BR112014028420A2 - regime de dosagem para um inibidor de quinase pi-3 - Google Patents

regime de dosagem para um inibidor de quinase pi-3

Info

Publication number
BR112014028420A2
BR112014028420A2 BR112014028420A BR112014028420A BR112014028420A2 BR 112014028420 A2 BR112014028420 A2 BR 112014028420A2 BR 112014028420 A BR112014028420 A BR 112014028420A BR 112014028420 A BR112014028420 A BR 112014028420A BR 112014028420 A2 BR112014028420 A2 BR 112014028420A2
Authority
BR
Brazil
Prior art keywords
kinase inhibitor
dosage regimen
regimen
dosage
kinase
Prior art date
Application number
BR112014028420A
Other languages
English (en)
Inventor
Massacesi Cristian
Hirawat Samit
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48626588&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR112014028420(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of BR112014028420A2 publication Critical patent/BR112014028420A2/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53771,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41961,2,4-Triazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
BR112014028420A 2012-05-16 2013-05-14 regime de dosagem para um inibidor de quinase pi-3 BR112014028420A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261647654P 2012-05-16 2012-05-16
PCT/US2013/040877 WO2013173283A1 (en) 2012-05-16 2013-05-14 Dosage regimen for a pi-3 kinase inhibitor

Publications (1)

Publication Number Publication Date
BR112014028420A2 true BR112014028420A2 (pt) 2017-09-19

Family

ID=48626588

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112014028420A BR112014028420A2 (pt) 2012-05-16 2013-05-14 regime de dosagem para um inibidor de quinase pi-3

Country Status (19)

Country Link
US (2) US10213432B2 (pt)
EP (1) EP2849756A1 (pt)
JP (2) JP6381523B2 (pt)
KR (1) KR20150009540A (pt)
CN (1) CN104349779A (pt)
AU (1) AU2013263043B2 (pt)
BR (1) BR112014028420A2 (pt)
CA (1) CA2872526A1 (pt)
CL (1) CL2014003101A1 (pt)
HK (1) HK1202435A1 (pt)
IL (1) IL235567B (pt)
MX (1) MX360892B (pt)
NZ (1) NZ700924A (pt)
PH (1) PH12014502547A1 (pt)
RU (1) RU2630975C2 (pt)
SG (2) SG11201406550QA (pt)
TN (1) TN2014000433A1 (pt)
WO (1) WO2013173283A1 (pt)
ZA (1) ZA201407406B (pt)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
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AU2012313888B2 (en) 2011-09-27 2016-03-31 Novartis Ag 3-pyrimidin-4-yl-oxazolidin-2-ones as inhibitors of mutant IDH
UY34632A (es) 2012-02-24 2013-05-31 Novartis Ag Compuestos de oxazolidin- 2- ona y usos de los mismos
US9296733B2 (en) 2012-11-12 2016-03-29 Novartis Ag Oxazolidin-2-one-pyrimidine derivative and use thereof for the treatment of conditions, diseases and disorders dependent upon PI3 kinases
AP2015008707A0 (en) 2013-03-14 2015-09-30 Novartis Ag 3-pyrimidin-4-yl-oxazolidin-2-ones as inhibitors of mutant idh
PL3076969T3 (pl) 2013-12-06 2022-01-17 Novartis Ag Schemat dawkowania selektywnego inhibitora 3-kinazy fosfatydynozytolu alfa-izoformy
WO2016109426A1 (en) * 2014-12-29 2016-07-07 Verastem, Inc. Oral dosing regimen of a dual mtor and pi3 inhibitor
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CA3002954A1 (en) * 2015-11-02 2017-05-11 Novartis Ag Dosage regimen for a phosphatidylinositol 3-kinase inhibitor
WO2018009895A1 (en) * 2016-07-08 2018-01-11 Autotelic Llc Methods for trabedersen dosing by auc

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Also Published As

Publication number Publication date
SG10201608469RA (en) 2016-11-29
ZA201407406B (en) 2015-11-25
RU2630975C2 (ru) 2017-09-15
SG11201406550QA (en) 2014-11-27
HK1202435A1 (en) 2015-10-02
IL235567B (en) 2019-08-29
US10213432B2 (en) 2019-02-26
NZ700924A (en) 2016-02-26
US20190134052A1 (en) 2019-05-09
CA2872526A1 (en) 2013-11-21
US20150141426A1 (en) 2015-05-21
TN2014000433A1 (en) 2016-03-30
AU2013263043B2 (en) 2016-06-16
EP2849756A1 (en) 2015-03-25
RU2014150860A (ru) 2016-07-10
CL2014003101A1 (es) 2015-02-27
MX2014013904A (es) 2015-01-16
CN104349779A (zh) 2015-02-11
IL235567A0 (en) 2015-01-29
WO2013173283A1 (en) 2013-11-21
JP2015517523A (ja) 2015-06-22
KR20150009540A (ko) 2015-01-26
PH12014502547A1 (en) 2015-01-21
AU2013263043A1 (en) 2014-10-30
MX360892B (es) 2018-11-20
JP2018108998A (ja) 2018-07-12
JP6381523B2 (ja) 2018-08-29

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Legal Events

Date Code Title Description
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
B06U Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
B11B Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements