DE60208364D1 - Chinolinderivate mit einer azolylgruppe und chinazolinderivate - Google Patents

Chinolinderivate mit einer azolylgruppe und chinazolinderivate

Info

Publication number
DE60208364D1
DE60208364D1 DE60208364T DE60208364T DE60208364D1 DE 60208364 D1 DE60208364 D1 DE 60208364D1 DE 60208364 T DE60208364 T DE 60208364T DE 60208364 T DE60208364 T DE 60208364T DE 60208364 D1 DE60208364 D1 DE 60208364D1
Authority
DE
Germany
Prior art keywords
derivatives
represent
chinazoline
chinoline
azolyl group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60208364T
Other languages
English (en)
Other versions
DE60208364T2 (de
Inventor
Kazuo Kubo
Teruyuki Sakai
Rika Nagao
Yasunari Fujiwara
Toshiyuki Isoe
Kazumasa Hasegawa
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Kirin Brewery Co Ltd
Original Assignee
Kirin Brewery Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=18980738&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DE60208364(D1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Kirin Brewery Co Ltd filed Critical Kirin Brewery Co Ltd
Publication of DE60208364D1 publication Critical patent/DE60208364D1/de
Application granted granted Critical
Publication of DE60208364T2 publication Critical patent/DE60208364T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
DE60208364T 2001-04-27 2002-04-26 Chinolinderivate mit einer azolylgruppe und chinazolinderivate Expired - Lifetime DE60208364T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2001132775 2001-04-27
JP2001132775 2001-04-27
PCT/JP2002/004279 WO2002088110A1 (fr) 2001-04-27 2002-04-26 Derives de quinoline ayant un groupe azolyle et derives de quinazoline

Publications (2)

Publication Number Publication Date
DE60208364D1 true DE60208364D1 (de) 2006-02-02
DE60208364T2 DE60208364T2 (de) 2006-09-28

Family

ID=18980738

Family Applications (2)

Application Number Title Priority Date Filing Date
DE60208364T Expired - Lifetime DE60208364T2 (de) 2001-04-27 2002-04-26 Chinolinderivate mit einer azolylgruppe und chinazolinderivate
DE60226912T Expired - Lifetime DE60226912D1 (de) 2001-04-27 2002-04-26 Chinolin- und Chianzolinderivate zur Behandlung von Tumoren

Family Applications After (1)

Application Number Title Priority Date Filing Date
DE60226912T Expired - Lifetime DE60226912D1 (de) 2001-04-27 2002-04-26 Chinolin- und Chianzolinderivate zur Behandlung von Tumoren

Country Status (25)

Country Link
US (2) US6821987B2 (de)
EP (2) EP1382604B1 (de)
JP (1) JP2010077131A (de)
KR (1) KR100879669B1 (de)
CN (1) CN1273466C (de)
AT (1) ATE396988T1 (de)
AU (1) AU2002255284B2 (de)
BE (1) BE2018C008I2 (de)
BR (1) BRPI0209216B8 (de)
CA (1) CA2445333C (de)
DE (2) DE60208364T2 (de)
DK (1) DK1382604T3 (de)
ES (1) ES2256466T3 (de)
FR (1) FR18C1006I2 (de)
HK (1) HK1070649A1 (de)
IL (1) IL158459A0 (de)
MX (1) MXPA03009662A (de)
NL (1) NL300927I9 (de)
NO (2) NO326325B1 (de)
NZ (1) NZ529046A (de)
PL (1) PL209822B1 (de)
RU (1) RU2283841C2 (de)
TW (1) TWI324154B (de)
WO (1) WO2002088110A1 (de)
ZA (1) ZA200307861B (de)

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US7718644B2 (en) * 2004-01-22 2010-05-18 The Trustees Of Columbia University In The City Of New York Anti-arrhythmic and heart failure drugs that target the leak in the ryanodine receptor (RyR2) and uses thereof
US20060293266A1 (en) * 2000-05-10 2006-12-28 The Trustees Of Columbia Phosphodiesterase 4D in the ryanodine receptor complex protects against heart failure
US6489125B1 (en) * 2000-05-10 2002-12-03 The Trustees Of Columbia University In The City Of New York Methods for identifying chemical compounds that inhibit dissociation of FKBP12.6 binding protein from type 2 ryanodine receptor
US20040048780A1 (en) * 2000-05-10 2004-03-11 The Trustees Of Columbia University In The City Of New York Method for treating and preventing cardiac arrhythmia
US20040229781A1 (en) * 2000-05-10 2004-11-18 Marks Andrew Robert Compounds and methods for treating and preventing exercise-induced cardiac arrhythmias
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BR0209216A (pt) 2004-07-06
HK1070649A1 (en) 2005-06-24
PL367105A1 (en) 2005-02-21
NO326325B1 (no) 2008-11-10
IL158459A0 (en) 2004-05-12
NZ529046A (en) 2005-10-28
RU2283841C2 (ru) 2006-09-20
CN1543459A (zh) 2004-11-03
WO2002088110A1 (fr) 2002-11-07
NO20034595L (no) 2003-12-19
CA2445333C (en) 2011-03-22
BE2018C008I2 (de) 2021-02-04
NL300927I9 (nl) 2019-02-05
ATE396988T1 (de) 2008-06-15
DK1382604T3 (da) 2006-04-18
US7211587B2 (en) 2007-05-01
ZA200307861B (en) 2004-10-08
DE60208364T2 (de) 2006-09-28
NL300927I1 (nl) 2018-12-04
EP1382604A4 (de) 2004-09-08
FR18C1006I1 (fr) 2018-03-16
FR18C1006I2 (fr) 2019-03-01
BRPI0209216B1 (pt) 2017-05-30
CN1273466C (zh) 2006-09-06
US6821987B2 (en) 2004-11-23
US20030087907A1 (en) 2003-05-08
BRPI0209216B8 (pt) 2021-05-25
US20040229876A1 (en) 2004-11-18
DE60226912D1 (de) 2008-07-10
TWI324154B (de) 2010-05-01
CA2445333A1 (en) 2002-11-07
EP1652847B1 (de) 2008-05-28
KR20040015143A (ko) 2004-02-18
JP2010077131A (ja) 2010-04-08
PL209822B1 (pl) 2011-10-31
KR100879669B1 (ko) 2009-01-21
EP1652847A3 (de) 2006-08-02
EP1652847A1 (de) 2006-05-03
ES2256466T3 (es) 2006-07-16
EP1382604B1 (de) 2005-12-28
AU2002255284B2 (en) 2007-10-04
RU2003134376A (ru) 2005-04-20
EP1382604A1 (de) 2004-01-21
MXPA03009662A (es) 2004-12-06
NO2018005I1 (no) 2018-02-05
NO20034595D0 (no) 2003-10-14

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