SG10201700889PA - P2x7 modulators - Google Patents

P2x7 modulators

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Publication number
SG10201700889PA
SG10201700889PA SG10201700889PA SG10201700889PA SG10201700889PA SG 10201700889P A SG10201700889P A SG 10201700889PA SG 10201700889P A SG10201700889P A SG 10201700889PA SG 10201700889P A SG10201700889P A SG 10201700889PA SG 10201700889P A SG10201700889P A SG 10201700889PA
Authority
SG
Singapore
Prior art keywords
modulators
Prior art date
Application number
SG10201700889PA
Other languages
English (en)
Inventor
Vaca Manuel Jesus Alcazar
Brett D Allison
Gil Jose Ignacio Andres
Christa C Chrovian
Heather R Coate
Angelis Meri De
Xiaohu Deng
Curt A Dvorak
Christine F Gelin
Michael A Letavic
Jimmy T Liang
Neelakandha S Mani
Jason C Rech
Brad M Savall
Akinola Soyode-Johnson
Brice M Stenne
Devin M Swanson
Jessica L Wall
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of SG10201700889PA publication Critical patent/SG10201700889PA/en

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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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    • A61K31/4965—Non-condensed pyrazines
    • A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
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    • C07D—HETEROCYCLIC COMPOUNDS
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SG10201700889PA 2013-03-14 2014-03-14 P2x7 modulators SG10201700889PA (en)

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US201361786260P 2013-03-14 2013-03-14

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SG10201700889PA true SG10201700889PA (en) 2017-03-30

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JP (1) JP6293861B2 (ar)
KR (4) KR20230049754A (ar)
CN (2) CN105209464B (ar)
AR (2) AR095530A1 (ar)
AU (5) AU2014239291B2 (ar)
BR (1) BR112015023142B1 (ar)
CA (1) CA2906085C (ar)
CL (3) CL2015002655A1 (ar)
CY (1) CY1119110T1 (ar)
DK (2) DK3239151T3 (ar)
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HR (1) HRP20171168T4 (ar)
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PL (1) PL2970267T6 (ar)
PT (2) PT3239151T (ar)
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SI (1) SI2970267T1 (ar)
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UA (1) UA116467C2 (ar)
UY (3) UY39887A (ar)
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JO3509B1 (ar) 2013-03-14 2020-07-05 Janssen Pharmaceutica Nv معدلات p2x7
JO3773B1 (ar) 2013-03-14 2021-01-31 Janssen Pharmaceutica Nv معدلات p2x7
TW201522307A (zh) 2013-03-14 2015-06-16 百靈佳殷格翰國際股份有限公司 經取代２－氮雜－雙環［２．２．１］庚烷－３－羧酸（苄基－氰基－甲基）－醯胺組織蛋白酶ｃ抑制劑
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WO2015172196A1 (en) * 2014-05-13 2015-11-19 Monash University Heterocyclic compounds and use of same
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ES2757052T3 (es) * 2015-07-31 2020-04-28 Merck Patent Gmbh Derivados heterocíclicos bicíclicos
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