US5620981A
(en)
*
|
1995-05-03 |
1997-04-15 |
Warner-Lambert Company |
Pyrido [2,3-D]pyrimidines for inhibiting protein tyrosine kinase mediated cellular proliferation
|
IL117923A
(en)
*
|
1995-05-03 |
2000-06-01 |
Warner Lambert Co |
Anti-cancer pharmaceutical compositions containing polysubstituted pyrido¬2,3-d¾pyrimidine derivatives and certain such novel compounds
|
PT912559E
(pt)
|
1996-07-13 |
2003-03-31 |
Glaxo Group Ltd |
Compostos heterociclicos fundidos como inibidores de proteina tirosina quinase
|
HRP970371A2
(en)
|
1996-07-13 |
1998-08-31 |
Kathryn Jane Smith |
Heterocyclic compounds
|
EP0964864B1
(de)
*
|
1997-02-05 |
2008-04-09 |
Warner-Lambert Company LLC |
Pyrido (2,3-d) pyrimidine und 4-amino-primidine als inhibitoren der zellulären proliferation
|
US6498163B1
(en)
|
1997-02-05 |
2002-12-24 |
Warner-Lambert Company |
Pyrido[2,3-D]pyrimidines and 4-aminopyrimidines as inhibitors of cellular proliferation
|
EP1806348A3
(de)
*
|
1997-02-05 |
2008-01-02 |
Warner-Lambert Company LLC |
Pyrido (2,3-D)Pyrimidine als Inhibitoren der zellulären Proliferation
|
US6150359A
(en)
*
|
1997-08-20 |
2000-11-21 |
Warner-Lambert Company |
Naphthyridinones for inhibiting protein tyrosine kinase and cell cycle kinase mediated cellular proliferation
|
EP1801112A1
(de)
*
|
1998-05-26 |
2007-06-27 |
Warner-Lambert Company LLC |
Bizyklische Pyrimidine und bizyklische 3,4-Dihydropyrimidine als Hemmer der Zellvermehrung
|
CN1138778C
(zh)
*
|
1998-05-26 |
2004-02-18 |
沃尼尔·朗伯公司 |
用作细胞增殖抑制剂的二环嘧啶及二环3,4-二氢嘧啶化合物及用途
|
GB9822450D0
(en)
*
|
1998-10-14 |
1998-12-09 |
Smithkline Beecham Plc |
Medicaments
|
GB9914486D0
(en)
|
1999-06-21 |
1999-08-18 |
Smithkline Beecham Plc |
Medicaments
|
GB9917408D0
(en)
|
1999-07-23 |
1999-09-22 |
Smithkline Beecham Plc |
Compounds
|
GB9917406D0
(en)
|
1999-07-23 |
1999-09-22 |
Smithkline Beecham Plc |
Compounds
|
US7053070B2
(en)
*
|
2000-01-25 |
2006-05-30 |
Warner-Lambert Company |
Pyrido[2,3-d]pyrimidine-2,7-diamine kinase inhibitors
|
AR030044A1
(es)
*
|
2000-01-25 |
2003-08-13 |
Warner Lambert Co |
Pirido (2,3-d ) pirimidin-2,7-diaminas inhibidores de quinasas
|
MXPA03000708A
(es)
|
2000-07-26 |
2003-06-04 |
Smithkline Beecham Plc |
Aminopiperidin quinolinas y sus analogos azaisostericos con actividad antibacteriana.
|
US6518276B2
(en)
*
|
2000-08-31 |
2003-02-11 |
Syntex (U.S.A.) Llc |
7-oxo-pyridopyrimidines (II)
|
US6506749B2
(en)
|
2000-08-31 |
2003-01-14 |
Syntex (U.S.A.) Llc |
7-oxo-pyridopyrimidines (I)
|
CA2420286A1
(en)
*
|
2000-08-31 |
2002-03-07 |
F. Hoffmann-La Roche Ag |
7-oxo pyridopyrimidines as inhibitors of a cellular proliferation
|
US20020119148A1
(en)
|
2000-09-01 |
2002-08-29 |
Gerritsen Mary E. |
ErbB4 antagonists
|
ATE320255T1
(de)
|
2001-01-19 |
2006-04-15 |
Smithkline Beecham Corp |
Tie2 rezeptor-kinase-inhibitoren zur behandlung von angiogenen erkrankungen
|
GB0101577D0
(en)
|
2001-01-22 |
2001-03-07 |
Smithkline Beecham Plc |
Compounds
|
BRPI0207172B8
(pt)
|
2001-02-12 |
2021-05-25 |
Hoffmann La Roche |
pirido-pirimidinas 6-substituída, sua composição e seu uso, bem como seu intermediário
|
WO2002090360A1
(en)
*
|
2001-05-10 |
2002-11-14 |
Smithkline Beecham Corporation |
Compounds useful as kinase inhibitors for the treatment of hyperproliferative diseases
|
GB0112834D0
(en)
|
2001-05-25 |
2001-07-18 |
Smithkline Beecham Plc |
Medicaments
|
GB0112836D0
(en)
|
2001-05-25 |
2001-07-18 |
Smithkline Beecham Plc |
Medicaments
|
AU2002324450A1
(en)
*
|
2001-06-21 |
2003-01-08 |
Ariad Pharmaceuticals, Inc. |
Novel pyridopyrimidines and uses thereof
|
KR20060111716A
(ko)
|
2002-01-22 |
2006-10-27 |
워너-램버트 캄파니 엘엘씨 |
2-(피리딘-2-일아미노)-피리도[2,3-d]피리미딘-7-온
|
JP4508650B2
(ja)
|
2002-01-29 |
2010-07-21 |
グラクソ グループ リミテッド |
アミノピペリジン化合物、当該化合物の製法および当該化合物を含有する医薬組成物
|
US7312212B2
(en)
|
2002-01-29 |
2007-12-25 |
Glaxo Group Limited |
Aminopiperidine derivatives
|
WO2003074045A1
(fr)
*
|
2002-03-05 |
2003-09-12 |
Eisai Co., Ltd. |
Agent antitumoral comprenant une combinaison d'un compose heterocyclique contenant un sulfamide et d'un inhibiteur d'angiogenese
|
PA8577501A1
(es)
|
2002-07-25 |
2004-02-07 |
Warner Lambert Co |
Inhibidores de quinasas
|
CA2492112A1
(en)
|
2002-08-06 |
2004-02-19 |
F. Hoffmann-La Roche Ag |
6-alkoxy-pyrido-pyrimidines as p-38 map kinase inhibitors
|
TW200502236A
(en)
|
2003-03-28 |
2005-01-16 |
Hoffmann La Roche |
Novel pyrido[2,3-d]pyrimidin-7-carboxylic acid derivatives, their manufacture and use as pharmaceutical agents
|
AU2004289428B2
(en)
|
2003-11-13 |
2010-06-03 |
F. Hoffmann-La Roche Ag |
Hydroxyalkyl substituted pyrido-7-pyrimidin-7-ones
|
EP2260849A1
(de)
|
2004-01-21 |
2010-12-15 |
Emory University |
Zusammensetzungen und Verfahren zur Verwendung von Tyrosinkinasehemmern zur Behandlung von krankheitserregenden Infektionen
|
SG150544A1
(en)
*
|
2004-03-15 |
2009-03-30 |
Hoffmann La Roche |
Novel dichloro-phenyl-pyrido [2,3-d] pyrimidine derivatives, their manufacture and use as pharmaceutical agents
|
FR2873118B1
(fr)
*
|
2004-07-15 |
2007-11-23 |
Sanofi Synthelabo |
Derives de pyrido-pyrimidine, leur application en therapeutique
|
CN101014600A
(zh)
*
|
2004-09-21 |
2007-08-08 |
霍夫曼-拉罗奇有限公司 |
用作蛋白激酶抑制剂的6-(2-烷基-苯基)-吡啶并[2,3-d]嘧啶类
|
US20070054916A1
(en)
†
|
2004-10-01 |
2007-03-08 |
Amgen Inc. |
Aryl nitrogen-containing bicyclic compounds and methods of use
|
US7846915B2
(en)
*
|
2004-10-20 |
2010-12-07 |
Resverlogix Corporation |
Stilbenes and chalcones for the prevention and treatment of cardiovascular diseases
|
CA2593718A1
(en)
*
|
2004-12-31 |
2007-05-31 |
Gpc Biotech Ag |
Napthyridine compounds as rock inhibitors
|
FR2887882B1
(fr)
*
|
2005-07-01 |
2007-09-07 |
Sanofi Aventis Sa |
Derives de pyrido[2,3-d] pyrimidine, leur preparation, leur application en therapeutique
|
NZ566180A
(en)
|
2005-07-29 |
2011-04-29 |
Resverlogix Corp |
Pharmaceutical compositions for the prevention and treatment of complex diseases and their delivery by insertable medical devices
|
JP2009504665A
(ja)
*
|
2005-08-09 |
2009-02-05 |
アイアールエム・リミテッド・ライアビリティ・カンパニー |
タンパク質キナーゼ阻害剤としての化合物および組成物
|
US20070082920A1
(en)
*
|
2005-10-06 |
2007-04-12 |
Yongsheng Song |
NAD+-dependent DNA ligase inhibitors
|
RU2445315C2
(ru)
*
|
2005-11-22 |
2012-03-20 |
Кудос Фармасьютиклз Лимитед |
ПРОИЗВОДНЫЕ ПИРИДО-, ПИРАЗО- И ПИРИМИДО-ПИРИМИДИНА И ИХ ПРИМЕНЕНИЕ В КАЧЕСТВЕ ИНГИБИТОРОВ mTOR
|
FR2896246B1
(fr)
|
2006-01-13 |
2008-08-15 |
Sanofi Aventis Sa |
Derives de pyrido-pyrimidone, leur preparation, leur application en therapeutique.
|
AU2007211684A1
(en)
|
2006-01-31 |
2007-08-09 |
F. Hoffmann-La Roche Ag |
7H-pyrido[3,4-d]pyrimidin-8-ones, their manufacture and use as protein kinase inhibitors
|
AP2710A
(en)
|
2006-09-15 |
2013-07-30 |
Pfizer Prod Inc |
Pyrido (2, 3-D) Pyrimidinone compounds and their use as P13 inhibitors
|
JP2010509265A
(ja)
*
|
2006-11-09 |
2010-03-25 |
エフ.ホフマン−ラ ロシュ アーゲー |
キナーゼ阻害剤としての置換6−フェニル−ピリド[2,3−d]ピリミジン−7−オン誘導体及びそれの使用方法
|
FR2910813B1
(fr)
|
2006-12-28 |
2009-02-06 |
Sanofi Aventis Sa |
Nouvelle utilisation therapeutique pour le traitement des leucemies
|
US8053440B2
(en)
|
2007-02-01 |
2011-11-08 |
Resverlogix Corporation |
Compounds for the prevention and treatment of cardiovascular diseases
|
WO2008104473A2
(en)
*
|
2007-02-28 |
2008-09-04 |
F. Hoffmann-La Roche Ag |
Pyrazolopyriidine derivatives and their use as kinase inhibitors
|
WO2009100176A2
(en)
*
|
2008-02-07 |
2009-08-13 |
Abbott Laboratories |
Pharmaceutical dosage form for oral administration of tyrosine kinase inhibitor
|
US8110578B2
(en)
*
|
2008-10-27 |
2012-02-07 |
Signal Pharmaceuticals, Llc |
Pyrazino[2,3-b]pyrazine mTOR kinase inhibitors for oncology indications and diseases associated with the mTOR/PI3K/Akt pathway
|
AU2010204106B2
(en)
|
2009-01-08 |
2014-05-08 |
Resverlogix Corp. |
Compounds for the prevention and treatment of cardiovascular disease
|
NZ617779A
(en)
|
2009-03-18 |
2015-08-28 |
Resverlogix Corp |
Novel anti-inflammatory agents
|
KR20180096823A
(ko)
|
2009-04-22 |
2018-08-29 |
리스버로직스 코퍼레이션 |
신규한 소염제
|
ES2347630B1
(es)
*
|
2009-04-29 |
2011-09-08 |
Universitat Ramon Llull |
Sintesis y usos de 4-cianopentanoatos y 4-cianopentenoatos sustituidos.
|
EP2332939A1
(de)
*
|
2009-11-26 |
2011-06-15 |
Æterna Zentaris GmbH |
Neuartige Naphthyridinderivate und ihre Verwendung als Kinasehemmer
|
GB0922589D0
(en)
*
|
2009-12-23 |
2010-02-10 |
Almac Discovery Ltd |
Pharmaceutical compounds
|
US8754114B2
(en)
|
2010-12-22 |
2014-06-17 |
Incyte Corporation |
Substituted imidazopyridazines and benzimidazoles as inhibitors of FGFR3
|
GB201104267D0
(en)
|
2011-03-14 |
2011-04-27 |
Cancer Rec Tech Ltd |
Pyrrolopyridineamino derivatives
|
RS58911B1
(sr)
|
2011-11-01 |
2019-08-30 |
Resverlogix Corp |
Oralne formulacije sa trenutnim otpuštanjem za supstituisane hinazolinone
|
EP3822273B1
(de)
|
2012-06-13 |
2024-04-10 |
Incyte Holdings Corporation |
Substituierte tricyclische verbindungen als fgfr-inhibitoren
|
RS62233B1
(sr)
*
|
2012-07-11 |
2021-09-30 |
Blueprint Medicines Corp |
Inhibitori receptora fibroblast faktora rasta
|
WO2014026125A1
(en)
|
2012-08-10 |
2014-02-13 |
Incyte Corporation |
Pyrazine derivatives as fgfr inhibitors
|
GB201216018D0
(en)
|
2012-09-07 |
2012-10-24 |
Cancer Rec Tech Ltd |
Pharmacologically active compounds
|
GB201216017D0
(en)
|
2012-09-07 |
2012-10-24 |
Cancer Rec Tech Ltd |
Inhibitor compounds
|
US9073878B2
(en)
|
2012-11-21 |
2015-07-07 |
Zenith Epigenetics Corp. |
Cyclic amines as bromodomain inhibitors
|
US9765039B2
(en)
|
2012-11-21 |
2017-09-19 |
Zenith Epigenetics Ltd. |
Biaryl derivatives as bromodomain inhibitors
|
US9266892B2
(en)
|
2012-12-19 |
2016-02-23 |
Incyte Holdings Corporation |
Fused pyrazoles as FGFR inhibitors
|
JP2016507496A
(ja)
|
2012-12-21 |
2016-03-10 |
ゼニス・エピジェネティクス・コーポレイションZenith Epigenetics Corp. |
ブロモドメイン阻害剤としての新規複素環式化合物
|
CN105307657B
(zh)
*
|
2013-03-15 |
2020-07-10 |
西建卡尔有限责任公司 |
杂芳基化合物和其用途
|
TWI647220B
(zh)
|
2013-03-15 |
2019-01-11 |
美商西建卡爾有限責任公司 |
雜芳基化合物及其用途
|
UA120248C2
(uk)
|
2013-03-15 |
2019-11-11 |
Селджен Кар Ллс |
Гетероарильні сполуки та їх застосування
|
SG10201708520YA
(en)
|
2013-04-19 |
2017-12-28 |
Incyte Corp |
Bicyclic heterocycles as fgfr inhibitors
|
CN110028491B
(zh)
|
2013-10-25 |
2022-02-11 |
缆图药品公司 |
纤维母细胞生长因子受体抑制剂
|
WO2015108992A1
(en)
|
2014-01-15 |
2015-07-23 |
Blueprint Medicines Corporation |
Heterobicyclic compounds and their use as fgfr4 receptor inhibitors
|
GB201403536D0
(en)
|
2014-02-28 |
2014-04-16 |
Cancer Rec Tech Ltd |
Inhibitor compounds
|
US10851105B2
(en)
|
2014-10-22 |
2020-12-01 |
Incyte Corporation |
Bicyclic heterocycles as FGFR4 inhibitors
|
WO2016134294A1
(en)
|
2015-02-20 |
2016-08-25 |
Incyte Corporation |
Bicyclic heterocycles as fgfr4 inhibitors
|
MA41551A
(fr)
|
2015-02-20 |
2017-12-26 |
Incyte Corp |
Hétérocycles bicycliques utilisés en tant qu'inhibiteurs de fgfr4
|
MX2017010673A
(es)
|
2015-02-20 |
2018-03-21 |
Incyte Corp |
Heterociclos biciclicos como inhibidores de receptores del factor de crecimiento fibroblastico (fgfr).
|
US10111885B2
(en)
|
2015-03-13 |
2018-10-30 |
Resverlogix Corp. |
Compositions and therapeutic methods for the treatment of complement-associated diseases
|
ES2864712T3
(es)
*
|
2015-04-14 |
2021-10-14 |
Eisai R&D Man Co Ltd |
Compuesto inhibidor de FGFR4 cristalino y usos del mismo
|
CN104774183B
(zh)
*
|
2015-04-24 |
2017-10-13 |
合肥新诺华生物科技有限公司 |
一种甲酰基瑞舒伐汀钙中间体的制备方法
|
WO2018023081A1
(en)
*
|
2016-07-29 |
2018-02-01 |
Achaogen, Inc. |
6-phenylpyrido[2,3-d]pyrimidine compounds as antibacterial agents
|
AR111960A1
(es)
|
2017-05-26 |
2019-09-04 |
Incyte Corp |
Formas cristalinas de un inhibidor de fgfr y procesos para su preparación
|
GB201709840D0
(en)
|
2017-06-20 |
2017-08-02 |
Inst Of Cancer Research: Royal Cancer Hospital |
Methods and medical uses
|
WO2019208505A1
(ja)
|
2018-04-23 |
2019-10-31 |
国立大学法人京都大学 |
増殖抑制剤
|
CN112566912A
(zh)
|
2018-05-04 |
2021-03-26 |
因赛特公司 |
Fgfr抑制剂的盐
|
CN112867716A
(zh)
|
2018-05-04 |
2021-05-28 |
因赛特公司 |
Fgfr抑制剂的固体形式和其制备方法
|
WO2020185532A1
(en)
|
2019-03-08 |
2020-09-17 |
Incyte Corporation |
Methods of treating cancer with an fgfr inhibitor
|
WO2021007269A1
(en)
|
2019-07-09 |
2021-01-14 |
Incyte Corporation |
Bicyclic heterocycles as fgfr inhibitors
|
MX2022003873A
(es)
*
|
2019-10-01 |
2022-06-02 |
Goldfinch Bio Inc |
Inhibidores de 1,6-naftiridina sustituida de cdk5.
|
AU2020366006A1
(en)
|
2019-10-14 |
2022-04-21 |
Incyte Corporation |
Bicyclic heterocycles as FGFR inhibitors
|
US11566028B2
(en)
|
2019-10-16 |
2023-01-31 |
Incyte Corporation |
Bicyclic heterocycles as FGFR inhibitors
|
KR20220131900A
(ko)
|
2019-12-04 |
2022-09-29 |
인사이트 코포레이션 |
Fgfr 억제제의 유도체
|
EP4069696A1
(de)
|
2019-12-04 |
2022-10-12 |
Incyte Corporation |
Tricyclische heterocyclen als fgfr-inhibitoren
|
US11939331B2
(en)
|
2021-06-09 |
2024-03-26 |
Incyte Corporation |
Tricyclic heterocycles as FGFR inhibitors
|