AR221203A1 - Un compuesto intermediario sin actividad terapeutica que consiste en un derivado de la tieno(4,5)benzodiazepina,y un procedimiento para preparar una tieno-(1,5)benzodiazepina partiendo de dicho intermediario - Google Patents

Un compuesto intermediario sin actividad terapeutica que consiste en un derivado de la tieno(4,5)benzodiazepina,y un procedimiento para preparar una tieno-(1,5)benzodiazepina partiendo de dicho intermediario

Info

Publication number: AR221203A1
Authority: AR; Argentina
Prior art keywords: benzodiazepina; tieno; intermediary; derivative; preparing
Prior art date: 1974-11-26

Application number

AR261340A

Other languages

English (en)

Spanish (es)

Original Assignee

Lilly Industries Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1974-11-26

Filing date

1975-11-25

Publication date

1981-01-15

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10459213&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR221203(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1975-11-25 Application filed by Lilly Industries Ltd filed Critical Lilly Industries Ltd

1981-01-15 Application granted granted Critical

1981-01-15 Publication of AR221203A1 publication Critical patent/AR221203A1/es

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D333/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

AR261340A 1974-11-26 1975-11-25 Un compuesto intermediario sin actividad terapeutica que consiste en un derivado de la tieno(4,5)benzodiazepina,y un procedimiento para preparar una tieno-(1,5)benzodiazepina partiendo de dicho intermediario AR221203A1 (es)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB51240/74A GB1533235A (en)	1974-11-26	1974-11-26	Benzodiazepine derivatives

Publications (1)

Publication Number	Publication Date
AR221203A1 true AR221203A1 (es)	1981-01-15

Family

ID=10459213

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AR261340A AR221203A1 (es)	1974-11-26	1975-11-25	Un compuesto intermediario sin actividad terapeutica que consiste en un derivado de la tieno(4,5)benzodiazepina,y un procedimiento para preparar una tieno-(1,5)benzodiazepina partiendo de dicho intermediario

Country Status (30)

Country	Link
JP (1)	JPS6044314B2 (de)
AR (1)	AR221203A1 (de)
AT (1)	AT351547B (de)
AU (1)	AU506340B2 (de)
BE (1)	BE835932A (de)
BG (1)	BG29573A3 (de)
CA (1)	CA1075687A (de)
CH (2)	CH613455A5 (de)
CS (1)	CS236753B2 (de)
DD (1)	DD123343A5 (de)
DE (1)	DE2552403C2 (de)
DK (1)	DK146887C (de)
ES (1)	ES443011A1 (de)
FR (1)	FR2292479A1 (de)
GB (1)	GB1533235A (de)
HK (1)	HK58681A (de)
HU (1)	HU172493B (de)
IE (1)	IE42564B1 (de)
IL (1)	IL48502A (de)
KE (1)	KE3163A (de)
MY (1)	MY8200149A (de)
NL (1)	NL186088C (de)
NZ (1)	NZ179335A (de)
PH (2)	PH11669A (de)
PL (1)	PL100135B1 (de)
RO (1)	RO69912A (de)
SE (2)	SE421209B (de)
SU (2)	SU629879A3 (de)
YU (1)	YU298375A (de)
ZA (1)	ZA757344B (de)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IL62792A (en) *	1980-05-07	1985-02-28	Byk Gulden Lomberg Chem Fab	Acylated dihydrothienodiazepinone compounds,process for their preparation,and medicaments containing them
GB8819059D0 (en) *	1988-08-11	1988-09-14	Lilly Industries Ltd	Benzodiazepine compounds & their use as pharmaceuticals
GB9009229D0 (en)	1990-04-25	1990-06-20	Lilly Industries Ltd	Pharmaceutical compounds
NZ247703A (en) *	1992-05-29	1995-07-26	Lilly Industries Ltd	Thienobenzdiazepine derivatives and medicaments thereof
CA2234641A1 (en) *	1995-11-01	1997-05-09	Merck & Co., Inc.	Hexahydro-5-imino-1,4-heteroazepine derivatives as inhibitors of nitric oxide synthases
US6043358A (en)	1995-11-01	2000-03-28	Merck & Co., Inc.	Hexahydro-5-imino-1,4-heteroazepine derivatives as inhibitors of nitric oxide synthases
HUP0003718A3 (en)	1997-09-02	2002-11-28	Welfide Corp	Fused thiophene derivatives, use thereof and pharmaceutical compositions containing them
PL199016B1 (pl) *	2002-06-20	2008-08-29	Adamed Sp Z Oo	Sposób wytwarzania olanzapiny
SI21270A (sl)	2002-07-15	2004-02-29	Krka, Tovarna Zdravil, D.D., Novo Mesto	Kristalne oblike olanzapina in postopki za njihovo pripravo
DE10301923B3 (de) *	2003-01-17	2004-09-16	Krka Tovarna Zdravil, D.D.	Verfahren und Zwischenprodukte zur Herstellung von Olanzapin
AR047460A1 (es) *	2004-01-27	2006-01-18	Synthon Bv	Proceso para la fabricacion de acetato de 2-metil-4-(4-metil-1-piperazinil)-10h-tieno[2,3-b][1,5]benzodiazepina (acetato de olanzapina)
AR048272A1 (es)	2004-03-18	2006-04-12	Lek Pharmaceuticals	Sintesis de 2 metil - 4- (4- metil -1- piperazinil) - 10 h- tieno ( 2,3-b) (1,5) benzodiazepina y sus sales, metodos para su preparacion, composiciones farmaceuticas que la contienen y su uso en la fabricacion de medicamentos para el tratamiento de enfermedades mentales.
CN1980710B (zh) *	2004-06-30	2013-06-12	阿特西斯公司	作为5-羟色胺受体调节剂的取代的氮杂环庚烯衍生物
EP2292624A1 (de)	2009-07-20	2011-03-09	LEK Pharmaceuticals d.d.	Olanzapinreinigungsverfahren

1974
- 1974-11-25 SU SU742191705A patent/SU629879A3/ru active
- 1974-11-26 GB GB51240/74A patent/GB1533235A/en not_active Expired
1975
- 1975-11-20 DK DK524175A patent/DK146887C/da active
- 1975-11-20 IL IL48502A patent/IL48502A/xx unknown
- 1975-11-20 CA CA240,082A patent/CA1075687A/en not_active Expired
- 1975-11-21 PH PH17788A patent/PH11669A/en unknown
- 1975-11-21 AU AU86858/75A patent/AU506340B2/en not_active Expired
- 1975-11-22 DE DE2552403A patent/DE2552403C2/de not_active Expired
- 1975-11-24 CH CH604478A patent/CH613455A5/xx not_active IP Right Cessation
- 1975-11-24 CH CH1517275A patent/CH613454A5/xx not_active IP Right Cessation
- 1975-11-24 ZA ZA757344A patent/ZA757344B/xx unknown
- 1975-11-24 SE SE7513185A patent/SE421209B/xx not_active IP Right Cessation
- 1975-11-24 NZ NZ179335A patent/NZ179335A/xx unknown
- 1975-11-25 AR AR261340A patent/AR221203A1/es active
- 1975-11-25 YU YU02983/75A patent/YU298375A/xx unknown
- 1975-11-25 DD DD189666A patent/DD123343A5/xx unknown
- 1975-11-25 FR FR7535900A patent/FR2292479A1/fr active Granted
- 1975-11-25 JP JP50141080A patent/JPS6044314B2/ja not_active Expired
- 1975-11-25 IE IE2565/75A patent/IE42564B1/en unknown
- 1975-11-25 RO RO7584018A patent/RO69912A/ro unknown
- 1975-11-25 BE BE6045266A patent/BE835932A/xx not_active IP Right Cessation
- 1975-11-26 HU HU75LI00000284A patent/HU172493B/hu unknown
- 1975-11-26 ES ES443011A patent/ES443011A1/es not_active Expired
- 1975-11-26 BG BG7531601A patent/BG29573A3/xx unknown
- 1975-11-26 AT AT898275A patent/AT351547B/de not_active IP Right Cessation
- 1975-11-26 PL PL1975184991A patent/PL100135B1/pl unknown
- 1975-11-26 CS CS757991A patent/CS236753B2/cs unknown
- 1975-11-26 NL NLAANVRAGE7513833,A patent/NL186088C/xx not_active IP Right Cessation
1976
- 1976-10-07 SU SU762406250A patent/SU626702A3/ru active
1977
- 1977-02-22 PH PH19480A patent/PH24534A/en unknown
1978
- 1978-11-27 SE SE7812194A patent/SE429045B/sv not_active IP Right Cessation
1981
- 1981-09-24 KE KE3163A patent/KE3163A/xx unknown
- 1981-11-26 HK HK586/81A patent/HK58681A/xx unknown
1982
- 1982-12-30 MY MY149/82A patent/MY8200149A/xx unknown

Also Published As

Publication number	Publication date
CH613454A5 (en)	1979-09-28
IE42564L (en)	1976-05-26
AU506340B2 (en)	1979-12-20
NL7513833A (nl)	1976-05-31
PH11669A (en)	1978-05-19
IE42564B1 (en)	1980-09-10
SE7513185L (sv)	1976-05-27
PH24534A (en)	1990-08-03
JPS6044314B2 (ja)	1985-10-02
DD123343A5 (de)	1976-12-12
FR2292479A1 (fr)	1976-06-25
SE421209B (sv)	1981-12-07
ZA757344B (en)	1976-11-24
IL48502A0 (en)	1976-01-30
YU298375A (en)	1982-10-31
NZ179335A (en)	1978-11-13
KE3163A (en)	1981-10-16
SE7812194L (sv)	1978-11-27
DK146887B (da)	1984-01-30
DE2552403C2 (de)	1986-06-19
DK524175A (da)	1976-05-27
AT351547B (de)	1979-07-25
MY8200149A (en)	1982-12-31
CH613455A5 (en)	1979-09-28
HK58681A (en)	1981-12-04
SU626702A3 (ru)	1978-09-30
SE429045B (sv)	1983-08-08
CS236753B2 (en)	1985-05-15
DK146887C (da)	1984-07-09
NL186088B (nl)	1990-04-17
JPS5176296A (en)	1976-07-01
HU172493B (hu)	1978-09-28
NL186088C (nl)	1990-09-17
FR2292479B1 (de)	1978-07-28
PL100135B1 (pl)	1978-09-30
BE835932A (fr)	1976-05-25
RO69912A (ro)	1980-08-15
IL48502A (en)	1980-01-31
CA1075687A (en)	1980-04-15
ATA898275A (de)	1979-01-15
GB1533235A (en)	1978-11-22
ES443011A1 (es)	1977-07-01
AU8685875A (en)	1977-05-26
SU629879A3 (ru)	1978-10-25
DE2552403A1 (de)	1976-08-12
BG29573A3 (en)	1980-12-12

Publication	Publication Date	Title
AR213097A1 (es)	1978-12-15	Procedimiento para preparar derivados de la 1,4-dihidropirina
MX3620E (es)	1981-04-02	Procedimiento para preparar 2(4(tetrahidro-2-furoil)-piperazino)-4-amino-6,7-dimetoxiquinazolina
AR208425A1 (es)	1976-12-27	Procedimiento para la preparacion de una suspension acuosa conteniendo un peroxido organico solido a una temperatura de aproximadamente 20 c
AR212176A1 (es)	1978-05-31	Procedimiento para preparar derivados de(4-hidroxipirrolidin-2-on-il)acilamida
IT1069986B (it)	1985-03-25	Procedimento perfezionato adiabatico per la monoitrazione di composti aromatici
AR221203A1 (es)	1981-01-15	Un compuesto intermediario sin actividad terapeutica que consiste en un derivado de la tieno(4,5)benzodiazepina,y un procedimiento para preparar una tieno-(1,5)benzodiazepina partiendo de dicho intermediario
AR210349A1 (es)	1977-07-29	Procedimiento para la preparacion de 6-coloro-2(piperacinil)piracina
AR218851A1 (es)	1980-07-15	Procedimiento para la preparacion de monoesteres de 17 alpha o 16 alpha o 21-retinoato de 11 beta,17 alpha,21-trihidroxi-3,20-diceto-4-pregnanos y-1,4-pregnatrienos
MX3636E (es)	1981-04-13	Procedimiento para la preparacion de propargil-2-fenilamino-imidazolinas-(2)
MX3932E (es)	1981-10-02	Procedimiento para la preparacion de 4,5-diaril-2-(tiosustituido) imidazoles
RO76721A (ro)	1982-10-11	Procedeu pentru prepararea 3.12.-hidroxi-4-fenil-cicloalcanonei
AR207182A1 (es)	1976-09-15	Procedimiento para preparar derivados de la l-3-(3,4-dihidroxi-fenil)-2-metil-alanina
MX3878E (es)	1981-08-26	Procedimiento para preparar derivados de 6-aril-pirrolo (1,2-a) imidazola
SE433210B (sv)	1984-05-14	Forfarande for framstellning av ny cyklohexylfenylderivat
GR60368B (en)	1978-05-22	Means against anti-histomoniasis(blackhead disease of birds)
MX144201A (es)	1981-09-10	Procedimiento mejorado para la preparacion de ciclohexanodionas (1,3)
AR221031A1 (es)	1980-12-30	Procedimiento para preparar un compuesto de benzoil-fenilindina y benzoil-fenilnaftaleno
RO72564A (ro)	1982-02-26	Procedeu pentru prepararea unor derivati ai triaminoandrostanului
MX146606A (es)	1982-07-15	Procedimiento mejorado para preparar la cubierta de una microcapsula
BE848072A (fr)	1977-03-01	Stethoscope nucleaire,
AR210162A1 (es)	1977-06-30	Procedimiento para la preparacion de un 2-alquilindano
NL7601500A (nl)	1976-08-17	Werkwijze ter bereiding van halogeenacyl-en thiohalogeenacylarylgesubstitueerde oxazolidi- nen en thiazolidinen-herbicide tegengiffen als- mede preparaten die deze verbindingen bevatten.
SU605537A3 (ru)	1978-04-30	Тормозной цилиндр
RO74536A (ro)	1980-11-30	Procedeu pentru prepararea 2,3-dicloranisolului
AR210480A1 (es)	1977-08-15	Procedimiento para preparar derivados 1,5-disubstituidos de 2-aminiomidazol