SE8304408L - Desoxiuridinderivat, forfaranden for deras framstellning och deras anvendning som lekemedel - Google Patents

Desoxiuridinderivat, forfaranden for deras framstellning och deras anvendning som lekemedel

Info

Publication number
SE8304408L
SE8304408L SE8304408A SE8304408A SE8304408L SE 8304408 L SE8304408 L SE 8304408L SE 8304408 A SE8304408 A SE 8304408A SE 8304408 A SE8304408 A SE 8304408A SE 8304408 L SE8304408 L SE 8304408L
Authority
SE
Sweden
Prior art keywords
derivatives
desoxiuride
procedures
preparation
medicinal product
Prior art date
Application number
SE8304408A
Other languages
English (en)
Swedish (sv)
Other versions
SE8304408D0 (sv
Inventor
H Griengl
E Wanek
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ag filed Critical Sandoz Ag
Publication of SE8304408D0 publication Critical patent/SE8304408D0/xx
Publication of SE8304408L publication Critical patent/SE8304408L/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06Pyrimidine radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/20Antivirals for DNA viruses
    • A61P31/22Antivirals for DNA viruses for herpes viruses

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Virology (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biotechnology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
SE8304408A 1982-08-17 1983-08-15 Desoxiuridinderivat, forfaranden for deras framstellning och deras anvendning som lekemedel SE8304408L (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH492282 1982-08-17

Publications (2)

Publication Number Publication Date
SE8304408D0 SE8304408D0 (sv) 1983-08-15
SE8304408L true SE8304408L (sv) 1984-02-18

Family

ID=4284858

Family Applications (1)

Application Number Title Priority Date Filing Date
SE8304408A SE8304408L (sv) 1982-08-17 1983-08-15 Desoxiuridinderivat, forfaranden for deras framstellning och deras anvendning som lekemedel

Country Status (16)

Country Link
JP (1) JPS5953499A (da)
AU (1) AU1800483A (da)
BE (1) BE897516A (da)
DE (1) DE3390162T1 (da)
DK (1) DK372283A (da)
ES (1) ES8604943A1 (da)
FI (1) FI832884A (da)
FR (1) FR2531962B1 (da)
GB (1) GB2125401B (da)
IL (1) IL69497A0 (da)
IT (1) IT1169765B (da)
NL (1) NL8302859A (da)
PT (1) PT77209B (da)
SE (1) SE8304408L (da)
WO (1) WO1984000759A1 (da)
ZA (1) ZA836072B (da)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4526988A (en) * 1983-03-10 1985-07-02 Eli Lilly And Company Difluoro antivirals and intermediate therefor
CA1295998C (en) * 1985-07-29 1992-02-18 Sai P. Sunkara Nucleosides and their use as antineoplastic agents
SE8605503D0 (sv) * 1986-12-19 1986-12-19 Astra Laekemedel Ab Novel medicinal use
US5215971A (en) * 1986-12-19 1993-06-01 Medivir Ab Antiviral pharmaceutical composition comprising 5-substituted pyrimidine nucleosides
US5215970A (en) * 1987-04-16 1993-06-01 Medivir Ab Nucleosides and nucleotide analogues, pharmaceutical composition and processes for the preparation of the compounds
US4863927A (en) * 1987-05-11 1989-09-05 Merck & Co., Inc. 1-(2-hydroxymethyl)cycloalkylmethyl)-5-substituted uracils
US5401838A (en) * 1992-06-22 1995-03-28 Eli Lilly And Company Stereoselective fusion glycosylation process for preparing 2'-deoxy-2',2'-difluoronucleosides and 2'-deoxy-2'-fluoronucleosides
MX9303708A (es) * 1992-06-22 1994-05-31 Lilly Co Eli Proceso de glucosilacion anionica estereoselectiva para preparar 2'-desoxifluoro-beta nucleosidos.
US5821357A (en) * 1992-06-22 1998-10-13 Eli Lilly And Company Stereoselective glycosylation process for preparing 2'-deoxy-2',2'-difluoropurine and triazole nucleosides
US5426183A (en) * 1992-06-22 1995-06-20 Eli Lilly And Company Catalytic stereoselective glycosylation process for preparing 2'-deoxy-2',2'-difluoronucleosides and 2'-deoxy-2'-fluoronucleosides
US5594124A (en) * 1992-06-22 1997-01-14 Eli Lilly And Company Stereoselective glycosylation process for preparing 2'-Deoxy-2',2'-difluoropyrimidine nucleosides and 2'-deoxy-2'-fluoropyrimidine nucleosides and intermediates thereof
US5606048A (en) * 1992-06-22 1997-02-25 Eli Lilly And Company Stereoselective glycosylation process for preparing 2'-Deoxy-2', 2'-difluoronucleosides and 2'-deoxy-2'-fluoronucleosides
US5371210A (en) * 1992-06-22 1994-12-06 Eli Lilly And Company Stereoselective fusion glycosylation process for preparing 2'-deoxy-2',2'-difluoronucleosides and 2'-deoxy-2'-fluoronucleosides
US5424416A (en) * 1993-08-25 1995-06-13 Eli Lilly And Company Process for preparation of 2-deoxy-2,2-difluoro-D-ribofuranosyl-3,5-hydroxy protected-1-alkyl and aryl sulfonates and their use in preparation of 2',2'-difluoro-2'-deoxy nucleosides
SE9701219D0 (sv) * 1997-04-04 1997-04-04 Astra Pharma Prod New compounds
WO2003018030A1 (en) * 2001-08-24 2003-03-06 Koronis Pharmaceuticals, Inc. Mutagenic nucleoside analogs for the treatment of viral disease

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3709874A (en) * 1970-03-19 1973-01-09 Syntex Corp 1-beta-d-arabinofuranosyl cytosine derivatives and methods of preparing
GB1601020A (en) * 1978-04-24 1981-10-21 Stichting Grega Vzw 2'-deoxy-5 (2-halogenovinyl)-uridines
GB2060604B (en) * 1979-10-03 1983-11-23 Univ Birmingham And Stichting E15-(2-halogenovinyl)-2'-deoxycytidines
DE3002197A1 (de) * 1980-01-22 1981-07-23 Robugen Gmbh Pharmazeutische Fabrik Esslingen A.N., 7300 Esslingen 5-alkylsubstituierte pyrimidin-nukleoside, verfahren zu deren herstellung und daraus hergestellte virostatische und cytostatische mittel
DE3010399A1 (de) * 1980-03-18 1981-09-24 Kailash Kumar Dr. 2359 Lentföhrden Gauri Verwendung von 5-haloalkyl-pyrimidin-nukleosiden als virostatika und cytostatika
HU183567B (en) * 1981-09-07 1984-05-28 Mta Koezponti Kemiai Kutato In Process for preparing /e/-5-/2-bromo-vinyl/-uridine and derivatives thereof

Also Published As

Publication number Publication date
NL8302859A (nl) 1984-03-16
GB2125401A (en) 1984-03-07
IT1169765B (it) 1987-06-03
ES8604943A1 (es) 1986-02-16
GB2125401B (en) 1985-10-16
PT77209A (en) 1983-09-01
ES524997A0 (es) 1986-02-16
BE897516A (fr) 1984-02-13
ZA836072B (en) 1985-03-27
WO1984000759A1 (en) 1984-03-01
FI832884A (fi) 1984-02-18
DE3390162T1 (de) 1985-02-21
SE8304408D0 (sv) 1983-08-15
IT8322565A0 (it) 1983-08-16
AU1800483A (en) 1984-02-23
DK372283D0 (da) 1983-08-15
FR2531962A1 (fr) 1984-02-24
GB8321880D0 (en) 1983-09-14
FR2531962B1 (fr) 1986-11-14
DK372283A (da) 1984-02-18
IL69497A0 (en) 1983-11-30
JPS5953499A (ja) 1984-03-28
PT77209B (en) 1986-03-18
FI832884A0 (fi) 1983-08-10

Similar Documents

Publication Publication Date Title
SE8304408L (sv) Desoxiuridinderivat, forfaranden for deras framstellning och deras anvendning som lekemedel
PT100199A (pt) Combinacao antiviral de nucleosidos e processo para a sua preparacao
FI963424A0 (fi) Menetelmä terapeuttisesti aktiivisten tiofeenisulfonamidien valmistamiseksi
GR3007202T3 (da)
PT83872A (de) Arzneimittel
SE8804629D0 (sv) New therapeutically active compounds
SE8000435L (sv) N-bensylimidazoler med selektivt inhiberande verkan pa tromboxansyntetasenzymet jemte farmaceutiska beredningar innehallande sadana n-bensylimidazoler och sett for deras framstellning
IT8319857A0 (it) Agenti antiflogistici/antipiretici/analgesici contenenti derivati di teobromina o teofillina come ingrediente attivo.
NL184833C (nl) 2-gesubstitueerd aminopyrimidinederivaten en farmaceutische preparaten die ze bevatten.
DK0479093T3 (da) Oligosaccharidderivater og deres anvendelse som lægemidler
ATE70445T1 (de) Pharmazeutische praeparate.
ES499363A0 (es) Procedimiento para la obtencion de derivados de fenilpipera-cina de 1,3,4-oxadiazolilfenoles
DE10299023I1 (de) Antineoplastisch wirkender und den Antineoplastischen effekt Verstaerkender Wirkstoff
IE810123L (en) N-(tetrazol-5-yl) retinamides
ES2032476T3 (es) Un procedimiento para preparar nuevos derivados de 2-anilinotiazolina.
PT89582B (pt) Processo para a preparacao de antibioticos beta-lactamicos uteis como medicamentos
DE3579140D1 (de) Arzneimittel mit einem 6-substituierten adenosin als aktives bestandteil.
MX9302929A (es) Derivados de tetrahidro y perhidroisoquinolina y medios terapeuticos que los contienen.
IT8220537A0 (it) Derivati della cefuroxima attivi per via orale procedimenti per laloro preparazione e relative composizioni farmaceutuche.
ES1032723Y (es) Bloqueador del embolo para jeringuilla desechable.
SE8503513D0 (sv) Farmaceutiska och kosmetiska kompositioner, vilka som verksam bestandsdel innehaller acetyl-10-triacetoxi-1,8,9-antracen
IT1166217B (it) Composizione farmaceutica per la terapia delle sterilita' maschile
ES2054453T3 (es) Excipiente para principio activo terapeutico de uso externo y preparado antiseptico que comprende dicho excipiente.
AR227989A1 (es) Procedimiento para la elaboracion del nuevo 1-(2,3-dihidro-1,4-benzodioxin-2s-il)-5-(2,3-dihidro-1,4 benzodioxin-2r--il)-3-azapetan-1r,5s-diol"
ITMI920232A1 (it) Procedimento per la preparazione di derivati del glicerolo otticamente attivi.

Legal Events

Date Code Title Description
NAV Patent application has lapsed

Ref document number: 8304408-1

Effective date: 19871225