PH9329A - 6-phenyl-1-substituted-4h-s-triazolo(4,3-a)-benzodiazepines - Google Patents

6-phenyl-1-substituted-4h-s-triazolo(4,3-a)-benzodiazepines

Info

Publication number
PH9329A
PH9329A PH11194*UA PH11194A PH9329A PH 9329 A PH9329 A PH 9329A PH 11194 A PH11194 A PH 11194A PH 9329 A PH9329 A PH 9329A
Authority
PH
Philippines
Prior art keywords
benzodiazepines
triazolo
phenyl
substituted
Prior art date
Application number
PH11194*UA
Other languages
English (en)
Inventor
J Hester
Original Assignee
J Hester
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27123060&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PH9329(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by J Hester filed Critical J Hester
Priority to PH13274*UA priority Critical patent/PH9316A/en
Publication of PH9329A publication Critical patent/PH9329A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/20—Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Fodder In General (AREA)
PH11194*UA 1969-03-17 1970-02-27 6-phenyl-1-substituted-4h-s-triazolo(4,3-a)-benzodiazepines PH9329A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
PH13274*UA PH9316A (en) 1969-03-17 1972-02-16 2-acylhydrazino benzodiazepines

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US80793369A 1969-03-17 1969-03-17
US04/872,394 US3987052A (en) 1969-03-17 1969-10-29 6-Phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines

Publications (1)

Publication Number Publication Date
PH9329A true PH9329A (en) 1975-09-23

Family

ID=27123060

Family Applications (1)

Application Number Title Priority Date Filing Date
PH11194*UA PH9329A (en) 1969-03-17 1970-02-27 6-phenyl-1-substituted-4h-s-triazolo(4,3-a)-benzodiazepines

Country Status (18)

Country Link
US (1) US3987052A (de)
JP (1) JPS4940239B1 (de)
AU (2) AU490626B2 (de)
BE (1) BE747493A (de)
BR (1) BR7017488D0 (de)
CH (1) CH535788A (de)
DE (1) DE2012190C3 (de)
ES (1) ES376689A1 (de)
FR (1) FR2034999A1 (de)
GB (1) GB1291631A (de)
HK (1) HK61677A (de)
IL (1) IL33859A (de)
NL (2) NL172510C (de)
OA (1) OA03446A (de)
PH (1) PH9329A (de)
PL (1) PL80541B1 (de)
SE (1) SE387641B (de)
YU (1) YU35139B (de)

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YU34997B (en) * 1970-03-27 1980-06-30 Hiroyuki Tawada Process for preparing benzodiazepine derivatives
DE2156472A1 (de) * 1970-11-23 1972-05-31 Ciba-Geigy Ag, Basel (Schweiz) Verfahren zur Herstellung von neuen Diazepinderivaten
CH544764A (de) * 1971-01-21 1974-01-15 Ciba Geigy Ag Verfahren zur Herstellung von neuen Triazolo-benzodiazepinderivaten
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US3759943A (en) * 1971-04-28 1973-09-18 Upjohn Co Amido and amino triazolo benzodiazepines
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US3709899A (en) 1971-04-28 1973-01-09 Upjohn Co 6-phenyl-4h-s-triazolo(4,3-a)(1,4)benzodiazepines and their production
GB1323277A (en) * 1971-05-10 1973-07-11 Upjohn Co Triazolobenzodiazepines
US3734922A (en) * 1971-05-11 1973-05-22 Upjohn Co Certain 4h-s-triazolo(4,3-a)(1,4)benzodiazepines
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BE787251A (fr) * 1971-08-04 1973-02-05 Upjohn Co Nouvelles benzodiazepines et leur preparation
US3870793A (en) * 1971-08-09 1975-03-11 Upjohn Co Animal feed and process
GB1373300A (en) * 1971-09-08 1974-11-06 Upjohn Co Triazolobenzodiazepines and the manufacture thereof
US3767661A (en) * 1971-09-13 1973-10-23 Upjohn Co 4h-s-triazolo(4,3-a)(1,4)benzodiazepines
GB1381158A (en) * 1971-09-13 1975-01-22 Upjohn Co Benzodiazepines and the manufacture thereof
US3714178A (en) * 1971-09-30 1973-01-30 Upjohn Co 6,7-DIHYDRO-7-ALKYL-5H-1,2,4-TRIAZOLO[4,3-d][1,4]BENZODIAZEPINES AND THEIR PRODUCTION
BE790838A (fr) * 1971-11-02 1973-04-30 Upjohn Co Nouvelles 1-aminophenyl-6-phenyl-s-triazolo (4,3-a) (1,4)- benzodiazepines, leur procede de preparation et medicament les contenant
FI53821C (fi) * 1971-11-15 1978-08-10 Ciba Geigy Ag Foerfarande foer framstaellning av farmakologiskt vaerdefull 6-fenyl-8-klor-4h-s-triazolo(4 3-a)(1 4)bensodiazepin-1-metanol
FR2128552A2 (en) * 1972-03-02 1972-10-20 Upjohn Co S-triazolo (4,3-a) (1,4) benzodiazepines - as anxiolytic agents, muscle relaxants
CH572056A5 (de) * 1972-11-28 1976-01-30 Ciba Geigy Ag
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US4431589A (en) * 1980-12-11 1984-02-14 Lilly House Benzodiazepine compounds and their use as pharmaceuticals
US4455307A (en) * 1982-01-04 1984-06-19 The Upjohn Company Antihypertensive use of triazolobenzodiazepines
US4375473A (en) * 1982-01-04 1983-03-01 The Upjohn Company Method
US4508726A (en) * 1982-09-16 1985-04-02 The Upjohn Company Treatment of panic disorders with alprazolam
DE3332830A1 (de) * 1982-09-16 1984-03-22 The Upjohn Co., 49001 Kalamazoo, Mich. Verwendung von benzodiazepinen zur bekaempfung oder bei der behandlung von panikzustaenden
US4481208A (en) * 1983-06-06 1984-11-06 The Upjohn Company Treatment of panic disorders with estazolam
US4514407A (en) * 1983-03-17 1985-04-30 The Upjohn Company 1-Ethanamine-triazolo-benzodiazepines as diuretics
US4689413A (en) * 1983-03-17 1987-08-25 The Upjohn Company Triazolo-benzodiazepine-1-ethanamines as diuretics
US4474699A (en) * 1983-05-25 1984-10-02 The Upjohn Company Preparing 1-aminomethyl-6-substituted-4H-s-triazolo[4,3-a][1,4]benzodiazepines in improved procedures
US4588721A (en) * 1983-09-12 1986-05-13 The Upjohn Company Treatment of negative symptoms of schizophrenia
US4547499A (en) * 1984-05-10 1985-10-15 The Upjohn Company 2,4-Dihydro-2(omega-aminoalkyl)-1H-[1,2,4]triazolo[3,4-c]benzoxazin-1-one anti-allergy drug compounds, compositions and use
US4634703A (en) * 1985-10-25 1987-01-06 Bristol-Myers Company Method for alleviation of panic disorders
US4959361A (en) * 1987-12-18 1990-09-25 Hoffmann-La Roche Inc. Triazolo(4,3-A)(1,4)benzodiazepines and thieno (3,2-F)(1,2,4)triazolo(4,3-A)(1,4)diazepine compounds which have useful activity as platelet activating factor (PAF) antagonists
US5334592A (en) * 1988-04-27 1994-08-02 Schering Corporation Certain PAF antagonist antihistamine combinations and methods
US4856303A (en) * 1988-07-21 1989-08-15 Whirlpool Corporation Agitator thrust spacer for automatic washer
US5225198A (en) * 1991-08-27 1993-07-06 Cygnus Therapeutic Systems Transdermal administration of short or intermediate half-life benzodiazepines
US5900250A (en) * 1992-05-13 1999-05-04 Alza Corporation Monoglyceride/lactate ester permeation enhancer for oxybutnin
DE69420419T2 (de) * 1993-09-29 1999-12-23 Alza Corp Hautpermeabilitaetserhöher bestehend aus monoglycerid/laktat estern
ATE247967T1 (de) 1998-06-09 2003-09-15 Takeda Chemical Industries Ltd Pharmazeutische kombination mit einem trizyclischen komponent und mindestens einem aus zolpidem, zopiclone und brotizolam, zur behandlung von schlafstörungen
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Also Published As

Publication number Publication date
CH535788A (de) 1973-04-15
NL170857B (nl) 1982-08-02
NL170857C (nl) 1983-01-03
NL172510B (nl) 1983-04-18
ES376689A1 (es) 1972-05-01
NL172510C (nl) 1983-09-16
FR2034999A1 (fr) 1970-12-18
AU8550075A (en) 1975-12-18
BR7017488D0 (pt) 1973-02-13
BE747493A (fr) 1970-09-17
YU34570A (en) 1979-04-30
DE2012190A1 (de) 1970-09-24
SE387641B (sv) 1976-09-13
AU8549975A (en) 1975-12-18
OA03446A (fr) 1971-03-30
NL8100081A (nl) 1981-04-29
DE2012190B2 (de) 1980-03-06
IL33859A (en) 1973-01-30
NL7003750A (nl) 1970-09-21
AU490626B2 (en) 1975-12-18
HK61677A (en) 1977-12-23
FR2034999B1 (de) 1973-07-13
PL80541B1 (pl) 1975-08-30
YU35139B (en) 1980-09-25
GB1291631A (en) 1972-10-04
US3987052A (en) 1976-10-19
DE2012190C3 (de) 1980-11-13
JPS4940239B1 (de) 1974-10-31
AU491139B2 (en) 1975-12-18
IL33859A0 (en) 1970-04-20

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