BRPI0916890A2 - composto, composição farmacêutica, métodos para elicitar um efeito agonista, e um efeito antagonista de um receptor de gip, para tratar condições ou doeças, para tratar distúrbios, para tratar ou prevenir causas secundárias de diabete, e para estimular secreção de insulina em um indivíduo, e, uso de um composto - Google Patents

composto, composição farmacêutica, métodos para elicitar um efeito agonista, e um efeito antagonista de um receptor de gip, para tratar condições ou doeças, para tratar distúrbios, para tratar ou prevenir causas secundárias de diabete, e para estimular secreção de insulina em um indivíduo, e, uso de um composto

Info

Publication number: BRPI0916890A2
Authority: BR; Brazil
Prior art keywords: treating; compound; effect; eliciting; diabetes
Prior art date: 2008-08-07

Application number

BRPI0916890A

Other languages

English (en)

Inventor

Xin Dong Zheng

Original Assignee

Ipsen Pharma Sas

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2008-08-07

Filing date

2009-08-07

Publication date

2019-09-24

2009-08-07 Application filed by Ipsen Pharma Sas filed Critical Ipsen Pharma Sas

2019-09-24 Publication of BRPI0916890A2 publication Critical patent/BRPI0916890A2/pt

Links

150000001875 compounds Chemical class 0.000 title 2
208000037265 diseases, disorders, signs and symptoms Diseases 0.000 title 2
230000000694 effects Effects 0.000 title 2
239000000556 agonist Substances 0.000 title 1
239000005557 antagonist Substances 0.000 title 1
206010012601 diabetes mellitus Diseases 0.000 title 1
201000010099 disease Diseases 0.000 title 1
230000003914 insulin secretion Effects 0.000 title 1
239000008194 pharmaceutical composition Substances 0.000 title 1
230000004936 stimulating effect Effects 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/645—Secretins
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/62—Insulins
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/28—Insulins
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P13/12—Drugs for disorders of the urinary system of the kidneys
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
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- A61P3/00—Drugs for disorders of the metabolism
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A—HUMAN NECESSITIES
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- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
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- A—HUMAN NECESSITIES
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- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/605—Glucagons
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K19/00—Hybrid peptides, i.e. peptides covalently bound to nucleic acids, or non-covalently bound protein-protein complexes
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides

BRPI0916890A 2008-08-07 2009-08-07 composto, composição farmacêutica, métodos para elicitar um efeito agonista, e um efeito antagonista de um receptor de gip, para tratar condições ou doeças, para tratar distúrbios, para tratar ou prevenir causas secundárias de diabete, e para estimular secreção de insulina em um indivíduo, e, uso de um composto BRPI0916890A2 (pt)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US18819108P	2008-08-07	2008-08-07
US20062908P	2008-12-02	2008-12-02
PCT/US2009/004552 WO2010016940A2 (en)	2008-08-07	2009-08-07	Analogues of glucose-dependent insulinotropic polypeptide

Publications (1)

Publication Number	Publication Date
BRPI0916890A2 true BRPI0916890A2 (pt)	2019-09-24

Family

ID=41664129

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BRPI0916890A BRPI0916890A2 (pt)	2008-08-07	2009-08-07	composto, composição farmacêutica, métodos para elicitar um efeito agonista, e um efeito antagonista de um receptor de gip, para tratar condições ou doeças, para tratar distúrbios, para tratar ou prevenir causas secundárias de diabete, e para estimular secreção de insulina em um indivíduo, e, uso de um composto

Country Status (11)

Country	Link
US (2)	US9074014B2 (pt)
EP (2)	EP2328922A4 (pt)
JP (2)	JP2011530508A (pt)
KR (2)	KR20110043686A (pt)
CN (2)	CN104829706A (pt)
AU (1)	AU2009280017B2 (pt)
BR (1)	BRPI0916890A2 (pt)
CA (1)	CA2732949C (pt)
EA (1)	EA020019B1 (pt)
MX (1)	MX2011001031A (pt)
WO (1)	WO2010016940A2 (pt)

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KR20110043689A (ko)	2008-08-07	2011-04-27	입센 파마 에스.에이.에스	Ｎ-말단이 변형된 포도당 의존적인 인슐린 분비 자극성 폴리펩타이드(ｇｉｐ)의 유사체
MX2011001031A (es) *	2008-08-07	2011-04-26	Ipsen Pharma Sas	Analogos de polipeptidos insulinotropicos dependientes de glucosa.
MX2011001028A (es)	2008-08-07	2011-04-26	Ipsen Pharma Sas	Analogos truncados de polipeptidos de insulinotropicos dependientes de glucosa.
WO2010016938A2 (en)	2008-08-07	2010-02-11	Ipsen Pharma S.A.S.	Glucose-dependent insulinotropic polypeptide analogues

2009
- 2009-08-07 MX MX2011001031A patent/MX2011001031A/es active IP Right Grant
- 2009-08-07 CA CA2732949A patent/CA2732949C/en not_active Expired - Fee Related
- 2009-08-07 KR KR1020117003753A patent/KR20110043686A/ko active Application Filing
- 2009-08-07 CN CN201510177971.8A patent/CN104829706A/zh active Pending
- 2009-08-07 EP EP20090805293 patent/EP2328922A4/en not_active Withdrawn
- 2009-08-07 AU AU2009280017A patent/AU2009280017B2/en not_active Ceased
- 2009-08-07 EA EA201170304A patent/EA020019B1/ru not_active IP Right Cessation
- 2009-08-07 KR KR1020137020218A patent/KR101417873B1/ko not_active IP Right Cessation
- 2009-08-07 WO PCT/US2009/004552 patent/WO2010016940A2/en active Application Filing
- 2009-08-07 EP EP15186505.2A patent/EP2987805A3/en not_active Withdrawn
- 2009-08-07 JP JP2011522070A patent/JP2011530508A/ja active Pending
- 2009-08-07 US US13/057,760 patent/US9074014B2/en not_active Expired - Fee Related
- 2009-08-07 BR BRPI0916890A patent/BRPI0916890A2/pt not_active IP Right Cessation
- 2009-08-07 CN CN200980139514.2A patent/CN102171244B/zh not_active Expired - Fee Related
2013
- 2013-10-04 JP JP2013209264A patent/JP5865324B2/ja not_active Expired - Fee Related
2015
- 2015-05-20 US US14/717,186 patent/US20150252092A1/en not_active Abandoned

Also Published As

Publication number	Publication date
US20110136733A1 (en)	2011-06-09
JP2014028846A (ja)	2014-02-13
CA2732949A1 (en)	2010-02-11
EP2987805A3 (en)	2016-04-13
KR20110043686A (ko)	2011-04-27
CN104829706A (zh)	2015-08-12
US20150252092A1 (en)	2015-09-10
JP5865324B2 (ja)	2016-02-17
WO2010016940A3 (en)	2010-04-15
US9074014B2 (en)	2015-07-07
EA201170304A1 (ru)	2011-10-31
EP2328922A4 (en)	2013-01-02
JP2011530508A (ja)	2011-12-22
CA2732949C (en)	2016-12-20
CN102171244B (zh)	2015-05-13
AU2009280017B2 (en)	2013-01-10
WO2010016940A2 (en)	2010-02-11
AU2009280017A1 (en)	2010-02-11
KR20130093692A (ko)	2013-08-22
KR101417873B1 (ko)	2014-07-09
EA020019B1 (ru)	2014-08-29
MX2011001031A (es)	2011-04-26
CN102171244A (zh)	2011-08-31
EP2328922A2 (en)	2011-06-08
EP2987805A2 (en)	2016-02-24

Legal Events

Date	Code	Title	Description
2019-10-01	B08F	Application fees: application dismissed [chapter 8.6 patent gazette]
2020-01-21	B08K	Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]	Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2543 DE 01-10-2019 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.

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