CY1111071T1 - Φαρμακευτικες ενωσεις που περιεχουν τα παραγωγα αζετιδινης, τα νεα παραγωγα αζετιδινης και η παρασκευη τους - Google Patents

Φαρμακευτικες ενωσεις που περιεχουν τα παραγωγα αζετιδινης, τα νεα παραγωγα αζετιδινης και η παρασκευη τους

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Publication number
CY1111071T1
CY1111071T1 CY20101101042T CY101101042T CY1111071T1 CY 1111071 T1 CY1111071 T1 CY 1111071T1 CY 20101101042 T CY20101101042 T CY 20101101042T CY 101101042 T CY101101042 T CY 101101042T CY 1111071 T1 CY1111071 T1 CY 1111071T1
Authority
CY
Cyprus
Prior art keywords
azetidin
producers
preparation
compounds containing
pharmaceutical compounds
Prior art date
Application number
CY20101101042T
Other languages
English (en)
Inventor
Daniel Achard
Hervé Bouchard
Jean Bouquerel
Bruno Filoche
Serge Grisoni
Augustin Hittinger
Michael Myers
Original Assignee
Aventis Pharma S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma S.A. filed Critical Aventis Pharma S.A.
Publication of CY1111071T1 publication Critical patent/CY1111071T1/el

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
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    • C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Abstract

Η παρούσα εφεύρεση αφορά τις φαρμακευτικές ενώσεις που περιέχουν ως βασικό δραστικό στοιχείο τουλάχιστον μία ένωση του τύπου όπου το R1 δηλώνει μια ρίζα -N(R4)R5, -N(R4)-CO-R5, -N(R4)-SΟ2R6 ή ένα από τα φαρμακευτικώς αποδεκτά άλατα αυτών, τα νέα παράγωγα του τύπου (I), τα φαρμακευτικώς αποδεκτά άλατα και την παρασκευή τους.
CY20101101042T 2000-03-03 2010-11-18 Φαρμακευτικες ενωσεις που περιεχουν τα παραγωγα αζετιδινης, τα νεα παραγωγα αζετιδινης και η παρασκευη τους CY1111071T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0002776A FR2805817B1 (fr) 2000-03-03 2000-03-03 Compositions pharmaceutiques contenant des derives d'azetidine, les nouveaux derives d'azetidine et leur preparation
EP01909939A EP1263722B1 (fr) 2000-03-03 2001-03-01 Compositions pharmaceutiques contenant des derives d'azetidine, les nouveaux derives d'azetidine et leur preparation

Publications (1)

Publication Number Publication Date
CY1111071T1 true CY1111071T1 (el) 2015-06-11

Family

ID=8847706

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CY20101101042T CY1111071T1 (el) 2000-03-03 2010-11-18 Φαρμακευτικες ενωσεις που περιεχουν τα παραγωγα αζετιδινης, τα νεα παραγωγα αζετιδινης και η παρασκευη τους

Country Status (36)

Country Link
EP (1) EP1263722B1 (el)
JP (1) JP4883867B2 (el)
KR (1) KR100819572B1 (el)
CN (1) CN100386314C (el)
AT (1) ATE478841T1 (el)
AU (1) AU780880B2 (el)
BG (1) BG66001B1 (el)
BR (1) BR0108893B1 (el)
CA (1) CA2400141C (el)
CY (1) CY1111071T1 (el)
CZ (1) CZ301254B6 (el)
DE (1) DE60142891D1 (el)
DK (1) DK1263722T3 (el)
DZ (1) DZ3312A1 (el)
EA (1) EA007109B1 (el)
EE (1) EE05103B1 (el)
ES (1) ES2351276T3 (el)
FR (1) FR2805817B1 (el)
HR (1) HRP20020712B1 (el)
HU (1) HUP0400636A3 (el)
IL (2) IL151321A0 (el)
MA (1) MA26880A1 (el)
ME (1) MEP9509A (el)
MX (1) MXPA02008349A (el)
NO (1) NO324524B1 (el)
NZ (1) NZ521077A (el)
OA (1) OA12222A (el)
PL (1) PL208021B1 (el)
PT (1) PT1263722E (el)
SI (1) SI1263722T1 (el)
SK (1) SK287445B6 (el)
TW (1) TWI304399B (el)
UA (1) UA73554C2 (el)
WO (1) WO2001064634A1 (el)
YU (1) YU66002A (el)
ZA (1) ZA200206912B (el)

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