSA-N 0.000 title 2

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/82—Benzo [b] furans; Hydrogenated benzo [b] furans with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D307/84—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D307/85—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 2
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

DK00949229T 1999-07-10 2000-06-29 Benzofuranderivater DK1194426T3 (da)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
DE19932314A DE19932314A1 (de)	1999-07-10	1999-07-10	Benzofuranderivate
PCT/EP2000/006089 WO2001004112A2 (de)	1999-07-10	2000-06-29	Benzofuranderivate
EP00949229A EP1194426B1 (de)	1999-07-10	2000-06-29	Benzofuranderivate

Publications (1)

Publication Number	Publication Date
DK1194426T3 true DK1194426T3 (da)	2004-12-20

Family

ID=7914351

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK00949229T DK1194426T3 (da)	1999-07-10	2000-06-29	Benzofuranderivater

Country Status (29)

Country	Link
US (1)	US6531503B1 (da)
EP (1)	EP1194426B1 (da)
JP (1)	JP4908706B2 (da)
KR (1)	KR100709378B1 (da)
CN (1)	CN1178934C (da)
AR (1)	AR024671A1 (da)
AT (1)	ATE273973T1 (da)
AU (1)	AU767413B2 (da)
BR (1)	BRPI0012329B8 (da)
CA (1)	CA2378603C (da)
CZ (1)	CZ301441B6 (da)
DE (2)	DE19932314A1 (da)
DK (1)	DK1194426T3 (da)
ES (1)	ES2226884T3 (da)
HK (1)	HK1047275B (da)
HU (1)	HU229135B1 (da)
IL (2)	IL147494A0 (da)
MX (1)	MXPA02000316A (da)
MY (1)	MY122667A (da)
NO (1)	NO328209B1 (da)
PL (1)	PL196477B1 (da)
PT (1)	PT1194426E (da)
RU (1)	RU2278862C2 (da)
SI (1)	SI1194426T1 (da)
SK (1)	SK287360B6 (da)
TR (1)	TR200200017T2 (da)
UA (1)	UA73310C2 (da)
WO (1)	WO2001004112A2 (da)
ZA (1)	ZA200201085B (da)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE102006060597A1 (de) *	2006-12-21	2008-06-26	Merck Patent Gmbh	Verfahren zur Herstellung von Benzofuran-2-carboxamiden
EP2110374A1 (en) *	2008-04-18	2009-10-21	Merck Sante	Benzofurane, benzothiophene, benzothiazol derivatives as FXR modulators
TWI477497B (zh)	2009-03-10	2015-03-21	Takeda Pharmaceutical	苯并呋喃衍生物
WO2011140161A1 (en)	2010-05-06	2011-11-10	Bristol-Myers Squibb Company	Benzofuranyl analogues as gpr119 modulators
EP2566860B1 (en)	2010-05-06	2014-09-10	Bristol-Myers Squibb Company	Bicyclic heteroaryl compounds as gpr119 modulators
CN102964323B (zh) *	2012-11-13	2015-03-25	苏州永健生物医药有限公司	一种5-（哌嗪-1-基）苯并呋喃-2-甲酰胺的合成方法
PL3009424T3 (pl) *	2013-06-10	2018-03-30	Astellas Pharma Inc.	Bicykliczny zawierający azot aromatyczny heterocykliczny związek amidowy

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US2724915A (en) *		1955-11-29		Snow remover
DE2757532A1 (de) *	1977-12-23	1979-07-05	Hoechst Ag	N,n'-disubstituiertes cyclisches diamin und verfahren zu dessen herstellung
WO1994029290A1 (en) *	1993-06-14	1994-12-22	Pfizer Inc.	Secondary amines as antidiabetic and antiobesity agents
DE4333254A1 (de)	1993-09-30	1995-04-06	Merck Patent Gmbh	Piperidine und Piperazine
DE19514567A1 (de) *	1995-04-20	1996-10-24	Merck Patent Gmbh	Benzofurane

1999
- 1999-07-10 DE DE19932314A patent/DE19932314A1/de not_active Withdrawn
2000
- 2000-06-29 HU HU0201903A patent/HU229135B1/hu not_active IP Right Cessation
- 2000-06-29 EP EP00949229A patent/EP1194426B1/de not_active Expired - Lifetime
- 2000-06-29 JP JP2001509722A patent/JP4908706B2/ja not_active Expired - Fee Related
- 2000-06-29 CA CA2378603A patent/CA2378603C/en not_active Expired - Fee Related
- 2000-06-29 DK DK00949229T patent/DK1194426T3/da active
- 2000-06-29 UA UA2002021055A patent/UA73310C2/uk unknown
- 2000-06-29 PT PT00949229T patent/PT1194426E/pt unknown
- 2000-06-29 MX MXPA02000316A patent/MXPA02000316A/es active IP Right Grant
- 2000-06-29 RU RU2002102234/04A patent/RU2278862C2/ru not_active IP Right Cessation
- 2000-06-29 SI SI200030518T patent/SI1194426T1/xx unknown
- 2000-06-29 CZ CZ20020011A patent/CZ301441B6/cs not_active IP Right Cessation
- 2000-06-29 AU AU62665/00A patent/AU767413B2/en not_active Ceased
- 2000-06-29 IL IL14749400A patent/IL147494A0/xx active IP Right Grant
- 2000-06-29 BR BRPI0012329A patent/BRPI0012329B8/pt not_active IP Right Cessation
- 2000-06-29 KR KR1020017015565A patent/KR100709378B1/ko not_active IP Right Cessation
- 2000-06-29 US US10/030,471 patent/US6531503B1/en not_active Expired - Lifetime
- 2000-06-29 AT AT00949229T patent/ATE273973T1/de active
- 2000-06-29 SK SK6-2002A patent/SK287360B6/sk not_active IP Right Cessation
- 2000-06-29 CN CNB008093083A patent/CN1178934C/zh not_active Expired - Fee Related
- 2000-06-29 WO PCT/EP2000/006089 patent/WO2001004112A2/de active IP Right Grant
- 2000-06-29 DE DE50007501T patent/DE50007501D1/de not_active Expired - Lifetime
- 2000-06-29 PL PL353157A patent/PL196477B1/pl not_active IP Right Cessation
- 2000-06-29 TR TR2002/00017T patent/TR200200017T2/xx unknown
- 2000-06-29 ES ES00949229T patent/ES2226884T3/es not_active Expired - Lifetime
- 2000-07-06 MY MYPI20003075A patent/MY122667A/en unknown
- 2000-07-07 AR ARP000103465A patent/AR024671A1/es active IP Right Grant
2002
- 2002-01-06 IL IL147494A patent/IL147494A/en not_active IP Right Cessation
- 2002-01-09 NO NO20020095A patent/NO328209B1/no not_active IP Right Cessation
- 2002-02-07 ZA ZA200201085A patent/ZA200201085B/en unknown
- 2002-11-29 HK HK02108676.2A patent/HK1047275B/zh unknown

Also Published As

Publication number	Publication date
WO2001004112A2 (de)	2001-01-18
NO20020095L (no)	2002-01-09
SK287360B6 (sk)	2010-08-09
HUP0201903A3 (en)	2005-02-28
NO20020095D0 (no)	2002-01-09
JP2003504364A (ja)	2003-02-04
AU767413B2 (en)	2003-11-06
EP1194426A2 (de)	2002-04-10
SK62002A3 (en)	2002-05-09
CZ301441B6 (cs)	2010-03-03
PL353157A1 (en)	2003-10-20
CN1356996A (zh)	2002-07-03
JP4908706B2 (ja)	2012-04-04
ZA200201085B (en)	2003-07-30
BRPI0012329B8 (pt)	2021-05-25
HK1047275B (zh)	2005-09-02
KR20020016815A (ko)	2002-03-06
EP1194426B1 (de)	2004-08-18
CA2378603C (en)	2010-05-11
US6531503B1 (en)	2003-03-11
DE19932314A1 (de)	2001-01-11
PT1194426E (pt)	2005-01-31
ATE273973T1 (de)	2004-09-15
CN1178934C (zh)	2004-12-08
SI1194426T1 (en)	2005-02-28
MY122667A (en)	2006-04-29
NO328209B1 (no)	2010-01-11
KR100709378B1 (ko)	2007-04-20
AR024671A1 (es)	2002-10-23
AU6266500A (en)	2001-01-30
CA2378603A1 (en)	2001-01-18
DE50007501D1 (de)	2004-09-23
WO2001004112A3 (de)	2001-08-02
IL147494A0 (en)	2002-08-14
HUP0201903A2 (en)	2002-10-28
PL196477B1 (pl)	2008-01-31
ES2226884T3 (es)	2005-04-01
HU229135B1 (en)	2013-08-28
IL147494A (en)	2008-03-20
UA73310C2 (en)	2005-07-15
RU2278862C2 (ru)	2006-06-27
BR0012329A (pt)	2002-03-19
MXPA02000316A (es)	2002-07-30
CZ200211A3 (cs)	2002-04-17
BR0012329B1 (pt)	2013-03-19
TR200200017T2 (tr)	2002-05-21
HK1047275A1 (en)	2003-02-14

Publication	Publication Date	Title
NO20016115L (no)	2002-02-12	Substituerte heterosykelkondenserte gamma-karbolin
PT1224180E (pt)	2003-11-28	Azois substituidos
DE122007000064I1 (de)	2008-01-03	Erythropoietinkonjugate
DE19983871T1 (de)	2002-01-31	Fönvorrichtung
DE10084676T1 (de)	2003-04-30	Einmallanzettvorrichtung
DE50002834D1 (de)	2003-08-14	Handstempel
ATE357433T1 (de)	2007-04-15	4-pyrimidinyl-n-acyl-l-phenylanine
ATE297895T1 (de)	2005-07-15	4-pyridinyl-n-acyl-l-phenylalanine
FI4433U1 (fi)	2000-06-02	Hiustenmuotoilusakset
DE50000805D1 (de)	2003-01-09	Aufsitzspanner
DE10085008T1 (de)	2002-10-10	Oberflächenbehandlungsdüse
DK1194426T3 (da)	2004-12-20	Benzofuranderivater
NO20025474L (no)	2003-01-07	Benzofuranderivater
DE19983890T1 (de)	2002-03-07	Ventiltaktgebungsjustiereinrichtung
NO20022927D0 (no)	2002-06-18	Substituerte pyrrazoler
DE50001640D1 (de)	2003-05-08	Nahfeldoptische untersuchungsvorrichtung
ATE269311T1 (de)	2004-07-15	Benzoylpyridazine
DE10082008D2 (de)	2002-12-19	Ausbeulgerät
DE50003921D1 (de)	2003-11-06	Substituierte phenyluracile
DE60020365D1 (de)	2005-06-30	Säurekatalysierte umsetzungen
ATE440824T1 (de)	2009-09-15	Nitro-sulfobenzamide
ATA107599A (de)	2002-06-15	Heizwasserbereiter
DE50002156D1 (de)	2003-06-18	Azofarbstoffmischungen
DE10085167T1 (de)	2002-11-07	Gangumschalteinrichtung
NO20013625L (no)	2001-09-24	Megsinpromotor