DK0970084T3 - Pyrrolo[2,3-d]pyrimidiner og deres anvendelse som inhibitorer for tyrosinkinase - Google Patents

Pyrrolo[2,3-d]pyrimidiner og deres anvendelse som inhibitorer for tyrosinkinase

Info

Publication number
DK0970084T3
DK0970084T3 DK98913690T DK98913690T DK0970084T3 DK 0970084 T3 DK0970084 T3 DK 0970084T3 DK 98913690 T DK98913690 T DK 98913690T DK 98913690 T DK98913690 T DK 98913690T DK 0970084 T3 DK0970084 T3 DK 0970084T3
Authority
DK
Denmark
Prior art keywords
optionally substituted
group
phenyl
alkyl group
formula
Prior art date
Application number
DK98913690T
Other languages
English (en)
Inventor
David John Calderwood
David Norman Johnston
Paul Rafferty
Helen Louise Twigger
Rainer Munschauer
Lee Arnold
Original Assignee
Abbott Gmbh & Co Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Gmbh & Co Kg filed Critical Abbott Gmbh & Co Kg
Application granted granted Critical
Publication of DK0970084T3 publication Critical patent/DK0970084T3/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK98913690T 1997-03-19 1998-03-09 Pyrrolo[2,3-d]pyrimidiner og deres anvendelse som inhibitorer for tyrosinkinase DK0970084T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US4083697P 1997-03-19 1997-03-19
PCT/EP1998/001357 WO1998041525A1 (en) 1997-03-19 1998-03-09 Pyrrolo[2,3d]pyrimidines and their use as tyrosine kinase inhibitors

Publications (1)

Publication Number Publication Date
DK0970084T3 true DK0970084T3 (da) 2003-09-29

Family

ID=21913242

Family Applications (1)

Application Number Title Priority Date Filing Date
DK98913690T DK0970084T3 (da) 1997-03-19 1998-03-09 Pyrrolo[2,3-d]pyrimidiner og deres anvendelse som inhibitorer for tyrosinkinase

Country Status (23)

Country Link
US (1) US6001839A (da)
EP (1) EP0970084B1 (da)
JP (1) JP2001516353A (da)
KR (1) KR20000076426A (da)
CN (1) CN1134439C (da)
AT (1) ATE242245T1 (da)
AU (1) AU748884B2 (da)
BG (1) BG64282B1 (da)
BR (1) BR9808281A (da)
CA (1) CA2283961A1 (da)
DE (1) DE69815317T2 (da)
DK (1) DK0970084T3 (da)
ES (1) ES2202827T3 (da)
HU (1) HUP0001507A3 (da)
ID (1) ID24653A (da)
IL (1) IL131582A0 (da)
NO (1) NO313962B1 (da)
NZ (1) NZ337529A (da)
PL (1) PL335685A1 (da)
PT (1) PT970084E (da)
SK (1) SK125999A3 (da)
TR (1) TR199902301T2 (da)
WO (1) WO1998041525A1 (da)

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KR20000064601A (ko) * 1996-03-15 2000-11-06 한스 루돌프 하우스, 헨리테 브룬너, 베아트리체 귄터 신규의n-7-헤테로시클릴피롤로[2,3-d]피리딘및�그의용도

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DE69815317D1 (de) 2003-07-10
ES2202827T3 (es) 2004-04-01
SK125999A3 (en) 2000-05-16
PT970084E (pt) 2003-10-31
ATE242245T1 (de) 2003-06-15
EP0970084B1 (en) 2003-06-04
HUP0001507A2 (hu) 2000-10-28
WO1998041525A1 (en) 1998-09-24
DE69815317T2 (de) 2005-04-07
PL335685A1 (en) 2000-05-08
ID24653A (id) 2000-07-27
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NO994509D0 (no) 1999-09-17
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EP0970084A1 (en) 2000-01-12
CN1259950A (zh) 2000-07-12
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KR20000076426A (ko) 2000-12-26
AU748884B2 (en) 2002-06-13
HUP0001507A3 (en) 2002-01-28
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