UA81641C2 - Process for the preparation of zaleplon - Google Patents

Process for the preparation of zaleplon

Info

Publication number: UA81641C2
Authority: UA; Ukraine
Prior art keywords: zaleplon; preparation; alkoxyalcohol; ethy1; carbonitrile
Prior art date: 2002-10-25

Application number

UAA200504945A

Other languages

English (en)

Inventor

Станислав Радл

Original Assignee

ЗЕНТИВА, а.с.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-10-25

Filing date

2003-10-21

Publication date

2008-01-25

2003-10-21 Application filed by ЗЕНТИВА, а.с. filed Critical ЗЕНТИВА, а.с.

2008-01-25 Publication of UA81641C2 publication Critical patent/UA81641C2/ru

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

UAA200504945A 2002-10-25 2003-10-21 Process for the preparation of zaleplon UA81641C2 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
CZ20023575A CZ293015B6 (cs)	2002-10-25	2002-10-25	Způsob výroby N-ethyl-N-[3-(3-methyl-pyrazolo[1,5-a]pyrimidin-7-yl)-fenyl]-acetamidu (zaleplonu)
PCT/CZ2003/000057 WO2004037824A1 (en)	2002-10-25	2003-10-21	Process for the preparation of zaleplon

Publications (1)

Publication Number	Publication Date
UA81641C2 true UA81641C2 (en)	2008-01-25

Family

ID=29751097

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
UAA200504945A UA81641C2 (en)	2002-10-25	2003-10-21	Process for the preparation of zaleplon

Country Status (12)

Country	Link
US (1)	US20050245742A1 (ru)
EP (1)	EP1554279B1 (ru)
JP (1)	JP2006507278A (ru)
AU (1)	AU2003273390A1 (ru)
CA (1)	CA2503152A1 (ru)
CZ (1)	CZ293015B6 (ru)
DE (1)	DE60317817D1 (ru)
EA (1)	EA007505B1 (ru)
PL (1)	PL374911A1 (ru)
SK (1)	SK50402005A3 (ru)
UA (1)	UA81641C2 (ru)
WO (1)	WO2004037824A1 (ru)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US20050032818A1 (en) *	2001-06-12	2005-02-10	Entire Interest	N-[3-(3-cyanopyrazolo[1,5-a]pyrimidin-5-yl)phenyl]-N-ethylacetamide and crystalline forms of zaleplon
US6852858B2 (en) *	2001-08-01	2005-02-08	Biogal Gyogyszergyar Rt.	Process for purifying N-[3-(3-cyanopyrazolo[1,5-a]pyrimidin-7-yl)phenyl]-N-ethylacetamide (zaleplon) and crystalline forms of zaleplon accessible with the process

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5356897A (en) *	1991-09-09	1994-10-18	Fujisawa Pharmaceutical Co., Ltd.	3-(heteroaryl)-pyrazololi[1,5-a]pyrimidines
AU734009B2 (en) *	1997-05-30	2001-05-31	Merck & Co., Inc.	Novel angiogenesis inhibitors
AR029780A1 (es) *	2000-12-13	2003-07-16	Gador Sa	Procedimiento mejorado para la obtencion de n-[3(3-ciano-pirazolo[1,5-a]pirimidin-7-il)fenil]-n-etil-acetamida
US6852858B2 (en) *	2001-08-01	2005-02-08	Biogal Gyogyszergyar Rt.	Process for purifying N-[3-(3-cyanopyrazolo[1,5-a]pyrimidin-7-yl)phenyl]-N-ethylacetamide (zaleplon) and crystalline forms of zaleplon accessible with the process
ES2223311T1 (es) *	2001-06-12	2005-03-01	Biogal Gyogyszergyar Rt.	Procedimiento para la preparacion de n-(3-(3-cianopirazol(1,5-a)pirimidin-7-il)fenil)-n-etilacetamida (zaleplon).

2002
- 2002-10-25 CZ CZ20023575A patent/CZ293015B6/cs not_active IP Right Cessation
2003
- 2003-10-21 AU AU2003273390A patent/AU2003273390A1/en not_active Abandoned
- 2003-10-21 JP JP2004545691A patent/JP2006507278A/ja active Pending
- 2003-10-21 UA UAA200504945A patent/UA81641C2/ru unknown
- 2003-10-21 CA CA002503152A patent/CA2503152A1/en not_active Abandoned
- 2003-10-21 PL PL03374911A patent/PL374911A1/xx not_active Application Discontinuation
- 2003-10-21 DE DE60317817T patent/DE60317817D1/de not_active Expired - Lifetime
- 2003-10-21 EP EP03755542A patent/EP1554279B1/en not_active Expired - Lifetime
- 2003-10-21 SK SK5040-2005A patent/SK50402005A3/sk not_active Application Discontinuation
- 2003-10-21 WO PCT/CZ2003/000057 patent/WO2004037824A1/en active IP Right Grant
- 2003-10-21 EA EA200500702A patent/EA007505B1/ru not_active IP Right Cessation
2005
- 2005-04-22 US US11/111,818 patent/US20050245742A1/en not_active Abandoned

Also Published As

Publication number	Publication date
CZ20023575A3 (cs)	2004-01-14
SK50402005A3 (sk)	2005-08-04
EP1554279A1 (en)	2005-07-20
AU2003273390A1 (en)	2004-05-13
PL374911A1 (en)	2005-11-14
DE60317817D1 (de)	2008-01-10
EP1554279B1 (en)	2007-11-28
EA200500702A1 (ru)	2005-10-27
US20050245742A1 (en)	2005-11-03
EA007505B1 (ru)	2006-10-27
CZ293015B6 (cs)	2004-01-14
CA2503152A1 (en)	2004-05-06
JP2006507278A (ja)	2006-03-02
WO2004037824A1 (en)	2004-05-06

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